Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(C#N)cc(C(C)(C)O)c3o2)cc1 CHEMBL593709 IC50 28.0 nM
CCC(C)(O)c1cc(C#N)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL596491 IC50 31.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(Br)cc(C(C)(C)O)c3o2)cc1 CHEMBL595357 IC50 44.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(C#N)cc(C(C)O)c3o2)cc1 CHEMBL595352 IC50 46.0 nM
CCCC(C)(O)c1cc(C#N)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL596476 IC50 58.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(Br)cc(C(C)O)c3o2)cc1 CHEMBL596490 IC50 59.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(C#N)cc(C)c3o2)cc1 CHEMBL596130 IC50 60.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(C#N)cc(F)c3o2)cc1 CHEMBL606349 IC50 62.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(C#N)cc(C(C)(O)C(C)C)c3o2)cc1 CHEMBL594868 IC50 80.0 nM
CC(=O)c1cc(C#N)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL595359 IC50 86.0 nM
C#CC(C)(O)c1cc(Br)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL593247 IC50 94.0 nM
CCC(C)(O)c1cc(Br)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL606696 IC50 110.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(C#N)ccc3o2)cc1 CHEMBL260546 IC50 130.0 nM
CC#CC(C)(O)c1cc(C#N)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL592998 IC50 160.0 nM
CCCC(C)(O)c1cc(Br)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL594183 IC50 200.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(Br)cc(C(C)(O)C(C)C)c3o2)cc1 CHEMBL593246 IC50 210.0 nM
CC#CC(C)(O)c1cc(Br)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL595358 IC50 210.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(C#N)cc(C#N)c3o2)cc1 CHEMBL594978 IC50 270.0 nM
CC(=O)c1cc(Br)cc2nc(-c3ccc(NC(=O)COc4ccccc4C)cc3)oc12 CHEMBL593007 IC50 380.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3ccc(C#N)cc3o2)cc1 CHEMBL596131 IC50 410.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cccc(C(C)(C)O)c3o2)cc1 CHEMBL593966 IC50 440.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(Br)cc(C)c3o2)cc1 CHEMBL606983 IC50 510.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(Cl)cc([N+](=O)[O-])c3o2)cc1 CHEMBL407147 IC50 570.0 nM
COc1ccc2oc(-c3ccc(NC(=O)COc4ccccc4C)cc3)nc2c1 CHEMBL411258 IC50 840.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc(Br)cc(F)c3o2)cc1 CHEMBL594182 IC50 910.0 nM
Cc1ccccc1OCC(=O)Nc1ccc(-c2nc3cc([N+](=O)[O-])ccc3o2)cc1 CHEMBL261273 IC50 940.0 nM