CCCN1CCC(C(=O)N(C)Cc2cc(Cl)cc(-c3cc(-c4cc(C(F)(F)F)ccc4I)c(C#N)c(=O)[nH]3)c2O)CC1 CHEMBL4793552 Kd 34.0 nM
CCCN1CCC(C(=O)N(C)Cc2cc(Cl)cc(-c3cc(-c4cc(C(F)(F)F)ccc4Cl)c(C#N)c(=O)[nH]3)c2O)CC1 CHEMBL234358 Kd 37.0 nM
CC(=O)N1CCC(C(=O)NCc2cc(Cl)cc(-c3cc(-c4cc(C(F)(F)F)ccc4Cl)c(C#N)c(=O)[nH]3)c2O)CC1 CHEMBL233848 Kd 48.0 nM
CCCC(=O)N1CCC(C(=O)N(C)Cc2cc(Cl)cc(-c3cc(-c4cc(C(F)(F)F)ccc4Cl)c(C#N)c(=O)[nH]3)c2O)CC1 CHEMBL272921 Kd 60.0 nM
COCC(=O)N1CCC(C(=O)N(C)Cc2cc(Cl)cc(-c3cc(-c4cc(C(F)(F)F)ccc4Cl)c(C#N)c(=O)[nH]3)c2O)CC1 CHEMBL234330 Kd 64.0 nM
CN(Cc1cc(Cl)cc(-c2cc(-c3cc(C(F)(F)F)ccc3Cl)c(C#N)c(=O)[nH]2)c1O)C(=O)CCN1CCOCC1 CHEMBL234040 Kd 76.0 nM
CC(=O)N1CCC(C(=O)N(C)Cc2cc(Cl)cc(-c3cc(-c4cc(C(F)(F)F)ccc4Cl)c(C#N)c(=O)[nH]3)c2O)CC1 CHEMBL232404 Kd 86.0 nM
CN(Cc1cc(Cl)cc(-c2cc(-c3cc(C(F)(F)F)ccc3Cl)c(C#N)c(=O)[nH]2)c1O)C(=O)C1CCN(C(=O)C2CCCCC2)CC1 CHEMBL234421 Kd 100.0 nM
COC1CCC(C(=O)N(C)Cc2cc(Cl)cc(-c3cc(-c4cc(C(F)(F)F)ccc4Cl)c(C#N)c(=O)[nH]3)c2O)CC1 CHEMBL234041 Kd 200.0 nM
CCCCCN1CCC(C(=O)N(C)Cc2cc(Cl)cc(-c3cc(-c4cc(C(F)(F)F)ccc4Cl)c(C#N)c(=O)[nH]3)c2O)CC1 CHEMBL396856 Kd 220.0 nM
Cc1cccc(Nc2nc3nonc3nc2N/N=C/c2ccc(-c3cccc(C(=O)O)c3)o2)c1C CHEMBL4637348 Kd 240.0 nM
CN(Cc1cc(Cl)cc(-c2cc(-c3cc(C(F)(F)F)ccc3Cl)c(C#N)c(=O)[nH]2)c1O)C(=O)C1CCN(C(=O)OC(C)(C)C)CC1 CHEMBL394046 Kd 260.0 nM
CN(Cc1cc(Cl)cc(-c2cc(-c3cc(C(F)(F)F)ccc3Cl)c(C#N)c(=O)[nH]2)c1O)C(=O)CCN1CCCC1 CHEMBL428195 Kd 440.0 nM
N#Cc1c(-c2cc(C(F)(F)F)ccc2Cl)cc(-c2cc(Br)ccc2O)[nH]c1=O CHEMBL236619 Kd 490.0 nM
N#Cc1c(-c2cc(Cl)ccc2Cl)cc(-c2cc(C3CCCC3)ccc2O)[nH]c1=O CHEMBL232402 Kd 510.0 nM
N#Cc1c(-c2cc(C(F)(F)F)ccc2Cl)cc(-c2cc(Cl)ccc2O)[nH]c1=O CHEMBL236620 Kd 520.0 nM
CN(Cc1cc(Cl)cc(-c2cc(-c3cc(C(F)(F)F)ccc3Cl)c(C#N)c(=O)[nH]2)c1O)C(=O)C1CCNCC1 CHEMBL392286 Kd 530.0 nM
CN(Cc1cc(Cl)cc(-c2cc(-c3cc(C(F)(F)F)ccc3Cl)c(C#N)c(=O)[nH]2)c1O)C(=O)C1CCCCC1 CHEMBL392285 Kd 620.0 nM
Cc1ccc(-c2cc(-c3cc(Br)ccc3O)[nH]c(=O)c2C#N)c(C)c1 CHEMBL391681 Kd 700.0 nM
N#Cc1c(-c2cc(Cl)ccc2Cl)cc(-c2cc(-c3ccccc3)ccc2O)[nH]c1=O CHEMBL391106 Kd 700.0 nM
N#Cc1c(-c2cc(Cl)ccc2Cl)cc(-c2cc(Br)ccc2O)[nH]c1=O CHEMBL393124 Kd 800.0 nM
N#Cc1c(-c2cc(C(F)(F)F)ccc2Cl)cc(-c2cc(Cl)cc(CNC(=O)C3CCCCC3)c2O)[nH]c1=O CHEMBL234608 Kd 880.0 nM