CN(C)CCNC1=CC(=O)c2nc(-c3cc(F)ccc3F)oc2C1=O CHEMBL5271462 IC50 23.0 nM
Cc1nc2c(s1)C(=O)C=C(NCCN(C)C)C2=O CHEMBL5288122 IC50 23.0 nM
O=C1C(SCCO)=C(SCCO)C(=O)c2ccccc21 CHEMBL429095 IC50 56.9 nM
CC(NC1=C(Cl)C(=O)c2cccnc2C1=O)c1cn(-c2ccc(CO)cc2)nn1 CHEMBL5423941 IC50 60.0 nM
O=C1C(Cl)=C(NCCN2CCOCC2)C(=O)c2ncccc21 CHEMBL337173 Ki 89.0 nM
Cc1ccc(Cn2cc(CNC3=C(Cl)C(=O)c4cccnc4C3=O)nn2)cc1 CHEMBL4521092 IC50 90.0 nM
O=C1C=CC(=O)c2c1ccc1c2c(=O)oc2c3ccccc3ccc12 CHEMBL4093222 IC50 100.0 nM
CCc1nc2c(o1)C(O)=C/C(=N\CCN(C)C)C2=O CHEMBL199359 IC50 130.0 nM
CCc1nc2c(o1)C(=O)C(NCCN(C)C)=CC2=O CHEMBL382593 IC50 130.0 nM
Cc1nc2c(s1)C(O)=C/C(=N\CCN(C)C)C2=O CHEMBL373195 IC50 150.0 nM
CC1=C(NCCN(C)C)C(=O)c2nc(C)sc2C1=O CHEMBL1765351 IC50 170.0 nM
N#Cc1cccc(Cn2cc(CNC3=C(Cl)C(=O)c4cccnc4C3=O)nn2)c1 CHEMBL4566962 IC50 210.0 nM
CN(C)CC/N=C1\C=C(O)c2oc(-c3ccccc3)nc2C1=O CHEMBL199360 IC50 230.0 nM
CN(C)CC/N=C1\C=C(O)c2nc(-c3ccccc3)oc2C1=O CHEMBL200805 IC50 230.0 nM
CCN(CC)c1ccc2c(c1)oc(=O)c1c3c(ccc12)C(=O)C=CC3=O CHEMBL4066424 IC50 300.0 nM
O=C1C=CC(=O)c2c1ccc1c2c(=O)oc2ccc(F)cc21 CHEMBL4085485 IC50 400.0 nM
CCOC(=O)c1ccccc1Nc1cccc2ccccc12 CHEMBL4570006 Ki 400.0 nM
N#Cc1ccccc1Cn1cc(CNC2=C(Cl)C(=O)c3cccnc3C2=O)nn1 CHEMBL4466461 IC50 420.0 nM
CC(C)=CCC/C(C)=C/CC/C(C)=C/Cc1cccc2c(C3=C(O)C(O)=CC(=O)C3=O)c[nH]c12 CHEMBL314400 Ki 640.0 nM
O=C1C=CC(=O)c2c1ccc1c2c(=O)oc2cc(F)ccc21 CHEMBL4060132 IC50 690.0 nM
O=C1C=CC(=O)c2c1ccc1c2c(=O)oc2cc(Cl)ccc21 CHEMBL4097725 IC50 770.0 nM
O=C1C=CC(=O)c2c1ccc1c2c(=O)oc2cc(O)ccc21 CHEMBL4086414 IC50 800.0 nM
COc1ccc2c(CSC3=CC(=O)c4ccccc4C3=O)cc(=O)oc2c1 CHEMBL3623325 IC50 900.0 nM
COc1ccc2c(c1)oc(=O)c1c3c(ccc12)C(=O)C=CC3=O CHEMBL4066643 IC50 980.0 nM
Cc1ccc2c(c1)oc(=O)c1c3c(ccc12)C(=O)C=CC3=O CHEMBL4094178 IC50 1000.0 nM