CCCOc1ccn2c(C(C)=O)cc(-c3ccccc3S(C)(=O)=O)c2c1 CHEMBL3739699 Kd 60.0 nM
Cn1cc(CCn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)cc2)cn1 CHEMBL4296718 Kd 170.0 nM
CC(=O)c1cc(-c2ccccc2CO)c2cc(C)ccn12 CHEMBL3771216 IC50 370.0 nM
CCCOc1cc(OCCCCN(C)C)cc(Oc2cc3c(cc2NS(=O)(=O)c2ccc(OC)c(OC)c2)n(C)c(=O)n3C)c1 CHEMBL3774575 Kd 400.0 nM
COc1ccn2c(C(C)=O)cc(-c3ccccc3CO)c2c1 CHEMBL3770155 IC50 410.0 nM
CC(=O)c1cc(-c2ccccc2CO)c2cc(N3CCOCC3)ccn12 CHEMBL3770449 IC50 540.0 nM
CC(=O)c1cc(-c2ccccc2CO)c2cc(Oc3ccccc3)ccn12 CHEMBL3770493 IC50 610.0 nM
CC(=O)c1cc(-c2ccccc2S(C)(=O)=O)c2cc(CNC(=O)OC(C)(C)C)ccn12 CHEMBL3770199 IC50 670.0 nM
Cc1cn(Cn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)cc2F)nn1 CHEMBL3415184 IC50 770.0 nM
Cc1cn(Cn2cnc(-c3cnn(C)c3)c2-c2ccc(C#N)c(F)c2)nn1 CHEMBL3415185 IC50 790.0 nM
COc1ccn2c(C(C)=O)cc(-c3ccccc3S(C)(=O)=O)c2c1 CHEMBL3770214 IC50 820.0 nM
CC(=O)c1cc(-c2ccccc2S(C)(=O)=O)c2cc(Oc3ccccc3)ccn12 CHEMBL3770277 IC50 840.0 nM
CN1C[C@H](Nc2cnn(C)c(=O)c2Br)C[C@H](c2ccccc2)C1 CHEMBL4069412 Ki 840.0 nM
CC(=O)c1cc(-c2ccccc2CO)c2ccccn12 CHEMBL3770112 IC50 1000.0 nM
Cc1cc2c(C3=CCOCC3)cnc(NC3CCN(C(=O)C(F)(F)CN)CC3)c2[nH]c1=O CHEMBL4864027 pKi 1000.0 nM