O=C(O)c1cc(CCn2cnc3c2NC=NCC3O)c2c(c1Br)CCCC2 CHEMBL346040 Ki 2.0 nM
O=C(O)c1cc(CCn2cnc3c2NC=NCC3O)c2c(c1OCc1ccccc1)CCCC2 CHEMBL157468 Ki 9.0 nM
O=C(O)c1cc2c(c(CCn3cnc4c3NC=NCC4O)c1)CCCC2 CHEMBL157949 Ki 15.0 nM
O=C(O)c1cc(CCn2cnc3c2NC=NCC3O)c2ccccc2c1 CHEMBL346360 Ki 20.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)(Cc1cccc(C(F)(F)F)c1)C(=O)O CHEMBL37273 Ki 29.0 nM
COc1c(C(=O)O)cc(CCn2cnc3c2NC=NCC3O)c2c1CCCC2 CHEMBL160174 Ki 30.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)(Cc1ccc(C(F)(F)F)cc1)C(=O)O CHEMBL289398 Ki 40.0 nM
COc1c(C(=O)O)cc2c(c1CCn1cnc3c1NC=NCC3O)CCCC2 CHEMBL157743 Ki 40.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)(Cc1ccccc1C(F)(F)F)C(=O)O CHEMBL288742 Ki 41.0 nM
O=C(O)c1c(Cl)c2c(c(CCn3cnc4c3NC=NCC4O)c1Cl)CCCC2 CHEMBL280097 Ki 50.0 nM
CC(C)Oc1c(C(=O)O)cc(CCn2cnc3c2NC=NCC3O)c2c1CCCC2 CHEMBL158023 Ki 90.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)(Cc1ccccc1)C(=O)O CHEMBL39940 Ki 170.0 nM
O=C(O)c1cc(CCn2cnc3c2NC=NCC3O)c2cccc(C(F)(F)F)c2c1 CHEMBL157426 Ki 220.0 nM
O=C(OCc1ccccc1)C(CCCCn1cnc2c1NC=NCC2O)(Cc1ccccc1C(F)(F)F)C(=O)OCc1ccccc1 CHEMBL37079 Ki 250.0 nM
CCOC(=O)c1cc(CCn2cnc3c2NC=NCC3O)c2c(c1OCc1ccccc1)CCCC2 CHEMBL158136 Ki 300.0 nM
O=C(OCc1ccccc1)c1c(Cl)c2c(c(CCn3cnc4c3NC=NCC4O)c1Cl)CCCC2 CHEMBL350676 Ki 300.0 nM
CCOC(=O)C(CCCCn1cnc2c1NC=NCC2O)(Cc1ccccc1C(F)(F)F)C(=O)OCC CHEMBL286566 Ki 360.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)C(=O)OCc1ccccc1 CHEMBL39406 Ki 360.0 nM
O=C(O)C(CCCCn1cnc2c1NC=NCC2O)Cc1ccccc1 CHEMBL35929 Ki 410.0 nM
CCOC(=O)c1c(Cl)c2c(c(CCn3cnc4c3NC=NCC4O)c1Cl)CCCC2 CHEMBL154259 Ki 500.0 nM
O=C(O)c1cccc(CCn2cnc3c2NC=NCC3O)c1 CHEMBL35524 Ki 500.0 nM
CC(CCCCn1cnc2c1NC=NCC2O)(C(=O)O)C(=O)OCc1ccccc1 CHEMBL37278 Ki 900.0 nM
O=C(O)c1cc2c(c(CCc3cnc4cncnn34)c1)CCCC2 CHEMBL2042530 IC50 900.0 nM
O=C(O)c1cc(CCn2cnc3c2NC=NCC3O)c2cc(Br)ccc2c1 CHEMBL156217 Ki 960.0 nM
CCOC(=O)c1cc(CCn2cnc3c2NC=NCC3O)c2c(c1Br)CCCC2 CHEMBL157669 Ki 1000.0 nM