C[C@@H](n1c(=O)[nH]c2ccc(C3=NC(=O)[C@](C)(c4ccc(C(F)(F)F)nc4)N3)cc21)C(C)(C)C CHEMBL5418011 IC50 8.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=NC(=O)[C@](C)(c4cnc(C(F)(F)F)nc4)N3)cc21)C(C)(C)C CHEMBL5410549 IC50 9.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=N[C@@](Cc4ccccc4)(c4cnc(C(F)(F)F)nc4)NC3=O)cc21)C(C)(C)C CHEMBL5398949 IC50 13.0 nM
Cc1ncc([C@]2(C)NC(c3ccc4[nH]c(=O)n([C@H](C)C(C)(C)C)c4c3)=NC2=O)cn1 CHEMBL5433694 IC50 24.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=N[C@@](C)(c4cnc(C(F)(F)F)nc4)NC3=O)cc21)C(C)(C)C CHEMBL5417333 IC50 24.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=N[C@@](c4cccnc4)(c4nnc[nH]4)NC3=O)cc21)C(C)(C)C CHEMBL5418761 IC50 26.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=C[C@@](C)(c4cnc(C(F)(F)F)nc4)OC3=O)cc21)C(C)(C)C CHEMBL5410730 IC50 28.0 nM
Cc1ccc([C@]2(C)NC(c3ccc4[nH]c(=O)n([C@H](C)C(C)(C)C)c4c3)=NC2=O)cn1 CHEMBL5437335 IC50 29.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=NC(=O)[C@](C)(c4ccc(C(F)(F)F)cn4)N3)cc21)C(C)(C)C CHEMBL5402041 IC50 30.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=N[C@](c4ccc(Cl)nc4)(c4ccccn4)NC3=O)cc21)C(C)(C)C CHEMBL5419626 IC50 39.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=N[C@]4(CCc5cc(Br)ccc54)NC3=O)cc21)C(C)(C)C CHEMBL5415169 IC50 53.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=N[C@@](C)(c4cc5ccccc5[nH]4)NC3=O)cc21)C(C)(C)C CHEMBL5413800 IC50 55.0 nM
Cc1[nH]c2cc(NC(=O)c3ccc4[nH]c(=O)n([C@H](C)C(C)(C)C)c4c3)ccc2c1C CHEMBL5432994 IC50 60.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=NC(=O)[C@](C)(c4ccc(Cl)cn4)N3)cc21)C(C)(C)C CHEMBL5404438 IC50 66.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=N[C@@](C)(c4ccc(Cl)cn4)NC3=O)cc21)C(C)(C)C CHEMBL5434394 IC50 69.0 nM
C[C@H](NC(=O)c1ccc2[nH]c(=O)n([C@H](C)C(C)(C)C)c2c1)c1cnc(C(F)(F)F)nc1 CHEMBL5410194 IC50 70.0 nM
C[C@H](NC(=O)c1ccc2[nH]c(=O)n([C@H](C)C(C)(C)C)c2c1)c1cnc(Cl)nc1 CHEMBL5405463 IC50 76.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=NC(=O)[C@](C)(c4ncc(Cl)cn4)N3)cc21)C(C)(C)C CHEMBL5420091 IC50 82.0 nM
Cc1ccc([C@H](C)NC(=O)c2ccc3[nH]c(=O)n([C@H](C)C(C)(C)C)c3c2)nc1 CHEMBL5399837 IC50 93.0 nM
Cc1ccc([C@]2(C)NC(c3ccc4[nH]c(=O)n([C@H](C)C(C)(C)C)c4c3)=NC2=O)nc1 CHEMBL5431279 IC50 96.0 nM
C[C@H](NC(=O)c1ccc2[nH]c(=O)n([C@H](C)C(C)(C)C)c2c1)c1ccc(Br)cn1 CHEMBL5406719 IC50 100.0 nM
Cc1ncc([C@H](C)NC(=O)c2ccc3[nH]c(=O)n([C@H](C)C(C)(C)C)c3c2)cn1 CHEMBL5407611 IC50 120.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=NC(c4ccc(Cl)cn4)(c4ccc(Cl)cn4)NC3=O)cc21)C(C)(C)C CHEMBL5432221 IC50 200.0 nM
C[C@H](NC(=O)c1ccc2[nH]c(=O)n([C@H](C)C(C)(C)C)c2c1)c1ccc(Cl)cn1 CHEMBL5413528 IC50 230.0 nM
C[C@H](NC(=O)c1ccc2[nH]c(=O)n([C@H](C)C(C)(C)C)c2c1)c1ccc(C(F)(F)F)cn1 CHEMBL5417424 IC50 230.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C(=O)O)cc21)C(C)(C)C CHEMBL5430292 IC50 260.0 nM
C[C@H](NC(=O)c1ccc2[nH]c(=O)n([C@H](C)C(C)(C)C)c2c1)c1ccc(Cl)cc1 CHEMBL5397909 IC50 290.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=N[C@@](C)(c4ccc5nccn5c4)NC3=O)cc21)C(C)(C)C CHEMBL5402738 IC50 370.0 nM
C[C@H](NC(=O)c1ccc2[nH]c(=O)n([C@H](C)C(C)(C)C)c2c1)c1ncc(Cl)cn1 CHEMBL5439813 IC50 430.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=NC(=O)[C@@](C)(c4ccc(Cl)cn4)N3)cc21)C(C)(C)C CHEMBL5403458 IC50 510.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=NC(=O)[C@](C)(c4ccccc4)N3)cc21)C(C)(C)C CHEMBL5424059 IC50 600.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C(=O)NCc3ccc(Cl)cc3)cc21)C(C)(C)C CHEMBL5413076 IC50 610.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C(=O)Nc3ccccc3)cc21)C(C)(C)C CHEMBL5432738 IC50 820.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C(=O)NC(C)(C)c3ccc(Cl)cc3)cc21)C(C)(C)C CHEMBL5401480 IC50 840.0 nM
C[C@H](NC(=O)c1ccc2[nH]c(=O)n([C@H](C)C(C)(C)C)c2c1)c1cnc(Cl)cn1 CHEMBL5414987 IC50 890.0 nM
C[C@@H](n1c(=O)[nH]c2ccc(C3=NOC(C)(c4ccccc4)N3)cc21)C(C)(C)C CHEMBL5436441 IC50 900.0 nM