O=C(CF)CNC(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc2c(F)cccc12 CHEMBL4581663 IC50 15.0 nM
O=C(CF)CNC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(F)c2ccccc12 CHEMBL4546760 IC50 60.0 nM
O=C(CF)CNC(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc2ccccc12 CHEMBL4520267 IC50 73.0 nM
CN(CC(=O)CF)C(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc2ccccc12 CHEMBL4520585 IC50 130.0 nM
O=C(CF)CNC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnnc2ccccc12 CHEMBL4553669 IC50 190.0 nM
O=C(CF)CNC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccnc2ccccc12 CHEMBL4567870 IC50 270.0 nM
Cc1sc2nc(C3CCCCC3)nc(SCC(=O)N3CC(=O)Nc4ccccc43)c2c1C CHEMBL1496397 IC50 316.0 nM
O=C(CF)CNC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1cccc2ccccc12 CHEMBL4469737 IC50 360.0 nM
CCc1ccc2c(c1)C(c1ccc([N+](=O)[O-])cc1)=NNC(c1ccccc1)=N2 CHEMBL1391013 IC50 399.0 nM
COc1ccc(C(C)=O)cc1CSc1nc2ccccc2c(=O)n1-c1cccc(C)c1 CHEMBL1538079 IC50 502.0 nM
Cc1nn(Cc2c(F)c(F)c(F)c(F)c2F)c(C)c1NC(=O)c1ccc(COc2cc(Cl)ccc2Cl)cc1 CHEMBL1427626 IC50 532.0 nM
O=C(NCc1ccc(Br)cc1)Nc1ncc([N+](=O)[O-])s1 CHEMBL4560825 IC50 610.0 nM
O=C(N[C@@H](Cc1ccccc1)C(=O)CCl)OCc1ccccc1 CHEMBL303579 IC50 630.0 nM
O=C(NCc1cnc2ccccc2c1)Nc1ncc([N+](=O)[O-])s1 CHEMBL4534968 IC50 640.0 nM
CCn1nc(/C=C/c2ccccc2)nc2c(=O)n(C)c(=O)nc1-2 CHEMBL599924 IC50 653.0 nM
COc1cccc(C(=O)N[C@@H](Cc2ccccc2)C(=O)NCC(=O)CF)c1 CHEMBL4578571 IC50 720.0 nM
O=C(NCc1cccc(Cl)c1)Nc1ncc([N+](=O)[O-])s1 CHEMBL4483776 IC50 730.0 nM
O=C(NCc1cccnc1)Nc1ncc([N+](=O)[O-])s1 CHEMBL4575072 IC50 850.0 nM
O=C(Nc1cccc(Cl)c1N1CCCC1)c1cccc(-c2cc3ccccc3oc2=O)c1 CHEMBL1494802 IC50 870.0 nM
O=C(NCc1ccc(C(F)(F)F)cc1)Nc1ncc([N+](=O)[O-])s1 CHEMBL4592322 IC50 880.0 nM
O=C(CF)CNC(=O)[C@H](Cc1ccccc1)NC(=O)Cc1ccccc1 CHEMBL4574173 IC50 920.0 nM
O=C(CF)CNC(=O)[C@H](Cc1ccccc1)NC(=O)c1cnccn1 CHEMBL4579064 IC50 950.0 nM
O=C(NCc1cccc(Br)c1)Nc1ncc([N+](=O)[O-])s1 CHEMBL4555963 IC50 950.0 nM
O=C(NCc1ccc(-c2ccccc2)cc1)Nc1ncc([N+](=O)[O-])s1 CHEMBL4542508 IC50 1000.0 nM
