CSc1cccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1 CHEMBL386051 Kd 10.0 nM
CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc21 CHEMBL1241674 Kd 18.0 nM
Cc1ccc(-c2cnc(N)c(C(=O)NC3CCCCC3)n2)cc1 CHEMBL4792978 IC50 180.0 nM
C=Cc1cn2ncc(-c3ccnc(OC)c3)c2nc1NC CHEMBL4741913 IC50 190.0 nM
Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCO)CC2)n1 CHEMBL5416410 Kd 210.0 nM
CNc1nc2c(-c3ccnc(OC)c3)cnn2cc1OC CHEMBL4752199 IC50 310.0 nM
O=C(c1ccc(/C=C/c2n[nH]c3ccccc23)cc1)N1CCNCC1 CHEMBL1908397 Kd 320.0 nM
COc1cc(-c2cnn3cc(OC)c(-c4cnn(C)c4)nc23)ccn1 CHEMBL4749011 IC50 530.0 nM
CNc1nc2c(-c3ccnc(OC)c3)cnn2cc1C1CC1 CHEMBL4744988 IC50 630.0 nM
CCc1cn2ncc(-c3ccnc(OC)c3)c2nc1NC CHEMBL4741185 IC50 700.0 nM
COc1cn2ncc(-c3ccnc(OC(C)(C)C)c3)c2nc1-c1cnn(C)c1 CHEMBL4747422 IC50 800.0 nM
COc1cn2ncc(-c3ccnc(OC4CC4)c3)c2nc1-c1cnn(C)c1 CHEMBL4744618 IC50 860.0 nM
COc1cc(-n2cnc3cc(-c4cnn(C)c4)ccc32)cc(OC(F)F)c1C(=O)NC1CC1 CHEMBL5417444 IC50 860.0 nM
CCc1nc2c(-c3ccnc(OC)c3)cnn2cc1OC CHEMBL4763122 IC50 960.0 nM
CN1C(=O)[C@@H](N2CCc3cn(Cc4ccccc4)nc3C2=O)COc2ccccc21 CHEMBL4088216 pIC50 1000.0 nM
CN1C(=O)[C@@H](N2CCc3c(nn(Cc4ccccc4)c3Br)C2=O)COc2ccccc21 CHEMBL4549667 pIC50 1000.0 nM
CN1C(=O)[C@@H](N2CCc3cn(CC4CCS(=O)(=O)CC4)nc3C2=O)COc2ccccc21 CHEMBL4097778 pIC50 1000.0 nM