C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3s2)c1 CHEMBL34896 IC50 6.0 nM
CCc1c(-c2nc(N)nc(Nc3ccc(C)cc3)n2)oc2ccccc12 CHEMBL5219455 IC50 8.4 nM
CCOc1ccc(Cl)cc1-c1cc(Nc2ccc([N+](=O)[O-])cc2)nc(N)n1 CHEMBL75167 IC50 10.0 nM
C#CCOC(=O)Nc1ccc(C)c(-c2nc3cc(Cl)ccc3s2)c1 CHEMBL35508 IC50 15.0 nM
N#CCC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3s2)c1 CHEMBL286394 IC50 15.0 nM
C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(C(F)(F)F)ccc3s2)c1 CHEMBL35388 IC50 15.0 nM
CCc1ccc(Nc2nc(N)nc(-c3oc4ccccc4c3C)n2)cc1 CHEMBL5219496 IC50 15.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(Cl)cc2)nc(N)n1 CHEMBL310136 IC50 16.0 nM
CCOc1ccc(Cl)cc1-c1cc(Nc2ccc(Cl)cc2)nc(N)n1 CHEMBL308945 IC50 17.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(C#N)cc2)nc(N)n1 CHEMBL77883 IC50 17.0 nM
Cc1ccc(Br)cc1-c1cc(Nc2ccc(Br)cc2)nc(N)n1 CHEMBL74548 IC50 18.0 nM
Nc1nc(Nc2ccc(Cl)cc2)cc(-c2cc(Cl)ccc2Cl)n1 CHEMBL307716 IC50 20.0 nM
Cc1ccc(Cl)cc1-c1cc(Nc2ccc(Cl)cc2)nc(N)n1 CHEMBL311379 IC50 22.0 nM
CCOc1ccc(Cl)cc1-c1cc(Nc2ccc3c[nH]nc3c2)nc(N)n1 CHEMBL74492 IC50 24.0 nM
N#CCC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL422579 IC50 27.0 nM
COc1ccc(Cl)cc1-c1cc(Nc2ccc(Br)cc2)nc(N)n1 CHEMBL424605 IC50 28.0 nM
CCOc1ccc(Cl)cc1-c1cc(Nc2ccc(CCO)cc2)nc(N)n1 CHEMBL74708 IC50 28.0 nM
Cc1ccc(Br)cc1-c1cc(Nc2ccc(Cl)cc2)nc(N)n1 CHEMBL74549 IC50 31.0 nM
Cc1ccc(Cl)cc1-c1cc(Nc2ccc(Br)cc2)nc(N)n1 CHEMBL73376 IC50 34.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(C(C)=O)cc2)nc(N)n1 CHEMBL72618 IC50 34.0 nM
C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL32894 IC50 35.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3s2)c1 CHEMBL284111 IC50 40.0 nM
COc1ccc(Cl)cc1-c1cc(N)nc(Nc2ccc(Cl)cc2)c1 CHEMBL193874 IC50 40.0 nM
COc1ccc(Cl)cc1-c1nc(N)nc(Nc2ccc(Cl)cc2)n1 CHEMBL195457 IC50 45.0 nM
N#CCC(=O)Nc1ccc(Cl)c(-c2nc3cc(C(F)(F)F)ccc3s2)c1 CHEMBL35564 IC50 50.0 nM
C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3ccccc3o2)c1 CHEMBL35165 IC50 50.0 nM
CCOc1ccc(Cl)cc1-c1cc(N)nc(Nc2ccc(Cl)cc2)c1 CHEMBL194604 IC50 50.0 nM
CCOc1ccc(Cl)cc1-c1cc(N)nc(Nc2ccc(C=O)cc2)c1 CHEMBL193911 IC50 50.0 nM
COc1ccc(Cl)cc1-c1cc(Nc2ccc(Cl)cc2)nc(N)n1 CHEMBL306107 IC50 54.0 nM
Cc1ccc(Cl)cc1-c1nc(N)nc(Nc2ccc(Br)cc2)n1 CHEMBL36501 IC50 60.0 nM
C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3n2C)c1 CHEMBL418604 IC50 60.0 nM
Cc1ccc(NC(=O)CC#N)cc1-c1nc2ccccc2s1 CHEMBL32731 IC50 70.0 nM
C#CCCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL32553 IC50 75.0 nM
CC#CCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL286639 IC50 75.0 nM
CCOc1ccc(Cl)cc1-c1cc(Nc2ccc(CO)cc2)nc(N)n1 CHEMBL75522 IC50 75.0 nM
COc1ccc(Cl)cc1-c1cc(Nc2ccc3c[nH]nc3c2)nc(N)n1 CHEMBL76274 IC50 80.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(/C(C)=N\O)cc2)nc(N)n1 CHEMBL72992 IC50 84.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(C(=O)NO)cc2)nc(N)n1 CHEMBL73574 IC50 88.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(B(O)O)cc2)nc(N)n1 CHEMBL74932 IC50 91.0 nM
CCOc1ccc(Cl)cc1-c1cc(N)nc(Nc2ccc(CO)cc2)c1 CHEMBL193588 IC50 99.0 nM
Cc1ccc2oc(-c3cc(NC(=O)CC#N)ccc3Cl)nc2c1 CHEMBL35006 IC50 100.0 nM
C#CCNC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL35967 IC50 100.0 nM
C#CCCC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL418404 IC50 100.0 nM
C#CCOC(=O)Nc1ccc(C)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL33773 IC50 100.0 nM
C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(C(F)(F)F)ccc3n2C)c1 CHEMBL34938 IC50 120.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccccc2)nc(N)n1 CHEMBL309911 IC50 120.0 nM
C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(C(F)(F)F)ccc3o2)c1 CHEMBL35051 IC50 140.0 nM
Cc1ccc(Cl)cc1-c1cc(Nc2ccc(C(F)(F)F)cc2)nc(N)n1 CHEMBL422414 IC50 140.0 nM
CCOc1ccc(Cl)cc1-c1nc(N)nc(Nc2ccc(Cl)cc2)n1 CHEMBL193589 IC50 140.0 nM
Cc1ccc(F)cc1-c1cc(Nc2ccc(Cl)cc2)nc(N)n1 CHEMBL73947 IC50 150.0 nM
C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3c(C)cccc3o2)c1 CHEMBL286925 IC50 160.0 nM
[N-]=[N+]=NCC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL34138 IC50 170.0 nM
C#CCOC(=O)Nc1ccc(Cl)c(-c2nc3cc(C)ccc3o2)c1 CHEMBL34585 IC50 190.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3cc(C(F)(F)F)ccc3s2)c1 CHEMBL33960 IC50 200.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(CC(=O)O)cc2)nc(N)n1 CHEMBL75714 IC50 210.0 nM
CCOc1ccc(Cl)cc1-c1cc(Nc2ccc(CCCO)cc2)nc(N)n1 CHEMBL75132 IC50 230.0 nM
COc1ccc(Cl)cc1-c1cc(N)nc(Nc2ccc(C)cc2)c1 CHEMBL193713 IC50 240.0 nM
COc1ccc(Cl)cc1-c1cc(N)nc(Nc2ccc(C=O)cc2)c1 CHEMBL194603 IC50 260.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL35582 IC50 300.0 nM
Cn1c(-c2cc(NC(=O)CC#N)ccc2Cl)nc2cc(Cl)ccc21 CHEMBL32938 IC50 300.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3ccc(C)cc3o2)c1 CHEMBL34636 IC50 400.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(CC(=O)NO)cc2)nc(N)n1 CHEMBL305915 IC50 400.0 nM
Nc1nc(Nc2ccc(Cl)cc2)cc(-c2cc(Br)ccc2O)n1 CHEMBL308275 IC50 450.0 nM
CCOc1ccc(Cl)cc1-c1cc(N)nc(Nc2ccc(C)cc2)c1 CHEMBL193910 IC50 490.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3ccccc3o2)c1 CHEMBL35458 IC50 500.0 nM
C#CCCC(=O)Nc1ccc(Cl)c(-c2nc3cc(C)ccc3o2)c1 CHEMBL33877 IC50 500.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3c(C)cccc3o2)c1 CHEMBL33823 IC50 500.0 nM
COC(=O)Nc1ccc(C)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL286185 IC50 550.0 nM
CCOc1ccc(Cl)cc1-c1cc(Nc2ccc(CC(=O)O)cc2)nc(N)n1 CHEMBL77790 IC50 580.0 nM
Cc1ccc2oc(-c3cc(NC(=O)CN=[N+]=[N-])ccc3Cl)nc2c1 CHEMBL35453 IC50 600.0 nM
Cc1ccc(Cl)cc1-c1cc(Nc2cccc(Br)c2)nc(N)n1 CHEMBL305688 IC50 610.0 nM
CCOc1ccc(Cl)cc1-c1cc(Nc2cccc([N+](=O)[O-])c2)nc(N)n1 CHEMBL73912 IC50 640.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3n2C)c1 CHEMBL290583 IC50 650.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2cccc(C#N)c2)nc(N)n1 CHEMBL74931 IC50 720.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(C(N)=O)cc2)nc(N)n1 CHEMBL308100 IC50 750.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3cc(C(F)(F)F)ccc3o2)c1 CHEMBL34886 IC50 800.0 nM
COc1ccc(Cl)cc1-c1cc(N)nc(Nc2ccc3c[nH]nc3c2)n1 CHEMBL75170 IC50 800.0 nM
CNC(=O)Nc1ccc(Cl)c(-c2nc3cc(Cl)ccc3o2)c1 CHEMBL35787 IC50 950.0 nM
CCOc1ccc(Br)cc1-c1cc(Nc2ccc(/C(C)=N\OC)cc2)nc(N)n1 CHEMBL75467 IC50 970.0 nM
COC(=O)Nc1ccc(Cl)c(-c2nc3cc(C)ccc3o2)c1 CHEMBL35001 IC50 1000.0 nM