COc1ccc([C@@H]2Sc3cc(OC)ccc3N(CCN(C)C)C(=O)[C@@H]2OC(C)=O)cc1 CHEMBL319525 Ki 42.0 nM
C=CC[C@H]1C(=O)N(CCN(C)C)c2ccccc2C[C@H]1c1ccc(OC)cc1 CHEMBL163740 Kd 52.0 nM
COc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CCN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL167935 Kd 75.0 nM
COc1ccc([C@@H]2Sc3cc(OC)ccc3N(CCN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL96454 Ki 85.0 nM
COc1ccc([C@@H]2Cc3c(ccc(Br)c3OC)N(CCN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL165086 Kd 120.0 nM
COc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CCN)C(=O)[C@@H]2OC(C)=O)cc1 CHEMBL168066 Kd 120.0 nM
COc1ccc([C@@H]2Cc3c(ccc(Br)c3OC)N(CCN(C)C)C(=O)[C@@H]2OC(C)=O)cc1 CHEMBL353757 Kd 120.0 nM
COc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CCN(C)C(C)C)C(=O)[C@@H]2C)cc1 CHEMBL353566 Kd 130.0 nM
CNCCN1C(=O)[C@H](OC(C)=O)[C@H](c2ccc(OC)cc2)Cc2c1cccc2C(F)(F)F CHEMBL164399 Kd 160.0 nM
COc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CCN(C)CCCCc3ccccc3)C(=O)[C@@H]2OC(C)=O)cc1 CHEMBL163771 Kd 220.0 nM
CCC[C@H]1C(=O)N(CCN(C)C)c2ccccc2C[C@H]1c1ccc(OC)cc1 CHEMBL350321 Kd 250.0 nM
COc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CC(C)N(C)C)C(=O)[C@@H]2C)cc1 CHEMBL349753 Kd 320.0 nM
COc1ccc([C@@H]2Sc3ccccc3N(CCN(C)C)C(=O)[C@@H]2OC(C)=O)cc1 CHEMBL23 Ki 380.0 nM
COc1ccc([C@@H]2Cc3c(OC)cccc3N(CCN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL168099 Kd 400.0 nM
C=CCN(C)CCN1C(=O)[C@H](OC(C)=O)[C@H](c2ccc(OC)cc2)Cc2c1cccc2C(F)(F)F CHEMBL164134 Kd 420.0 nM
CCCN(C)CCN1C(=O)[C@H](OC(C)=O)[C@H](c2ccc(OC)cc2)Cc2c1cccc2C(F)(F)F CHEMBL165444 Kd 520.0 nM
COc1ccc([C@@H]2Sc3ccccc3N(CCN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL262509 Ki 540.0 nM
COc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(C(C)CN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL167987 Kd 540.0 nM
CNc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CCN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL355684 Kd 570.0 nM
CC[C@H]1C(=O)N(CCN(C)C)c2cccc(C(F)(F)F)c2C[C@H]1c1ccc(OC)cc1 CHEMBL349193 Kd 600.0 nM
COc1ccc([C@@H]2Cc3ccccc3N(CCN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL98189 Ki 650.0 nM
COc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CCN(C)C)C(=O)[C@@H]2O)cc1 CHEMBL351235 Kd 660.0 nM
COc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CC[N+](C)(C)C)C(=O)[C@@H]2C)cc1 CHEMBL352750 Kd 840.0 nM
CCc1ccc([C@@H]2Cc3c(cccc3C(F)(F)F)N(CCN(C)C)C(=O)[C@@H]2C)cc1 CHEMBL165049 Kd 1000.0 nM