COc1cc(Nc2ccnc3cc(C#N)ccc23)cc(OC)c1OC CHEMBL4575895 Kd 66.0 nM
Nc1nc(N)c2nc(-c3cccc(O)c3)c(-c3cccc(O)c3)nc2n1 CHEMBL230011 Kd 94.0 nM
COc1cc(Nc2ccnc3ccc(Cl)cc23)cc(OC)c1OC CHEMBL4556662 Kd 170.0 nM
COc1cc(Nc2ccnc3ccc(C#N)cc23)cc(OC)c1OC CHEMBL4585158 Kd 170.0 nM
Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCO)CC2)n1 CHEMBL5416410 Kd 190.0 nM
COc1cc(Nc2ccnc3ccc(I)cc23)cc(OC)c1OC CHEMBL4517424 Kd 190.0 nM
COc1cc(Nc2ccnc3ccc(Br)cc23)cc(OC)c1OC CHEMBL4443342 Kd 190.0 nM
COc1cc(Nc2ccnc3ccc(C(F)(F)F)cc23)cc(OC)c1OC CHEMBL535429 Kd 220.0 nM
COc1cc2nccc(Nc3cc(OC)c(OC)c(OC)c3)c2cc1OC CHEMBL311959 Kd 250.0 nM
CN1CCN(CCOc2cc(OC3CCOCC3)c3c(Nc4c(Cl)ccc5c4OCO5)ncnc3c2)CC1 CHEMBL217092 Kd apparent 275.0 nM
Cn1c(=O)c(Oc2ccc(F)cc2F)cc2cnc(NC3CCOCC3)nc21 CHEMBL1230122 Kd 320.0 nM
CS(=O)(=O)CCCOc1cccc2c1ccn2-c1ccnc(N[C@H]2CC[C@H](C(=O)N3CCC(O)CC3)CC2)n1 CHEMBL2425628 Kd 490.0 nM
COc1cc(Nc2ccnc3ccc(C(C)(C)C)cc23)cc(OC)c1OC CHEMBL530635 Kd 740.0 nM
Nc1ncnc2c1c(-c1cccc(OCc3ccccc3)c1)cn2[C@H]1C[C@H](N2CCC2)C1 CHEMBL551064 Kd apparent 835.0 nM
CSc1cccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1 CHEMBL386051 Kd 910.0 nM