CCOc1ccc(-n2nc3c(N4CC[C@H](N)C4)nnc(C)c3c2C)cc1 CHEMBL1801177 IC50 10.0 nM
CCOc1ccc(-n2nc3c(N4CCCC4)nnc(C)c3c2C)cc1 CHEMBL1801206 IC50 22.0 nM
CCOc1ccc(-n2nc3c(N4CCC4)nnc(C)c3c2C)cc1 CHEMBL1801207 IC50 59.0 nM
CCOc1ccc(-n2nc3c(N4CC[C@@H](OC)C4)nnc(C)c3c2C)cc1 CHEMBL1801179 IC50 79.0 nM
CCOc1ccc(-n2nc3c(N4CC[C@@H](F)C4)nnc(C)c3c2C)cc1 CHEMBL1801186 IC50 85.0 nM
CC(C)C[C@H](CN)CC(=O)O CHEMBL1059 Ki 99.0 nM
CCOc1ccc(-n2nc3c(N4CC(OC)C4)nnc(C)c3c2C)cc1 CHEMBL1801180 IC50 126.0 nM
CCOc1ccc(-n2nc3c(N(C)C)nnc(C)c3c2C)cc1 CHEMBL1801205 IC50 158.0 nM
CCOc1ccc(-n2nc3c(N4CC(OC)C4)nnc(C)c3c2C)c(F)c1 CHEMBL1801192 IC50 200.0 nM
Cc1nnc(N2CCCC2)c2nn(-c3ccc(OC(C)C)cc3)c(C)c12 CHEMBL1801183 IC50 316.0 nM
CCOc1ccc(-n2nc3c(N4CCC(O)CC4)nnc(C)c3c2C)cc1 CHEMBL1801176 IC50 398.0 nM
Cc1nnc(N2CCCC2)c2nn(-c3ccc(OCC(F)(F)F)cc3)c(C)c12 CHEMBL1801182 IC50 398.0 nM
CCOc1ccc(-n2nc3c(NC)nnc(C)c3c2C)cc1 CHEMBL1801208 IC50 537.0 nM
Cc1nnc(N2CCCC2)c2nn(-c3ccc(Cl)cc3Cl)c(C)c12 CHEMBL1801184 IC50 631.0 nM
Cc1nnc(N2CC[C@@H](F)C2)c2nn(-c3ccc(OCC(F)(F)F)cc3)c(C)c12 CHEMBL1801188 IC50 631.0 nM
Cc1nnc(N2CCCC2)c2nn(-c3ccc(Cl)cc3OC(F)(F)F)c(C)c12 CHEMBL1801185 IC50 794.0 nM
CCOc1ccc(-n2nc3c(N4CCC(F)(F)C4)nnc(C)c3c2C)cc1 CHEMBL1801187 IC50 794.0 nM
CCOc1ccc(-n2nc3c(N4CCNCC4)nnc(C)c3c2C)cc1 CHEMBL1801211 IC50 1000.0 nM
CCOc1ccc(-n2nc3c(N4CCCNCC4)nnc(C)c3c2C)cc1 CHEMBL1801213 IC50 1000.0 nM