NCC(O)CNC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5087702 IC50 0.25 nM
NCCCNC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5077676 IC50 0.25 nM
O=C(NC1CC(O)C1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5076950 IC50 0.25 nM
CN1CCC(NC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)C1=O CHEMBL5080571 IC50 0.25 nM
CNC(=O)C(C)NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5093385 IC50 0.25 nM
CC(C)(NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)C(N)=O CHEMBL5094500 IC50 0.25 nM
CC(CO)CNC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5081620 IC50 0.25 nM
Cc1cc(NC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)no1 CHEMBL5089988 IC50 0.25 nM
O=C(N[C@@H]1CCOC1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5080245 IC50 0.25 nM
O=C1NCCCC1NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5087854 IC50 0.25 nM
O=C1CCC(NC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)C(=O)N1 CHEMBL5093715 IC50 0.25 nM
C[C@@H](NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)C(N)=O CHEMBL5084952 IC50 0.25 nM
O=C(NCC(F)(F)F)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5076369 IC50 0.25 nM
CS(=O)(=O)CCNC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5091210 IC50 0.25 nM
O=C1NCC[C@H]1NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5086503 IC50 0.25 nM
O=C(NC1(CO)CC1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5091964 IC50 0.25 nM
CN(CC(N)=O)C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5093734 IC50 0.25 nM
O=C([C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)N(CCO)C1CC1 CHEMBL5080929 IC50 0.25 nM
NC(=O)C1(NC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)CC1 CHEMBL5082430 IC50 0.25 nM
CN(C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)C1(CO)CC1 CHEMBL5082742 IC50 0.25 nM
O=C(NC1(CCO)CC1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5085955 IC50 0.25 nM
CN(C)C(=O)CN(C)C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5085019 IC50 0.25 nM
C[C@H](NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)C(=O)N(C)C CHEMBL5082103 IC50 0.25 nM
CC(NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)C(N)=O CHEMBL5092511 IC50 0.25 nM
Cn1ccc(CNC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)n1 CHEMBL5081854 IC50 0.25 nM
CC1(O)CN(C(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)C1 CHEMBL5092615 IC50 0.25 nM
CC(NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)c1ccn(C)n1 CHEMBL5093063 IC50 0.25 nM
O=C(NCc1ccn[nH]1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5080254 IC50 0.25 nM
C[C@H](O)CNC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5094600 IC50 0.25 nM
O=C(OC1CN(C(=O)C2CC(c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc34)C2)C1)C1CCOCC1 CHEMBL5074357 IC50 0.25 nM
O=C(NCCCO)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5094544 IC50 0.25 nM
O=C([C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)N1CCOC(O)C1 CHEMBL5081065 IC50 0.25 nM
CCN(CCO)C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5070651 IC50 0.25 nM
CC(O)CN(CCO)C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5076729 IC50 0.25 nM
O=C1CC[C@H](NC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)C1 CHEMBL5070196 IC50 0.25 nM
C[C@H](CO)N(C)C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5090454 IC50 0.25 nM
NC(=O)[C@H](CO)NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5088723 IC50 0.25 nM
O=C([C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)N1CCC[C@@H](O)C1 CHEMBL5080712 IC50 0.25 nM
NC(=O)[C@H]1CCCN1C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5079082 IC50 0.25 nM
O=C1NCC[C@@H]1NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5083779 IC50 0.25 nM
O=C(N[C@@H](CO)C(F)(F)F)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5091162 IC50 0.25 nM
O=C(N[C@H](CO)C(F)(F)F)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5084244 IC50 0.25 nM
CC(O)CNC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5087672 IC50 0.25 nM
O=C(NCc1cnoc1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5094530 IC50 0.25 nM
NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5078098 IC50 0.25 nM
O=C(NCc1nnco1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5082503 IC50 0.25 nM
Cc1nnc(CNC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)o1 CHEMBL5086262 IC50 0.25 nM
C[C@@H](O)CNC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5089404 IC50 0.25 nM
O=C(NC[C@H](O)C(F)(F)F)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5082754 IC50 0.25 nM
O=C(NC[C@@H](O)C(F)(F)F)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5089252 IC50 0.25 nM
O=C(N[C@H]1CC[C@H]1O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5089734 IC50 0.25 nM
O=C(NCC1(O)CC1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5083060 IC50 0.25 nM
O=C(N[C@H]1CCC[C@@H]1O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5083782 IC50 0.25 nM
O=C(NCC1(O)COC1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5090323 IC50 0.25 nM
O=C1OCC[C@@H]1NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5085628 IC50 0.25 nM
CC(C#N)(CO)NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5088084 IC50 0.25 nM
O=C([C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)N1CCC[C@@H]1CO CHEMBL5076966 IC50 0.25 nM
CC(CO)N(C)C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5083679 IC50 0.25 nM
C#CC(CO)NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5089805 IC50 0.25 nM
CC1(NC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)CCNC1=O CHEMBL5089445 IC50 0.25 nM
Cn1ncc(CNC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)n1 CHEMBL5092967 IC50 0.25 nM
O=C(NC(CO)C1CC1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5084737 IC50 0.25 nM
O=C(NC1(CO)CC(F)(F)C1)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5088072 IC50 0.25 nM
CCC(CO)NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5080687 IC50 0.25 nM
CC[C@@H](CO)NC(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5080173 IC50 0.25 nM
O=C([C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)N1CC[C@H]1CO CHEMBL5076370 IC50 0.25 nM
C[C@]1(NC(=O)[C@H]2C[C@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)C[C@@H](O)C1 CHEMBL5081016 IC50 0.25 nM
CC1(CO)CCN1C(=O)[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5079543 IC50 0.25 nM
O=C([C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)N1CCOC[C@@H]1CO CHEMBL5094728 IC50 0.25 nM
O=C(NCCO)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5081802 IC50 0.25 nM
O=C(NCC(F)F)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5091263 IC50 0.25 nM
O=C(NC1(CO)CCC1)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5087679 IC50 0.25 nM
CC(CO)(CO)NC(=O)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5089581 IC50 0.25 nM
CC(C)(CO)NC(=O)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5092759 IC50 0.25 nM
O=C(NCC(F)(F)F)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5079825 IC50 0.25 nM
Cc1ccn(CCNC(=O)[C@H]2C[C@@H](c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc43)C2)n1 CHEMBL5078818 IC50 0.25 nM
C[C@@H](CO)NC(=O)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5082896 IC50 0.25 nM
O=C(NC(CO)(CO)CO)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5085568 IC50 0.25 nM
O=C(N[C@@H](CO)C(F)F)[C@H]1C[C@@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5094254 IC50 0.25 nM
NC(=O)C1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5093949 IC50 0.25 nM
O=C(NCCO)C1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(C(F)(F)F)cc23)C1 CHEMBL5089131 IC50 0.25 nM
Cn1cnc(CNC(=O)C2(C)CC(c3c(-c4ccc(F)cc4)[nH]c4c(F)cc(F)cc34)C2)c1 CHEMBL5076913 IC50 0.25 nM
CC1(C(=O)NCCO)CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5082777 IC50 0.25 nM
CC1(C(=O)N[C@H]2CCNC2=O)CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5094558 IC50 0.25 nM
O=C(CN[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)NCO CHEMBL5083568 IC50 0.25 nM
CNC(=O)CN[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5084440 IC50 0.25 nM
C[C@@H](CO)NC(=O)N[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5074928 IC50 0.25 nM
O=C(NCCO)C1CC(Cc2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5081514 IC50 0.25 nM
O=C(NCCO)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5072040 IC50 0.25 nM
O=C(NCC(F)F)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5078102 IC50 0.25 nM
CC(C)(CO)NC(=O)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5087178 IC50 0.25 nM
O=C(NCc1cnco1)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5075363 IC50 0.25 nM
C[C@H](CO)NC(=O)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5086493 IC50 0.25 nM
NC(=O)CNC(=O)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5086512 IC50 0.25 nM
CC(CO)NC(=O)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5077067 IC50 0.25 nM
C[C@@H](CO)NC(=O)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5089466 IC50 0.25 nM
O=C(NC1CC1)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5074794 IC50 0.25 nM
O=C(N[C@@H]1CCNC1=O)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5087125 IC50 0.25 nM
COCC(C)NC(=O)O[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5075957 IC50 0.25 nM
CNC(=O)NC[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5082028 IC50 0.25 nM
C[C@H](NCC1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1)C(=O)N(C)C CHEMBL5085829 IC50 0.25 nM
CN(C)C(=O)CNCC1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5076194 IC50 0.25 nM
CNC(=O)C(C)NCC1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5078049 IC50 0.25 nM
NC(=O)C(CO)NCC1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5073628 IC50 0.25 nM
O=C(CNC[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1)NC1CC1 CHEMBL5093579 IC50 0.25 nM
CON(C)C(=O)CNC[C@H]1C[C@H](c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc32)C1 CHEMBL5088027 IC50 0.25 nM
O=C(CC1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1)NC1(CO)CC1 CHEMBL5094381 IC50 0.25 nM
CCNC(=O)N1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5089277 IC50 0.25 nM
O=C(NCC(F)F)N1CC(c2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C1 CHEMBL5088139 IC50 0.25 nM
O=C(CCc1cc(-c2c(F)cc(F)cc2Cl)[nH]c1-c1ccc(Cl)cc1)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5398930 pIC50 0.5012 nM
CC(C)(C)c1cc(CCC(=O)N[C@@H]2C(=O)NC[C@H]2O)c(-c2ccc(C(F)(F)F)cc2)[nH]1 CHEMBL5419825 pIC50 1.585 nM
O=C(CCc1c(-c2ccc(Cl)cc2)[nH]c(C2(C(F)(F)F)CC2)c1F)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5429041 pIC50 1.995 nM
O=C(CCc1cc(C2(C(F)(F)F)CC2)[nH]c1-c1ccc(C(F)(F)F)cc1)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5399768 pIC50 2.512 nM
O=C(CCc1cc(C2(C(F)(F)F)CC2)[nH]c1-c1ccc(Cl)cc1)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5420173 pIC50 2.512 nM
O=C(CCc1cc(-c2c(F)cc(F)cc2F)[nH]c1-c1ccc(Cl)cc1)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5408105 pIC50 3.162 nM
O=C1C[C@H](NC(=O)CCc2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C(=O)N1 CHEMBL5082079 IC50 250.0 nM
CC1C[C@H](NC(=O)CCc2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C(=O)N1 CHEMBL5079943 IC50 250.0 nM
O=C(CCc1c(-c2ccc(F)cc2)[nH]c2c(F)cc(F)cc12)N[C@H]1C(=O)NC[C@@H]1O CHEMBL5077076 IC50 250.0 nM
O=C(CCc1c(-c2ccc(F)cc2)[nH]c2c(F)cc(F)cc12)N[C@@H]1CCNC1=O CHEMBL5080704 IC50 250.0 nM
CC1(NC(=O)CCc2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)CCNC1=O CHEMBL5093005 IC50 250.0 nM
O=C(CCc1c(-c2ccc(F)cc2)[nH]c2c(F)cc(F)cc12)N[C@H]1C(=O)NC[C@H]1O CHEMBL5090167 IC50 250.0 nM
O=C1C[C@@H](NC(=O)CCc2c(-c3ccc(F)cc3)[nH]c3c(F)cc(F)cc23)C(=O)N1 CHEMBL5087107 IC50 250.0 nM
Cc1cc(F)c2[nH]c(-c3ccc(F)cc3)c(CCC(=O)N[C@H]3CCNC3=O)c2c1 CHEMBL5093288 IC50 250.0 nM
O=C(CCc1c(-c2ccc(F)cc2)[nH]c2c(F)cc(Cl)cc12)N[C@@H]1CCNC1=O CHEMBL5089322 IC50 250.0 nM
COc1cc(F)cc2c(CCC(=O)N[C@H]3CCNC3=O)c(-c3ccc(F)cc3)[nH]c12 CHEMBL5073518 IC50 250.0 nM
O=C(CCc1c(-c2ccc(F)cc2)[nH]c2ccc(F)cc12)N[C@@H]1CCNC1=O CHEMBL5083803 IC50 250.0 nM
CN(C(=O)CCc1c(-c2ccc(F)cc2)[nH]c2ccc(F)cc12)C1CCNC1=O CHEMBL5079167 IC50 250.0 nM
O=C(CCc1c(-c2ccc(F)cc2)[nH]c2ccc(OCc3ccccc3)cc12)N[C@H]1CCNC1=O CHEMBL5079077 IC50 250.0 nM
O=C(CCc1c(-c2ccc(F)cc2)[nH]c2c(F)c(F)ccc12)N[C@H]1CCNC1=O CHEMBL5078982 IC50 250.0 nM
O=C(CCc1c(-c2ccccc2)[nH]c2c(F)cccc12)N[C@H]1CCNC1=O CHEMBL5075252 IC50 250.0 nM
O=C(CCc1c(-c2ccccc2)[nH]c2c(C3CCOC3)cccc12)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5088583 IC50 250.0 nM
CC(C)(O)c1cccc2c(CCC(=O)N[C@@H]3C(=O)NC[C@H]3O)c(-c3ccccc3)[nH]c12 CHEMBL5091559 IC50 250.0 nM
C=C(C)c1cccc2c(CCC(=O)N[C@@H]3C(=O)NC[C@H]3O)c(-c3ccccc3)[nH]c12 CHEMBL5079789 IC50 250.0 nM
CC(C)c1cccc2c(CCC(=O)N[C@@H]3C(=O)NC[C@H]3O)c(-c3ccccc3)[nH]c12 CHEMBL5079185 IC50 250.0 nM
C[C@@H](Cc1c(-c2ccc(F)cc2)[nH]c2c(F)cc(F)cc12)C(=O)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5076398 IC50 250.0 nM
O=C(CCc1c(-c2ccccc2)[nH]c2c(C(F)(F)F)cccc12)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5077603 IC50 250.0 nM
Cc1cc(F)ccc1-c1[nH]c2ccccc2c1CCC(=O)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5079014 IC50 250.0 nM
O=C(CCc1c(-c2cc(F)cc(F)c2)[nH]c2ccccc12)N[C@@H]1C(=O)NC[C@H]1O CHEMBL5083381 IC50 250.0 nM
O=C(CCc1c(-c2ccc(F)cc2)[nH]c2ccccc12)N[C@H]1C(=O)NC[C@H]1O CHEMBL5082577 IC50 250.0 nM