C[C@H]1CCN(S(=O)(=O)c2cc(NC(=O)CN3C(=O)N[C@@](C)(C4CC4)C3=O)ccc2Br)C1 CHEMBL4449894 pKd 15.85 nM
CCCOc1ccn2c(C(C)=O)cc(-c3ccccc3S(C)(=O)=O)c2c1 CHEMBL3739699 Kd 60.0 nM
Cn1cc(CCn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)cc2)cn1 CHEMBL4296718 Kd 109.0 nM
CC(=O)c1cc(-c2ccccc2S(C)(=O)=O)c2cc(CNC(=O)OC(C)(C)C)ccn12 CHEMBL3770199 IC50 160.0 nM
Cc1cc(-c2nc3ccccc3n2CC2CCOCC2)cn(C)c1=O CHEMBL4456922 pIC50 316.23 nM
Cc1cn(Cn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)c(F)c2)nn1 CHEMBL3415185 IC50 450.0 nM
Cc1cc(-c2nc3ccccc3n2C(C)C2CCOCC2)cn(C)c1=O CHEMBL4466159 pIC50 501.19 nM
CC(=O)c1cc(-c2ccccc2S(C)(=O)=O)c2cc(Oc3ccccc3)ccn12 CHEMBL3770277 IC50 550.0 nM
COc1ccn2c(C(C)=O)cc(-c3ccccc3S(C)(=O)=O)c2c1 CHEMBL3770214 IC50 580.0 nM
Cc1cn(CCn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)cc2)nn1 CHEMBL3415182 IC50 600.0 nM
CC(=O)c1cc(-c2ccccc2S(C)(=O)=O)c2ccccn12 CHEMBL3770847 IC50 720.0 nM
CN(C)C(=O)c1cccc(-c2cn(C)c(=O)c3[nH]ccc23)c1 CHEMBL4436408 IC50 880.0 nM
CC(=O)c1cc(-c2ccccc2S(C)(=O)=O)c2cc(C)ccn12 CHEMBL3770738 IC50 890.0 nM
CC(=O)c1cc(-c2ccccc2CO)c2cc(C)ccn12 CHEMBL3771216 IC50 1000.0 nM