CCCOc1cc(OCCCCN(C)C)cc(Oc2cc3c(cc2NS(=O)(=O)c2ccc(OC)c(OC)c2)n(C)c(=O)n3C)c1 CHEMBL3774575 Kd 27.0 nM
CN1C[C@H](Nc2cnn(C)c(=O)c2Br)C[C@H](c2ccccc2)C1 CHEMBL4069412 Ki 100.0 nM
C[C@H]1CCN(S(=O)(=O)c2cc(NC(=O)CN3C(=O)N[C@@](C)(C4CC4)C3=O)ccc2Br)C1 CHEMBL4449894 pKd 125.89 nM
COc1cc(C#N)ccc1S(=O)(=O)Nc1ccc2c(c1)cc(C)c(=O)n2C CHEMBL3752151 IC50 140.0 nM
COc1cc2c(cc1NS(=O)(=O)c1ccc(C#N)cc1OC)cc(C)c(=O)n2C CHEMBL4103077 IC50 190.0 nM
Cc1cc2cc(NS(=O)(=O)c3ccc(C#N)cc3)ccc2n(C)c1=O CHEMBL4102050 IC50 260.0 nM
COc1cc2c(cc1NS(=O)(=O)c1ccc(C#N)cc1)cc(C)c(=O)n2C CHEMBL4059962 IC50 280.0 nM
COc1cc2c(cc1NS(=O)(=O)c1ccccc1)cc(C)c(=O)n2C CHEMBL4087315 IC50 590.0 nM
Cc1cncc(-c2cnc(N[C@@H]3CCN(C)C[C@H]3OCC3CCS(=O)(=O)CC3)c3[nH]c(=O)c(C)cc23)c1 CHEMBL3590408 pKi 794.33 nM
Cn1c(=O)ccc2cc(NS(=O)(=O)c3ccc(C#N)cc3)ccc21 CHEMBL4076056 IC50 1000.0 nM
COc1ccccc1C(=O)Nc1cc2c(cc1N1CCCC1)n(C)c(=O)n2C CHEMBL3356143 Kd 1000.0 nM