COc1cc(NC(C)=O)c(Cl)cc1C(=O)Nc1nccs1 CHEMBL4101927 Kd 0.3 nM
Oc1cccc(Nc2nc(-c3ccc(F)cc3F)cs2)c1 CHEMBL4077165 Kd 1.0 nM
Cc1nc2ccccc2n1CC(O)Cn1c2ccccc2c2ccccc21 CHEMBL1477694 Kd 1.0 nM
Oc1cccc(Nc2nc(-c3ccc([18F])cc3F)cs2)c1 CHEMBL5176926 Kd 1.0 nM
COC(=O)c1cc(O)c(O)cc1NC(=O)C1Oc2ccccc2OC1C CHEMBL4063929 Kd 2.0 nM
OC(Cn1ccc2ccccc21)Cn1cnc2ccccc21 CHEMBL4072531 Kd 2.0 nM
CC1=NN(c2nc3ccccc3[nH]2)C(=O)C1CCC(C)C CHEMBL4100986 Kd 3.0 nM
Cn1c(=O)n(CC(O)Cn2c3ccccc3c3ccccc32)c2ccccc21 CHEMBL4075539 Kd 4.0 nM
COc1cc(SC)ccc1C(=O)Nc1cccc(C)n1 CHEMBL1463447 Kd 6.0 nM
CCCCc1nc(-c2ccc(OCCCN(CC)CC)cc2)cn1-c1ccc(Oc2ccc(Cl)cc2)cc1 CHEMBL3989929 Kd 12.7 nM
O=C(c1ccc(F)cc1)N(Cc1ccccc1)C1CCCCC1 CHEMBL4066660 Kd 15.0 nM
O=C(c1ccc([18F])cc1)N(Cc1ccccc1)C1CCCCC1 CHEMBL5200484 Kd 15.0 nM
O=C(c1ccc(Cl)cc1)N(Cc1ccccc1)C1CCCCC1 CHEMBL4075936 Ki 25.0 nM
CC1NC(NCCC[C@H](N)C(=O)O)=NC1=O CHEMBL4085254 Kd 30.0 nM
Cc1c(Cl)cccc1NC(=O)CNC(=O)c1ccccc1F CHEMBL1547178 Kd 32.0 nM
O=C(O)c1cccnc1C(=O)O CHEMBL286204 Kd 43.0 nM
CCCCc1sc(Nc2ccc(OCCCN(CC)CC)cc2)nc1-c1ccc(Oc2ccc(Cl)cc2)cc1 CHEMBL3216782 IC50 550.0 nM
CCCCc1sc(-c2ccc(OCC3CCCN(CC)C3)cc2)nc1-c1ccc(Oc2ccc(Cl)cc2)cc1 CHEMBL2205559 IC50 660.0 nM
CCCCc1sc(-c2ccc(OCCN3CCCC3)cc2)nc1-c1ccc(Oc2ccc(Cl)cc2)cc1 CHEMBL2205572 IC50 910.0 nM