CCc1cc(-n2ccnc2)ccc1-c1ccc(-c2nnn[nH]2)cc1 CHEMBL4291042 IC50 6.1 nM
Clc1cc(-c2nnn[nH]2)ccc1-c1ccc(-n2ccnc2)cc1 CHEMBL4290485 IC50 9.2 nM
CCOc1cc([C@@H]2NC(=O)NC(c3ccccc3)=C2c2ccccc2)cc([N+](=O)[O-])c1O CHEMBL3650413 IC50 11.0 nM
CCOc1cc([C@@H]2NC(=O)N=C(c3ccccc3)C2c2ccccc2)cc([N+](=O)[O-])c1O CHEMBL3661058 IC50 11.0 nM
CCc1cc(-n2ccnc2)ccc1-c1ccc(-c2nnn[nH]2)cc1F CHEMBL4289979 IC50 11.0 nM
Cc1cc(-n2ccnc2)ccc1-c1ccc(-c2nnn[nH]2)cc1Cl CHEMBL4294439 IC50 12.0 nM
CCOc1cc(C2NC(=O)NC(c3cnn(C)c3)C2c2ccsc2)cc(C(=O)O)c1O CHEMBL3650428 IC50 13.0 nM
CCOc1cc([C@@H]2NC(=O)N=C(c3cnn(C)c3)C2c2ccsc2)cc(C(=O)O)c1O CHEMBL3661051 IC50 13.0 nM
Cc1cc(-n2ccnc2)ccc1-c1ccc(-c2nnn[nH]2)cc1 CHEMBL4283184 IC50 14.0 nM
Cc1cc(-n2ccnc2)cnc1-c1ccc(-c2nnn[nH]2)cc1F CHEMBL4289333 IC50 14.0 nM
CCOc1cc([C@@H]2NC(=O)NC(c3cccnc3)=C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3650426 IC50 16.0 nM
CCOc1cc(C2=NC(=O)NC(c3cccnc3)C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3661050 IC50 16.0 nM
Cc1cc(-n2ccnc2)cnc1-c1ccc(-c2nnn[nH]2)cc1 CHEMBL4286132 IC50 17.0 nM
CCOc1cc([C@@H]2NC(=O)NC(c3ccccc3)=C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3650415 IC50 18.0 nM
CCOc1cc([C@@H]2NC(=O)N=C(c3ccccc3)C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3661059 IC50 18.0 nM
CCOc1cc(C2NC(=O)NC(c3ccccc3)=C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3650420 IC50 19.0 nM
CCOc1cc(C2NC(=O)N=C(c3ccccc3)C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3661042 IC50 19.0 nM
Cc1cc(C(N)=O)ccc1-n1c(CCC(=O)O)ccc1-c1ccc(-n2ccnc2)cc1 CHEMBL1738699 IC50 20.0 nM
Fc1cc(-c2nnn[nH]2)ccc1-c1ccc(-n2ccnc2)cc1 CHEMBL4287066 IC50 20.0 nM
Cc1cc(-n2ccnc2)ccc1-c1ccc(C(=O)O)cc1 CHEMBL4283157 IC50 20.0 nM
Clc1cc(-n2ccnc2)cnc1-c1ccc(-c2nnn[nH]2)cc1 CHEMBL4278220 IC50 20.0 nM
c1cn(-c2ccc(-c3ccc(-c4nn[nH]n4)cc3)cc2)cn1 CHEMBL4290516 IC50 22.0 nM
Clc1cc(-n2ccnc2)ccc1-c1ccc(-c2nnn[nH]2)cc1 CHEMBL4277254 IC50 22.0 nM
Cn1cc(C2NC(=O)NC(c3ccc(C(=O)O)c(O)c3)C2c2ccsc2)cn1 CHEMBL3650432 IC50 23.0 nM
Cn1cc(C2=NC(=O)N[C@@H](c3ccc(C(=O)O)c(O)c3)C2c2ccsc2)cn1 CHEMBL3661057 IC50 23.0 nM
CCOc1cc(C2NC(=O)NC(c3cccnc3)=C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3650425 IC50 24.0 nM
CCOc1cc(C2NC(=O)N=C(c3cccnc3)C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3661044 IC50 24.0 nM
CCc1cc(-n2ccnc2C)ccc1-c1ccc(-c2nnn[nH]2)cc1 CHEMBL4286551 IC50 24.0 nM
Cc1cc(-c2nnn[nH]2)ccc1-c1ccc(-n2ccnc2)cc1 CHEMBL4279145 IC50 26.0 nM
CCOc1cc(C2NC(=O)N=C(c3cnn(C)c3)C2c2ccsc2)cc(C(=O)O)c1O CHEMBL3661049 IC50 27.0 nM
Fc1cc(-c2nnn[nH]2)ccc1-c1ncc(-n2ccnc2)cc1Cl CHEMBL4281451 IC50 27.0 nM
CCOc1cc([C@@H]2NC(=O)NC(c3cccnc3)=C2c2ccccc2)cc([N+](=O)[O-])c1O CHEMBL3650417 IC50 28.0 nM
CCOc1cc([C@@H]2NC(=O)N=C(c3cccnc3)C2c2ccccc2)cc([N+](=O)[O-])c1O CHEMBL3661061 IC50 28.0 nM
CCOc1cc(C2NC(=O)NC(c3ccccc3)=C2c2ccccc2)cc([N+](=O)[O-])c1O CHEMBL3650419 IC50 29.0 nM
CCOc1cc(C2NC(=O)N=C(c3ccccc3)C2c2ccccc2)cc([N+](=O)[O-])c1O CHEMBL3661041 IC50 29.0 nM
O=C(O)c1ccc(-c2ccc(-n3ccnc3)cc2)c(F)c1 CHEMBL4282722 IC50 29.0 nM
Cc1cc(C(=O)O)ccc1-c1ccc(-n2ccnc2)cc1 CHEMBL4285078 IC50 29.0 nM
O=C(O)c1ccc(-c2ccc(-n3ccnc3)cc2)c(Cl)c1 CHEMBL4292916 IC50 30.0 nM
c1cn(-c2ccc(-c3ccc(-c4nnn[nH]4)cc3)nc2)cn1 CHEMBL4279294 IC50 32.0 nM
CCOc1cc([C@@H]2NC(=O)NC(c3ccn(C)n3)=C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3650430 IC50 35.0 nM
CCOc1cc(C2=NC(=O)NC(c3ccn(C)n3)C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3661053 IC50 35.0 nM
Cc1cc(-n2ccnc2)cnc1-c1ccc(C(=O)O)cc1F CHEMBL4283715 IC50 36.0 nM
Cc1nccn1-c1ccc(-c2ccc(-c3nnn[nH]3)cc2Cl)cc1 CHEMBL4282612 IC50 37.0 nM
O=C(O)c1ccc(-c2ccc(-n3ccnc3)cc2)c(C(F)(F)F)c1 CHEMBL4281650 IC50 38.0 nM
Cn1ccc(C2=NC(=O)NC(c3ccc(C(=O)O)c(O)c3)C2c2ccsc2)n1 CHEMBL3661055 IC50 39.0 nM
FC(F)(F)c1cc(-c2nnn[nH]2)ccc1-c1ccc(-n2ccnc2)cc1 CHEMBL4285208 IC50 39.0 nM
CCOc1cc(C2NC(=O)NC(c3ccn(C)n3)=C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3650429 IC50 40.0 nM
CCOc1cc(C2NC(=O)N=C(c3ccn(C)n3)C2c2ccsc2)cc([N+](=O)[O-])c1O CHEMBL3661045 IC50 40.0 nM
Cc1cc(-n2ccnc2)cnc1-c1ccc(C(=O)O)cc1 CHEMBL4290901 IC50 41.0 nM
CCOc1cc(C2NC(=O)NC(c3cccnc3)=C2c2ccccc2)cc([N+](=O)[O-])c1O CHEMBL3650421 IC50 43.0 nM
CCOc1cc(C2NC(=O)N=C(c3cccnc3)C2c2ccccc2)cc([N+](=O)[O-])c1O CHEMBL3661043 IC50 43.0 nM
Cc1cc(-c2nnn[nH]2)ccc1-c1ccc(-n2ccnc2)cn1 CHEMBL4293362 IC50 44.0 nM
O=C(O)c1ccc(-c2ccc(-n3ccnc3)cc2Cl)cc1 CHEMBL4289534 IC50 59.0 nM
O=C(O)c1ccc(-c2ccc(-n3ccnc3)cc2)cc1 CHEMBL4279860 IC50 62.0 nM
CCc1cc(-n2ccnc2)cnc1-c1ccc(-c2nnn[nH]2)cc1F CHEMBL4282535 IC50 62.0 nM
CCc1cc(-n2ccnc2)cnc1-c1ccc(-c2nnn[nH]2)cc1 CHEMBL4277997 IC50 66.0 nM
CCOc1cc([C@@H]2NC(=O)NC(c3cccnc3)C2c2ccsc2)cc(C(=O)O)c1O CHEMBL3650423 IC50 67.0 nM
CCOc1cc([C@@H]2NC(=O)N=C(c3cccnc3)C2c2ccsc2)cc(C(=O)O)c1O CHEMBL3661047 IC50 67.0 nM
c1cn(-c2cnc(-c3ccc(-c4nnn[nH]4)cc3)c(C3CCCCC3)c2)cn1 CHEMBL4293137 IC50 74.0 nM
O=C(O)c1ccc(-c2ncc(-n3ccnc3)cc2Cl)cc1 CHEMBL4280261 IC50 89.0 nM
Cc1nccn1-c1ccc(-c2ccc(-c3nnn[nH]3)cc2)cc1 CHEMBL4294284 IC50 97.0 nM
CCOc1cc(C2NC(=O)NC(c3cccnc3)C2c2ccsc2)cc(C(=O)O)c1O CHEMBL3650422 IC50 150.0 nM
CCOc1cc(C2NC(=O)N=C(c3cccnc3)C2c2ccsc2)cc(C(=O)O)c1O CHEMBL3661048 IC50 150.0 nM
O=c1nc(-c2ccc(-c3ccc(-n4ccnc4)cc3)cc2)[nH]o1 CHEMBL4286678 IC50 152.0 nM
O=C(O)c1ccc(-c2ccc(-n3ccnc3)cn2)cc1 CHEMBL4291013 IC50 214.0 nM
Clc1cc(-c2nnn[nH]2)ccc1-c1ccc(-n2ccnc2)cn1 CHEMBL4282751 IC50 308.0 nM
CCOc1cc([C@H]2NC(=O)N=C(c3cnn(C)c3)C2c2ccsc2)cc(C(=O)O)c1O CHEMBL3661052 IC50 580.0 nM
Clc1cc(-c2nn[nH]n2)ccc1-c1ccc(-n2cnnc2)cc1 CHEMBL4286106 IC50 593.0 nM
Cc1cc(-c2nnn[nH]2)ccc1-c1ncc(-n2ccnc2)cc1Cl CHEMBL4285927 IC50 935.0 nM