COC(=O)[C@H]1COCCN1CCOc1ccccc1Cc1cn(C(F)F)nc1-c1cc(Cl)nc(N)n1 CHEMBL5220685 IC50 1.0 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2OCCN2CCO[C@@H](CO)C2)n1 CHEMBL5219579 Kd 1.1 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2OCCN2CCOC[C@H]2CO)n1 CHEMBL5219830 Kd 1.4 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2OCCN2CCNC(=O)C2)n1 CHEMBL5218878 IC50 2.1 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2OCCN2CCS(=O)(=O)CC2)n1 CHEMBL5218615 Kd 2.1 nM
COC(=O)[C@@H]1COCCN1CCOc1ccccc1Cc1cn(C(F)F)nc1-c1cc(Cl)nc(N)n1 CHEMBL5218552 IC50 2.2 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2OCCN2CCOC[C@@H]2CO)n1 CHEMBL5220647 Kd 2.3 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2OCCN2CCOCC2)n1 CHEMBL5218698 Kd 3.3 nM
CC1(O)CCN(CCOc2ccccc2Cc2cn(C(F)F)nc2-c2cc(Cl)nc(N)n2)CC1 CHEMBL5218702 Kd 3.6 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2OCCN2CCO[C@H](CO)C2)n1 CHEMBL5219443 Kd 3.7 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2OCC(=O)N2CCOCC2)n1 CHEMBL5220632 Kd 4.7 nM
Cn1cc(Cc2ccccc2OCCN2CC3CC(C2)O3)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL5220895 IC50 6.7 nM
Cn1cc(Cc2ccccc2OCCN2CC3(COC3)C2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL5220347 IC50 7.8 nM
Cn1cc(Cc2ccccc2OCCN2CCOCC2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL5220723 IC50 12.3 nM
Cn1cc(Cc2ccccc2OCCN2CCNC(=O)C2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL5219922 IC50 16.9 nM
COC(=O)c1ccccc1Cc1cn(C)nc1-c1cc(Cl)nc(N)n1 CHEMBL5219530 IC50 21.0 nM
COC(=O)c1c(Cc2ccccc2)c(-c2cc(Cl)nc(N)n2)nn1C CHEMBL4878379 IC50 28.0 nM
Cn1cc(Cc2ccccc2Cl)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL5221008 IC50 64.0 nM
COc1ccccc1Cc1cn(C)nc1-c1cc(Cl)nc(N)n1 CHEMBL5220075 IC50 67.0 nM
Cc1c(Cc2cccs2)c(-c2cc(Cl)nc(N)n2)nn1C CHEMBL4848035 IC50 74.0 nM
Cn1cc(Cc2ccccc2Oc2ccccc2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL5221093 IC50 87.1 nM
Cc1c(Cc2ccccc2)c(-c2cc(Cl)nc(N)n2)nn1C CHEMBL4854762 IC50 92.0 nM
Cc1c(Cc2cccc(Cl)c2)c(-c2cc(Cl)nc(N)n2)nn1C CHEMBL4868801 IC50 107.0 nM
Nc1nc(Cl)cc(-c2nn3ccccc3c2Cc2ccccc2)n1 CHEMBL5219193 IC50 112.0 nM
Cc1c(Cc2cccc(F)c2)c(-c2cc(Cl)nc(N)n2)nn1C CHEMBL4864668 IC50 126.0 nM
Cn1cc(Cc2ccccc2F)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL4857305 IC50 132.0 nM
Cn1cc(Cc2cccs2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL4849033 IC50 141.0 nM
Cn1cc(Cc2cccc(F)c2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL4874288 IC50 225.0 nM
Cc1c(Cn2cccn2)c(-c2cc(Cl)nc(N)n2)nn1C CHEMBL4866319 IC50 325.0 nM
Cn1cc(Cc2ccc(F)cc2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL4864843 IC50 342.0 nM
COc1cccc(Cc2cn(C)nc2-c2cc(Cl)nc(N)n2)c1 CHEMBL4867202 IC50 351.0 nM
Cn1cc(Cc2cccc(Cl)c2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL5219159 IC50 389.0 nM
COC(=O)c1cccc(Cc2cn(C)nc2-c2cc(Cl)nc(N)n2)c1 CHEMBL5219933 IC50 436.0 nM
Nc1nc(Cl)cc(-c2nn(C(F)(F)F)cc2Cc2ccccc2)n1 CHEMBL5220308 IC50 469.0 nM
Cn1cc(Cc2cncs2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL4866035 IC50 576.0 nM
C[C@H]1O[C@@H](n2cnc3c(N)ncnc32)C[C@@H]1OP(=O)(O)OP(=O)(O)OP(=O)(O)O CHEMBL1162355 IC50 700.0 nM
Cn1nc(-c2cc(Cl)nc(N)n2)c(Cc2ccccc2)c1C(=O)O CHEMBL4878049 IC50 700.0 nM
Nc1nc(Cl)cc(-c2nc3ccccn3c2Cc2ccccc2)n1 CHEMBL5219011 IC50 716.0 nM
Nc1nc(Cl)cc(-c2nn(C(F)F)cc2Cc2ccccc2)n1 CHEMBL5218555 IC50 829.0 nM
Cn1cc(Cc2ccccc2)c(-c2cc(Cl)nc(N)n2)n1 CHEMBL4874934 IC50 989.0 nM