CC1(C)CN(C(N)=O)c2cccc(F)c2N1Cc1ccccc1 CHEMBL5269095 IC50 30.0 nM
CC1(C)CN(C(N)=O)c2ccc(F)c(F)c2N1Cc1ccccc1 CHEMBL5271711 IC50 60.0 nM
CC1(C)CN(C(N)=O)c2ccc(F)c(F)c2N1Cc1ccc(COc2ccc(CO)cc2)cc1 CHEMBL5272816 IC50 100.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1ccc(COc2ccccc2)cc1 CHEMBL5270167 IC50 110.0 nM
CC1(C)CN(C(N)=O)c2ccc(F)c(F)c2N1Cc1ccc(COc2ccccc2)cc1 CHEMBL5287644 IC50 130.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1cccc(OC(F)(F)F)c1 CHEMBL5287535 IC50 140.0 nM
Cc1ccc(CN2c3ccccc3N(C(N)=O)CC2(C)C)cc1 CHEMBL5276735 IC50 170.0 nM
CC(=O)Nc1ccc(OCc2ccc(CN3c4c(ccc(F)c4F)N(C(N)=O)CC3(C)C)cc2)cc1 CHEMBL5281489 IC50 170.0 nM
CC1(C)CN(C(N)=O)c2cccc(Cl)c2N1Cc1ccccc1 CHEMBL5284620 IC50 180.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1ccc(Cl)cc1 CHEMBL5289502 IC50 190.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1cccc(Cl)c1 CHEMBL5271550 IC50 200.0 nM
CC1(C)CN(C(N)=O)c2ccc(F)c(F)c2N1Cc1ccc(COc2ccc(C(N)=O)cc2)cc1 CHEMBL5281034 IC50 200.0 nM
CC1(C)CN(C(N)=O)c2cc(F)ccc2N1Cc1ccccc1 CHEMBL5266374 IC50 240.0 nM
CC1(C)CN(C(N)=O)c2cc(F)cc(F)c2N1Cc1ccccc1 CHEMBL5283087 IC50 260.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1ccccc1 CHEMBL5280447 IC50 270.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1ccc(OC(F)(F)F)cc1 CHEMBL5284666 IC50 270.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)Cc1ccccc1Br CHEMBL36045 Ki 300.0 nM
Cc1cccc(CN2c3ccccc3N(C(N)=O)CC2(C)C)c1 CHEMBL5277889 IC50 300.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)Cc1ccccc1 CHEMBL35929 Ki 410.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1ccc(CCc2ccccc2)cc1 CHEMBL5280490 IC50 410.0 nM
CC1(C)CN(C(N)=O)c2c(F)cccc2N1Cc1ccccc1 CHEMBL5284646 IC50 500.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1cccc(CCc2ccccc2)c1 CHEMBL5282638 IC50 500.0 nM
CC(CCCCn1cnc2c1NC=NCC2O)(Cc1cccc(Br)c1)C(=O)O CHEMBL290887 Ki 640.0 nM
CC1(C)CN(C(N)=O)c2ccccc2N1Cc1ccc(OCc2ccccc2)cc1 CHEMBL5290923 IC50 740.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)Cc1cccc(Br)c1 CHEMBL38113 Ki 790.0 nM
CC(C)CC(CCCCn1cnc2c1NC=NCC2O)(CC(C)C)C(=O)O CHEMBL417506 Ki 860.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)(c1ccccc1)c1ccccc1 CHEMBL284799 Ki 920.0 nM
O=C(O)C1(CCCCn2cnc3c2NC=NCC3O)Cc2ccccc2C1 CHEMBL37713 Ki 970.0 nM