O=C(NCCCCc1ccccc1)n1c(=O)oc2cccc(-c3ccccc3)c21 CHEMBL3741996 IC50 0.8 nM
Nc1nc2ccccc2n1C(=O)NCCCCc1ccccc1 CHEMBL4093029 IC50 0.9 nM
Cc1nc2ccccc2n1C(=O)NCCCCc1ccccc1 CHEMBL4103207 IC50 1.0 nM
O=C(NCCCCc1ccccc1)n1nnc2ncccc21 CHEMBL4084295 IC50 1.3 nM
O=C(NCCCCc1ccccc1)n1nnc2ccccc21 CHEMBL4092051 IC50 2.1 nM
CCCCCCNC(=O)n1nnc2ncccc21 CHEMBL4062592 IC50 2.2 nM
CCCCCCNC(=O)n1c(N)nc2ccccc21 CHEMBL4065362 IC50 2.4 nM
O=C(NCCCCc1ccccc1)N1C(=O)c2ccccc2C1=O CHEMBL4075447 IC50 2.4 nM
O=C(NCCCCc1ccccc1)n1cnc2ccccc21 CHEMBL4100744 IC50 2.5 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccc([N+](=O)[O-])cc21 CHEMBL3741624 IC50 3.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc([N+](=O)[O-])ccc21 CHEMBL3741606 IC50 3.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cnccc21 CHEMBL4580541 IC50 3.0 nM
CCCCCCNC(=O)n1nnc2ccccc21 CHEMBL4071239 IC50 4.1 nM
O=C(NCCCCc1ccccc1)n1ncc2ccccc21 CHEMBL4075028 IC50 4.7 nM
O=C(NCCCCc1ccccc1)n1c(-c2ccc(Cl)cc2)coc1=O CHEMBL4742096 IC50 5.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccncc21 CHEMBL4592427 IC50 6.0 nM
CCCCCCNC(=O)n1cnc2ccccc21 CHEMBL66205 IC50 6.6 nM
CCCCCCNC(=O)N1C(=O)c2ccccc2C1=O CHEMBL4089655 IC50 7.0 nM
Cc1ccc(CNC(=O)n2c(N)nc3ccccc32)cc1 CHEMBL4096883 IC50 7.0 nM
CCCCCCNC(=O)n1cc(F)c(=O)n(C(=O)OCC(C)C)c1=O CHEMBL2333055 IC50 7.7 nM
Cc1cccc(CNC(=O)n2cnc3ccccc32)c1 CHEMBL4076230 IC50 8.3 nM
Cc1cccc(CNC(=O)n2c(N)nc3ccccc32)c1 CHEMBL4101140 IC50 8.5 nM
CCCCCCNC(=O)n1ncc2ccccc21 CHEMBL4095461 IC50 9.9 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccc(F)cc21 CHEMBL3741732 IC50 12.0 nM
CCCCCCNC(=O)n1cc(Cl)c(=O)n(C(=O)OCC(C)C)c1=O CHEMBL4777626 IC50 12.8 nM
COc1nc2ccccc2n1C(=O)NCCCCc1ccccc1 CHEMBL4094489 IC50 13.9 nM
O=C(c1ccc(Cl)cc1)c1ccc2c(c1)oc(=O)n2C(=O)NCCCCc1ccccc1 CHEMBL3740891 IC50 14.0 nM
CCCCCCNC(=O)n1cc(Br)c(=O)n(C(=O)OCC(C)C)c1=O CHEMBL3900210 IC50 14.0 nM
CCCCCCNC(=O)n1nc(C)cc1C(F)(F)F CHEMBL4754069 IC50 14.0 nM
Cc1ccc(CNC(=O)n2cnc3ccccc32)cc1 CHEMBL4075846 IC50 14.8 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccc(Cl)cc21 CHEMBL3740027 IC50 15.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(Cl)c(Cl)cc21 CHEMBL3739503 IC50 18.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2c(Br)cccc21 CHEMBL3739921 IC50 18.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccc(C(F)(F)F)cc21 CHEMBL3741563 IC50 18.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2ccncc2)oc1=O CHEMBL4777275 IC50 18.0 nM
CCCc1ccc(CNC(=O)n2c(=O)oc3ccccc32)cc1 CHEMBL3741565 IC50 19.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(C(F)(F)F)ccc21 CHEMBL3741712 IC50 20.0 nM
CCCCCCNC(=O)n1cc(F)c(=O)[nH]c1=O CHEMBL460499 IC50 20.7 nM
O=C(NCCCCc1ccccc1)n1c(=O)n(C(=O)NCCCCc2ccccc2)c2ccccc21 CHEMBL4099796 IC50 21.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccc(Br)cc21 CHEMBL3740148 IC50 22.0 nM
O=C(NCc1ccccc1)n1cnc2ccccc21 CHEMBL4076865 IC50 22.5 nM
Cc1cccc2c1oc(=O)n2C(=O)NCCCCc1ccccc1 CHEMBL3742201 IC50 23.0 nM
O=C(c1ccccc1)c1ccc2oc(=O)n(C(=O)NCCCCc3ccccc3)c2c1 CHEMBL3739808 IC50 24.0 nM
CN1CCC(c2cc3oc(=O)n(C(=O)NCCCCc4ccccc4)c3cc2F)CC1 CHEMBL4461146 IC50 24.0 nM
Cc1ccc(CCCCNC(=O)n2c(=O)oc3ccccc32)cc1 CHEMBL3739956 IC50 25.0 nM
CCCCCNC(=O)n1c(-c2ccccc2)coc1=O CHEMBL4753638 IC50 25.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2ccccn2)oc1=O CHEMBL4783041 IC50 25.0 nM
O=C(c1ccccc1)c1ccc2c(c1)oc(=O)n2C(=O)NCCCCc1ccccc1 CHEMBL3740970 IC50 29.0 nM
Nc1nc2ccccc2n1C(=O)NCc1ccccc1 CHEMBL4075647 IC50 29.3 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(F)ccc21 CHEMBL3740687 IC50 31.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(Br)ccc21 CHEMBL3740254 IC50 31.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2cnccn2)oc1=O CHEMBL4753408 IC50 32.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(Cl)ccc21 CHEMBL3741153 IC50 33.0 nM
CCCCCCNC(=O)n1cc(Br)c(=O)[nH]c1=O CHEMBL2333042 IC50 35.0 nM
O=C(NCCCCc1cccs1)n1c(=O)oc2ccccc21 CHEMBL3739472 IC50 37.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2cnc3ccccc3n2)oc1=O CHEMBL4740634 IC50 37.0 nM
CCCCCNC(=O)n1cc(-c2ccccc2)oc1=O CHEMBL4755627 IC50 39.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccc(-c3ccccc3)cc21 CHEMBL3740071 IC50 42.0 nM
Cc1oc(=O)n(C(=O)NCCCCc2ccccc2)c1-c1ccccc1 CHEMBL4778065 IC50 42.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2cscn2)oc1=O CHEMBL4794165 IC50 44.0 nM
O=C(NCCCCCCc1ccccc1)n1c(=O)oc2ccccc21 CHEMBL3741977 IC50 51.0 nM
CN1CCN(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)C(=O)C1 CHEMBL4541371 IC50 52.0 nM
CCCCCCCCCCCCCCC[C@@H](O)[C@H](CO)NC(=O)CBr CHEMBL4753296 IC50 52.0 nM
O=C(NCCCCCc1ccccc1)n1c(=O)oc2ccccc21 CHEMBL3742353 IC50 54.0 nM
O=C(NCCCc1ccccc1)n1c(=O)oc2ccccc21 CHEMBL3741093 IC50 55.0 nM
Cc1ccccc1CNC(=O)n1cnc2ccccc21 CHEMBL4077199 IC50 55.9 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccc(-c3ccc(F)cc3)cc21 CHEMBL3739598 IC50 56.0 nM
CCN1CCN(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4483813 IC50 56.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2nccs2)oc1=O CHEMBL4757770 IC50 59.0 nM
CCCCCNC(=O)n1c(=O)oc2cc(-c3ccc(F)cc3)ccc21 CHEMBL4515178 IC50 60.0 nM
COc1ccc(CCCCNC(=O)n2c(=O)oc3ccccc32)cc1 CHEMBL3741168 IC50 63.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2ccccc21 CHEMBL3742230 IC50 64.0 nM
CC(=O)N1CCC(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4471764 IC50 64.0 nM
O=C(NCCSCc1ccccc1)n1c(=O)oc2ccccc21 CHEMBL3740184 IC50 65.0 nM
Cc1ccc2c(c1)oc(=O)n2C(=O)NCCCCc1ccccc1 CHEMBL3740949 IC50 66.0 nM
COc1ccc(-c2ccc3oc(=O)n(C(=O)NCCCCc4ccccc4)c3c2)cc1 CHEMBL3741885 IC50 67.0 nM
COc1ccc(-c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)cc1 CHEMBL3742292 IC50 67.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(C3CCOCC3)ccc21 CHEMBL4471752 IC50 68.0 nM
Cc1ccccc1CNC(=O)n1c(N)nc2ccccc21 CHEMBL4090927 IC50 68.4 nM
Cc1c(-c2ccccc2)oc(=O)n1C(=O)NCCCCc1ccccc1 CHEMBL4780394 IC50 69.0 nM
O=C(NCCCCc1ccccc1)n1c(-c2ccccc2)coc1=O CHEMBL4764724 IC50 70.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2cccnc2)oc1=O CHEMBL4744299 IC50 70.0 nM
O=C(NCCCCc1ccc2ccccc2c1)n1c(=O)oc2ccccc21 CHEMBL3741632 IC50 71.0 nM
O=C(NCCCCc1ccc(F)cc1)n1c(=O)oc2ccccc21 CHEMBL3740594 IC50 75.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(-c3ccc(F)cc3)ccc21 CHEMBL3740827 IC50 79.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(N3CCCCC3)ccc21 CHEMBL4550439 IC50 80.0 nM
COc1cc(-c2cn(C(=O)NCCCCc3ccccc3)c(=O)o2)ccc1F CHEMBL4758195 IC50 80.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2ccc(Cl)cc2)oc1=O CHEMBL4783116 IC50 83.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(-c3ccccc3)ccc21 CHEMBL3740470 IC50 84.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(C3CCCCC3)ccc21 CHEMBL4454206 IC50 89.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2ccccc2)oc1=O CHEMBL4763533 IC50 90.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2c(-c3ccccc3)cccc21 CHEMBL3740884 IC50 91.0 nM
CCN1CCC(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4476617 IC50 92.0 nM
CN1CCN(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1=O CHEMBL4540417 IC50 92.0 nM
Cn1nc(-c2cn(C(=O)NCCCCc3ccccc3)c(=O)o2)c2ccccc21 CHEMBL4739945 IC50 92.0 nM
CC(C)N1CCC(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4474218 IC50 94.0 nM
CN1CCC(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccc(F)cc2)CC1 CHEMBL4590615 IC50 94.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(C3CCN(CC(F)F)CC3)ccc21 CHEMBL4584283 IC50 95.0 nM
CN1CCC(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1=O CHEMBL4455260 IC50 105.0 nM
CN1CCN(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4515811 IC50 116.0 nM
Cc1ccc2oc(=O)n(C(=O)NCCCCc3ccccc3)c2c1 CHEMBL3741313 IC50 117.0 nM
CC(C)CN1CCC(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4522065 IC50 120.0 nM
O=C(NCCc1ccccc1)n1c(=O)oc2ccccc21 CHEMBL3742264 IC50 121.0 nM
CC(C)CN1CCN(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4560335 IC50 127.0 nM
CN1CCC(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4534076 IC50 129.0 nM
CCCCCNC(=O)n1cc(-c2ccc(F)cc2C2CCN(C)CC2)oc1=O CHEMBL4746157 IC50 129.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(C3CCNCC3)ccc21 CHEMBL4443783 IC50 134.0 nM
CN1CCC(c2cccc(-c3cn(C(=O)NCCCCc4ccccc4)c(=O)o3)c2)CC1 CHEMBL4795472 IC50 153.0 nM
CCCCCCNC(=O)n1cc(-c2ccccc2)c(=O)[nH]c1=O CHEMBL2333040 IC50 155.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(N3CCS(=O)(=O)CC3)ccc21 CHEMBL4571748 IC50 160.0 nM
CC(C)CNC(=O)n1c(=O)oc2cc(C3CCN(C)CC3)ccc21 CHEMBL4451058 IC50 166.0 nM
COc1ccccc1-c1cn(C(=O)NCCCCc2ccccc2)c(=O)o1 CHEMBL4779233 IC50 177.0 nM
O=C(NCCCCc1ccccc1)n1cc(-c2ccc(F)cc2)oc1=O CHEMBL4757876 IC50 185.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(N3CCOCC3)ccc21 CHEMBL4587060 IC50 192.0 nM
CC(C)N1CCN(c2ccc3c(c2)oc(=O)n3C(=O)NCCCCc2ccccc2)CC1 CHEMBL4475836 IC50 211.0 nM
CN1CCC(c2ccc3c(c2)oc(=O)n3C(=O)NCCOCc2ccccc2)CC1 CHEMBL4439693 IC50 215.0 nM
O=C(NCCCCc1ccccc1)n1c2c(oc1=O)CCNC2 CHEMBL4545769 IC50 247.0 nM
CCCCCCNC(=O)n1cc(Br)c(=O)n(C(=O)OC)c1=O CHEMBL3957935 IC50 270.0 nM
CC(=O)N1CCc2oc(=O)n(C(=O)NCCCCc3ccccc3)c2C1 CHEMBL4448689 IC50 293.0 nM
CC(C)CNC(=O)n1c(=O)oc2ccc(C3CCN(C)CC3)cc21 CHEMBL4514724 IC50 295.0 nM
C[C@H]1[C@H](NC(=O)OCCCCC2CCCCC2)C(=O)N1Oc1ccccc1 CHEMBL4100592 IC50 300.0 nM
O=C(NCCCCc1ccc([N+](=O)[O-])cc1)n1c(=O)oc2ccccc21 CHEMBL3741541 IC50 312.0 nM
CN1CCC(c2cc(F)ccc2-c2cn(C(=O)NCCCCc3ccccc3)c(=O)o2)CC1 CHEMBL4778785 IC50 337.0 nM
O=C(NCCCCc1ccccc1)n1c2c(oc1=O)CNCC2 CHEMBL4459931 IC50 340.0 nM
COc1cccc(-c2cn(C(=O)NCCCCc3ccccc3)c(=O)o2)c1 CHEMBL4759179 IC50 341.0 nM
CN1CCC(c2cc(-c3cn(C(=O)NCCCCc4ccccc4)c(=O)o3)ccc2F)CC1 CHEMBL4796255 IC50 341.0 nM
O=C(NCCCCc1ccccc1)n1c(=O)oc2cc(N3CCNCC3)ccc21 CHEMBL4450809 IC50 363.0 nM
CCCCc1ccc(COC(=O)N[C@H]2CNC2=O)cc1 CHEMBL3770896 IC50 390.0 nM
CCCCCNC(=O)n1c(=O)oc2cc(C3CCN(C)CC3)ccc21 CHEMBL4460936 IC50 396.0 nM
COc1ccc(-c2cn(C(=O)NCCCCc3ccccc3)c(=O)o2)cc1 CHEMBL4776116 IC50 400.0 nM
O=C(NCCCCc1ccccc1)n1c2c(oc1=O)CCN(Cc1ccccc1)C2 CHEMBL4451320 IC50 436.0 nM
CN1CCc2oc(=O)n(C(=O)NCCCCc3ccccc3)c2C1 CHEMBL4543388 IC50 516.0 nM
CC(C)CNC(=O)n1c(=O)oc2c(C3CCN(C)CC3)cccc21 CHEMBL4535309 IC50 535.0 nM
O=C(NCCOCc1ccccc1)n1c(=O)oc2ccccc21 CHEMBL3742284 IC50 649.0 nM
CCCCCCCCCCCCCC(=O)N[C@H](C)[C@@H](O)c1ccccc1 CHEMBL429926 IC50 1000.0 nM