CC1=NN(c2ccc(OC(F)F)c(-c3ccncc3)c2)C(=O)C1C(=O)Nc1cccc(C(C)(F)F)c1 CHEMBL4467131 IC50 0.0028 nM
CCc1c(C(O)(c2ccccc2)c2ccccc2)nn2cc(Cl)c(C(=O)Nc3ncn(CC)n3)cc12 CHEMBL4846168 IC50 0.01 nM
CCc1cnc(NC(=O)c2cc3c(nc2OC)nc(C(O)(c2ccccc2)c2ccccc2)n3CC)o1 CHEMBL4873965 IC50 0.01 nM
CCn1cnc(NC(=O)c2cc3c(nc2OC)nc(C(O)(c2ccc(OC(F)F)cc2)c2ccccc2F)n3CC)n1 CHEMBL4850648 IC50 0.01 nM
CCn1cnc(NC(=O)c2cc3c(nc2OC)nc(C(O)(c2ccccc2F)c2ccccc2F)n3CC)n1 CHEMBL4876400 IC50 0.01 nM
CCn1cnc(NC(=O)c2cc3c(nc2OC)nc(C(O)(c2cccs2)c2cccs2)n3CC)n1 CHEMBL4867121 IC50 0.01 nM
CCc1coc(NC(=O)c2cc3c(nc2OC)nc(C(O)(c2ccccc2)c2ccccc2)n3CC)n1 CHEMBL4848186 IC50 0.01 nM
CCn1c(C(O)(c2ccccc2F)c2ccccc2F)nc2nc(OC)c(-c3nnn[nH]3)cc21 CHEMBL4870590 IC50 0.01 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2nc(OC)c(-c3nnn[nH]3)cc21 CHEMBL4853889 IC50 0.01 nM
CCn1c(C(O)(c2ccccc2)c2nccs2)nc2nc(OC)c(-c3nnn[nH]3)cc21 CHEMBL4855352 IC50 0.01 nM
CCn1c(C(O)(c2ccccc2)c2cccs2)nc2nc(OC)c(-c3nnn[nH]3)cc21 CHEMBL4859117 IC50 0.01 nM
CCn1c(C(O)(c2ccccc2)c2ccccn2)nc2nc(OC)c(-c3nnn[nH]3)cc21 CHEMBL4862805 IC50 0.01 nM
CC1=NN(c2ccc(OC(F)F)c(-c3cccnc3)c2)C(=O)C1C(=O)Nc1cccc(C(C)(F)F)c1 CHEMBL4550594 IC50 0.33 nM
CCC(F)(F)c1cccc(NC(=O)C2C(=O)N(c3ccc(OC)cc3)N=C2C)c1 CHEMBL4449652 IC50 0.4626 nM
COc1ccc(N2N=C(C)C(C(=O)Nc3cccc(C(C)(F)F)c3)C2=O)cc1OC CHEMBL4535842 IC50 1.0 nM
CCn1c(C(O)(c2ccccc2)c2ncccn2)nc2nc(OC)c(-c3nnn[nH]3)cc21 CHEMBL4870878 IC50 1.0 nM
COc1ccc(N2N=C(C)C(C(=O)Nc3cccc(C(C)(F)F)c3)C2=O)cc1-c1ncco1 CHEMBL4473187 IC50 1.1 nM
COC(=O)c1cccc(N2N=C(C)C(C(=O)Nc3cccc(-c4ccco4)c3)C2=O)c1 CHEMBL4463979 IC50 2.1 nM
CC1=NN(c2ccc(OC(F)F)cc2)C(=O)C1C(=O)Nc1cccc(C(C)(F)F)c1 CHEMBL4560160 IC50 2.66 nM
COc1ccc(N2N=C(C)C(C(=O)Nc3cccc(-c4ccco4)c3)C2=O)cc1 CHEMBL4548954 IC50 3.2 nM
COc1ccc(N2N=C(C)C(C(=O)Nc3cccc(-c4ccco4)c3)C2=O)cn1 CHEMBL4476365 IC50 3.9 nM
CC1=NN(c2ccccc2)C(=O)C1C(=O)Nc1cccc(C(C)(F)F)c1 CHEMBL4466204 IC50 4.0 nM
COc1ccc(N2N=C(C)C(C(=O)Nc3cccc(C(C)(F)F)c3)C2=O)cc1 CHEMBL4539904 IC50 4.5 nM
COc1ccc(N2N=C(C)C(C(=O)Nc3cccc(C(C)(F)F)c3)C2=O)cn1 CHEMBL4437243 IC50 5.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C)cc21 CHEMBL4520185 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)O)cc21 CHEMBL4570201 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)OC)cc21 CHEMBL4515458 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(NC(C)=O)cc21 CHEMBL4546463 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC)cc21 CHEMBL4572762 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C#N)cc21 CHEMBL4582559 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCC(=O)OC)cc21 CHEMBL4570193 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCC(=O)O)cc21 CHEMBL4513710 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCCO)cc21 CHEMBL4546851 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCCCO)cc21 CHEMBL4531943 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCCNC(C)=O)cc21 CHEMBL4557579 IC50 50.0 nM
CCNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC)c2c1 CHEMBL4555596 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC(C)C)cc21 CHEMBL4529333 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCCCOC)cc21 CHEMBL4559252 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3CCOCC3)cc21 CHEMBL4531805 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC(C)O)cc21 CHEMBL4536668 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3CCNCC3)cc21 CHEMBL4539409 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCCCO)cc21 CHEMBL4534808 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCCN)cc21 CHEMBL4544796 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3CCC(O)CC3)cc21 CHEMBL4544967 IC50 50.0 nM
CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(C)c2c1 CHEMBL4585951 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC[C@H](C)O)cc21 CHEMBL4563918 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC3CCOCC3)cc21 CHEMBL4535660 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC3CCNCC3)cc21 CHEMBL4562043 IC50 50.0 nM
CCC(O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC)c2c1 CHEMBL4522480 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3CCNC3)cc21 CHEMBL4569448 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC(O)COC)cc21 CHEMBL4555909 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CCC(=O)NC)cc21 CHEMBL4550328 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2cc(F)c(C(=O)NC)cc21 CHEMBL4536338 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(O)CO)cc21 CHEMBL4483595 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CC(O)CO)cc21 CHEMBL4558467 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CNC(C)=O)cc21 CHEMBL4541244 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CNC(=O)NC)cc21 CHEMBL4524544 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC)c(F)c21 CHEMBL4552862 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)Nc3ccccc3)cc21 CHEMBL4520121 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)Nc3ccc(OC)cc3)cc21 CHEMBL4570076 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CCO)cc21 CHEMBL4544685 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccc(F)cc2F)nc2ccc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4540658 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2F)nc2ccc(C(=O)NCCO)cc21 CHEMBL4518687 IC50 50.0 nM
CNC(=O)c1ccc2nc(C(O)(c3ccccc3F)c3ccccc3F)n(C)c2c1 CHEMBL4534121 IC50 50.0 nM
Cn1c(C(O)(c2ccccc2F)c2ccccc2F)nc2ccc(C(=O)NCCO)cc21 CHEMBL4520633 IC50 50.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3F)c3ccccc3F)n(C)c2c1 CHEMBL4533463 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2F)c2ccccc2F)nc2ccc(C(=O)NCCO)cc21 CHEMBL4579343 IC50 50.0 nM
CCn1c(C(O)(c2ccc(F)cc2F)c2ccc(F)cc2F)nc2ccc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4518936 IC50 50.0 nM
CCn1c(C(O)(c2ccc(F)cc2F)c2ccc(F)cc2F)nc2ccc(C(=O)NC)cc21 CHEMBL4586620 IC50 50.0 nM
CCONC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC)c2c1 CHEMBL4540863 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CC(CO)CO)cc21 CHEMBL4521785 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CNC(=O)COC)cc21 CHEMBL4558473 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccc3cnn(C)c3c2)nc2ccc(C(=O)NC)cc21 CHEMBL4593611 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NOCCO)cc21 CHEMBL4516420 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CNC(=O)CO)cc21 CHEMBL4548538 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(S(=O)(=O)NC[C@@H](C)O)cc21 CHEMBL4513666 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2F)c2ncccc2C)nc2ccc(CCCO)cc21 CHEMBL4590325 IC50 50.0 nM
CCN1CC[C@@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)C1 CHEMBL4536753 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(N)=O)cc21 CHEMBL4552386 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2F)c2ncccc2F)nc2ccc(CCCO)cc21 CHEMBL4564753 IC50 50.0 nM
CCn1c(C(O)(c2ccc(F)cc2)c2ncccc2F)nc2ccc(CCCO)cc21 CHEMBL4520461 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(S(=O)(=O)CC)cc21 CHEMBL4538603 IC50 50.0 nM
Cn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(S(C)(=O)=O)cc21 CHEMBL4559009 IC50 50.0 nM
CCS(=O)(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(C)c2c1 CHEMBL4543510 IC50 50.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(C)c2c1 CHEMBL4582788 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)N[C@H]3CCC(=O)N(C)C3)cc21 CHEMBL4572652 IC50 50.0 nM
CN1C[C@@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(C)c3c2)CCC1=O CHEMBL4571308 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2F)c2ccccc2F)nc2ccc(C(=O)N[C@H]3CCC(=O)N(C)C3)cc21 CHEMBL4576405 IC50 50.0 nM
CCn1c(C(O)(c2ccc(F)cc2)c2ccc(F)cc2)nc2ccc(C(N)=O)cc21 CHEMBL4547185 IC50 50.0 nM
CN1C[C@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(C)c3c2)CCC1=O CHEMBL4537750 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2F)c2ccccc2F)nc2ccc(C(=O)N[C@@H]3CCC(=O)N(C)C3)cc21 CHEMBL4537676 IC50 50.0 nM
CN1C[C@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4F)c4ccccc4F)n(C)c3c2)CCC1=O CHEMBL4551379 IC50 50.0 nM
CCN1C[C@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(C)c3c2)CCC1=O CHEMBL4483466 IC50 50.0 nM
CCN1C[C@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4F)c4ccccc4F)n(C)c3c2)CCC1=O CHEMBL4587824 IC50 50.0 nM
CCN1C[C@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)CCC1=O CHEMBL4539438 IC50 50.0 nM
CCN1C[C@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4F)c4ccccc4F)n(CC)c3c2)CCC1=O CHEMBL4538445 IC50 50.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CCO)c2c1 CHEMBL4593692 IC50 50.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CCF)c2c1 CHEMBL4517398 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC[C@@H](O)CO)cc21 CHEMBL4534971 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC[C@H](O)CO)cc21 CHEMBL4569292 IC50 50.0 nM
COc1ccc2c(c1)nc(C(O)(c1ccccc1)c1ccccc1)n2C CHEMBL4538145 IC50 50.0 nM
CCOc1ccc2c(c1)nc(C(O)(c1ccccc1)c1ccccc1)n2C CHEMBL4516953 IC50 50.0 nM
CC(C)Cn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4573778 IC50 50.0 nM
Cn1ccc(NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CCO)c3c2)n1 CHEMBL4550401 IC50 50.0 nM
Cn1ccc(NC(=O)c2ccc3nc(C(O)(c4ccccc4F)c4ccccc4F)n(CCO)c3c2)n1 CHEMBL4519592 IC50 50.0 nM
Cn1cc(NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CCO)c3c2)cn1 CHEMBL4519865 IC50 50.0 nM
Cn1cc(NC(=O)c2ccc3nc(C(O)(c4ccccc4F)c4ccccc4F)n(CCO)c3c2)cn1 CHEMBL4587654 IC50 50.0 nM
CC(O)Cn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4571587 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccc(O)cc2)nc2ccc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4573798 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)Nc3cnn(CCO)c3)cc21 CHEMBL4553763 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2O)nc2ccc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4570372 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)Nc3cn(C)cn3)cc21 CHEMBL4573475 IC50 50.0 nM
CCn1cc(-c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)cn1 CHEMBL4483024 IC50 50.0 nM
CCn1cc(-c2cc3c(cc2F)nc(C(O)(c2ccccc2)c2ccccc2)n3CC)cn1 CHEMBL4556583 IC50 50.0 nM
CCc1c[nH]c(NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)n1 CHEMBL4552144 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3COC3)cc21 CHEMBL4518393 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)N[C@@H]3CCC[C@H]3O)cc21 CHEMBL4561089 IC50 50.0 nM
CCc1cccc(OCc2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)c1 CHEMBL4526130 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)N[C@@H]3CCC[C@@H](O)C3)cc21 CHEMBL4537723 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(O)C(F)(F)F)cc21 CHEMBL4539005 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(NC(=O)OC(C)(C)C)cc21 CHEMBL4530261 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(N)cc21 CHEMBL4571034 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(OC(C)=O)C(F)(F)COC(C)=O)cc21 CHEMBL4516820 IC50 50.0 nM
C=CCC1(c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)COC1 CHEMBL4522596 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2cc(OCCO)ncc21 CHEMBL4539039 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccnc(OC)c21 CHEMBL4585029 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(NC(=O)COC)cc21 CHEMBL4541774 IC50 50.0 nM
CCn1c(C(O)(c2ccc(F)cc2)c2ccc(F)cc2)nc2ccc(C(=O)NCCF)cc21 CHEMBL4580881 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC3COC3)cc21 CHEMBL4522376 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC[C@H](C)O)c(F)c21 CHEMBL4518206 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC3CCO3)cc21 CHEMBL4516381 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3(C#N)CC3)cc21 CHEMBL4581283 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2c(F)cc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4558694 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(F)C#N)cc21 CHEMBL4520680 IC50 50.0 nM
CCOC(=O)C(F)(F)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC)c2c1 CHEMBL4542511 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(F)(F)C(=O)NC[C@@H](C)O)cc21 CHEMBL4541120 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC(F)(F)C(N)=O)cc21 CHEMBL4576336 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC(C)(C)C#N)cc21 CHEMBL4570964 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2cc(F)c(C(=O)NC[C@@H](C)O)cc21 CHEMBL4552105 IC50 50.0 nM
CCN1CC(NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)CC1=O CHEMBL4523028 IC50 50.0 nM
CN1C[C@@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4F)c4ccccc4F)n(C)c3c2)CCC1=O CHEMBL4572819 IC50 50.0 nM
Cn1c(C(O)(c2ccccc2)c2ncccc2F)nc2ccc(S(N)(=O)=O)cc21 CHEMBL4592456 IC50 50.0 nM
CCN1CC(NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CCO)c3c2)CCC1=O CHEMBL4591599 IC50 50.0 nM
Cc1cccnc1C(O)(c1ccc(F)cc1)c1nc2ccc(S(N)(=O)=O)cc2n1C CHEMBL4517962 IC50 50.0 nM
Cn1c(C(O)(c2ccc(F)cc2)c2ncccc2F)nc2ccc(S(N)(=O)=O)cc21 CHEMBL4542305 IC50 50.0 nM
Cn1c(C(O)(c2ccc(F)cc2F)c2ccc(F)cc2F)nc2ccc(S(N)(=O)=O)cc21 CHEMBL4579303 IC50 50.0 nM
Cn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(S(N)(=O)=O)c(F)c21 CHEMBL4593562 IC50 50.0 nM
CCN1CC(NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(C)c3c2)CN(CC)C1=O CHEMBL4540980 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)Nc3cnn(CC(C)O)c3)cc21 CHEMBL4574195 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)Nc3ccn(CC(C)C)n3)cc21 CHEMBL4526352 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)Nc3ccn(CCOC)n3)cc21 CHEMBL4557605 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)Nc3nc(C)c[nH]3)cc21 CHEMBL4566852 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC(C)(C)O)cc21 CHEMBL4527426 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC3(O)CC3)cc21 CHEMBL4589630 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(NC(=O)c3ccccc3)cc21 CHEMBL4565699 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(NC(=O)CCOC)cc21 CHEMBL4534058 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(S(=O)(=O)CCO)cc21 CHEMBL4529090 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C3(CCO)COC3)cc21 CHEMBL4531431 IC50 50.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OC)cc21 CHEMBL4573158 IC50 250.0 nM
CCOc1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC)c2c1 CHEMBL4534890 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(Cl)cc21 CHEMBL4550758 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCC(=O)N(C)C)cc21 CHEMBL4586732 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCC(=O)NC)cc21 CHEMBL4514374 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCc3ccccc3)cc21 CHEMBL4560193 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(OCC(O)CO)cc21 CHEMBL4542160 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC(C)C)cc21 CHEMBL4582954 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCCOC)cc21 CHEMBL4588975 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCCN(C)C)cc21 CHEMBL4590064 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3CCN(C)CC3)cc21 CHEMBL4537610 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCCO)cc21 CHEMBL4574556 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)N(C)C)cc21 CHEMBL4531525 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)N3CCC3)cc21 CHEMBL4553830 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)N3CC(O)C3)cc21 CHEMBL4579888 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC(C)CO)cc21 CHEMBL4567887 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3CCC3)cc21 CHEMBL4563593 IC50 250.0 nM
CC(C)NC(=O)c1cccc(C(O)(c2ccccc2)c2nc3ccc(Cl)cc3n2C)c1 CHEMBL4586972 IC50 250.0 nM
CCn1c(C(O)(c2ccc(F)cc2)c2ccc(F)cc2)nc2ccc(C(=O)NC)cc21 CHEMBL4544350 IC50 250.0 nM
CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(C3CC3)c2c1 CHEMBL4524748 IC50 250.0 nM
CNC(=O)c1ccc2nc(C(O)(c3ccc(F)cc3)c3ccc(F)cc3)n(C)c2c1 CHEMBL4532410 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2c(F)cc(C(=O)NC)cc21 CHEMBL4584643 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccc(F)cc2F)nc2ccc(C(=O)NCCO)cc21 CHEMBL4565867 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2cc(F)c(C(=O)NCCO)cc21 CHEMBL4546730 IC50 250.0 nM
CCc1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC)c2c1 CHEMBL4543567 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C3CC3)cc21 CHEMBL4542024 IC50 250.0 nM
CCn1c(C(O)(c2ccc(F)cc2F)c2ccc(F)cc2F)nc2ccc(C(=O)NCCO)cc21 CHEMBL4550227 IC50 250.0 nM
CCn1c(C(O)(c2ccc(F)cc2)c2ccc(F)cc2)nc2ccc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4517504 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccc(F)cc3)c3ccc(F)cc3)n(C)c2c1 CHEMBL4483510 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccc(F)cc3F)c3ccc(F)cc3F)n(C)c2c1 CHEMBL4538353 IC50 250.0 nM
Cn1c(C(O)(c2ccc(F)cc2F)c2ccc(F)cc2F)nc2ccc(C(=O)NCCO)cc21 CHEMBL4589418 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CNC(=O)[C@H](C)O)cc21 CHEMBL4557219 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(CNC(=O)[C@@H](C)O)cc21 CHEMBL4585220 IC50 250.0 nM
CCn1c(C(O)(c2ccc(C)cc2)c2ncccc2C)nc2ccc(CCCO)cc21 CHEMBL4535403 IC50 250.0 nM
CCN1CC[C@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)C1 CHEMBL4559124 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C3(O)CCCCC3)cc21 CHEMBL4516038 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C3(O)CCCC3)cc21 CHEMBL4573428 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C3(O)COC3)cc21 CHEMBL4525510 IC50 250.0 nM
CCN1CCC[C@@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)C1 CHEMBL4548495 IC50 250.0 nM
CCn1c(C(O)(c2ccc(C)cc2)c2ncccc2F)nc2ccc(CCCO)cc21 CHEMBL4560526 IC50 250.0 nM
CCN1CCC[C@H](NC(=O)c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)C1 CHEMBL4567990 IC50 250.0 nM
CCn1c(C(O)(c2ccc(F)cc2F)c2ncccc2F)nc2ccc(CCCO)cc21 CHEMBL4591217 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)N[C@@H]3CCC(=O)N(C)C3)cc21 CHEMBL4518944 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC(F)(F)F)c2c1 CHEMBL4514606 IC50 250.0 nM
Cc1cccnc1C(O)(c1ccccc1)c1nc2ccc(C(=O)NC[C@@H](C)O)cc2n1C CHEMBL4543817 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ncccc3F)n(C)c2c1 CHEMBL4558768 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccc(F)cc3)c3ncccc3F)n(C)c2c1 CHEMBL4517199 IC50 250.0 nM
Cc1cccnc1C(O)(c1ccc(F)cc1)c1nc2ccc(C(=O)NC[C@@H](C)O)cc2n1C CHEMBL4519599 IC50 250.0 nM
COCCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4573037 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(-c3ccccc3)c2c1 CHEMBL4571879 IC50 250.0 nM
Cc1ccc2c(c1)nc(C(O)(c1ccccc1)c1ccccc1)n2C CHEMBL4554553 IC50 250.0 nM
Cn1c(C(O)(c2ccccc2F)c2ccccc2F)nc2ccc(C(=O)NC(CO)CO)cc21 CHEMBL4515983 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CCN(C)C)c2c1 CHEMBL4543914 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CCN)c2c1 CHEMBL4583258 IC50 250.0 nM
C[C@@H](O)CNC(=O)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC(O)CO)c2c1 CHEMBL4551659 IC50 250.0 nM
CCn1ccc(-c2ccc3nc(C(O)(c4ccccc4)c4ccccc4)n(CC)c3c2)n1 CHEMBL4522530 IC50 250.0 nM
CCn1ccc(-c2cc3c(cc2F)nc(C(O)(c2ccccc2)c2ccccc2)n3CC)n1 CHEMBL4538344 IC50 250.0 nM
CC(=O)OCC(O)(c1ccccc1)c1nc2ccc(C)cc2n1C CHEMBL4589480 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC3CC(F)(F)C3)cc21 CHEMBL4555995 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(Oc3ccccc3)cc21 CHEMBL4566279 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(COc3ccccc3)cc21 CHEMBL4590968 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2cc(OC)ncc21 CHEMBL4555658 IC50 250.0 nM
CCOc1cc2c(cn1)nc(C(O)(c1ccccc1)c1ccccc1)n2CC CHEMBL4568541 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2cnc(OCCO)cc21 CHEMBL4558484 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2cnc(OCCCO)cc21 CHEMBL4549789 IC50 250.0 nM
C=CCC(CO)(CO)c1ccc2nc(C(O)(c3ccccc3)c3ccccc3)n(CC)c2c1 CHEMBL4545132 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccnc(OCCO)c21 CHEMBL4591487 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C)c(F)c21 CHEMBL4565404 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2c(Cl)cc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4561521 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C)c(OC)c21 CHEMBL4483524 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NC[C@@H](C)O)c(OC)c21 CHEMBL4483584 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(F)(F)C#N)cc21 CHEMBL4521543 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2c(OC)cc(C(=O)NC[C@@H](C)O)cc21 CHEMBL4523068 IC50 250.0 nM
CCn1c(C(OC)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCC(F)(F)C#N)cc21 CHEMBL4538910 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2c1cnn2C CHEMBL4546194 IC50 250.0 nM
CCn1c(C(O)(c2ccccc2)c2ccccc2)nc2ccc(C(=O)NCc3ccccc3)cc21 CHEMBL4526532 IC50 250.0 nM