CC(C)N(C#N)NC(=O)O[C@@H](C)CC1CCCCC1 CHEMBL371420 Ki 0.46 nM
C[C@@H](CC1CCCCC1)OC(=O)NN(C)C#N CHEMBL190121 Ki 1.4 nM
CCCC[C@@H](C=O)NC(=O)O[C@H](Cc1ccccc1)C(C)C CHEMBL113948 IC50 18.0 nM
C[C@@H](CC1CCCCC1)OC(=O)C1CCN1C#N CHEMBL183812 IC50 40.0 nM
CCCC[C@@H](C=O)NC(=O)O[C@@H](C)Cc1ccccc1 CHEMBL114161 IC50 40.0 nM
CCn1cnc2c(Nc3cc(F)cc(F)c3)nc(C#N)nc21 CHEMBL567341 pIC50 125.89 nM
CCC[C@H](N)C(=O)N[C@H](/C=C/S(=O)(=O)c1ccccc1)CCc1ccccc1 CHEMBL514348 Ki 137.0 nM
CC(=O)c1c(Nc2ccc(Cl)cc2)[nH]c2c(Cl)cc([N+](=O)[O-])cc2c1=O CHEMBL492175 IC50 145.0 nM
CCCC[C@@H](/C=N/NC(=O)N1CCOCC1)NC(=O)O[C@H](Cc1ccccc1)C(C)C CHEMBL203663 IC50 190.0 nM
CC(C)C[C@H](NC(=O)[C@H]1O[C@@H]1C(=O)O)C(=O)NCCCCN=C(N)N CHEMBL374508 IC50 190.0 nM
CCCC[C@@H](/C=N/NC(=O)N1CCOCC1)NC(=O)O[C@@H](C)Cc1ccccc1 CHEMBL204605 IC50 230.0 nM
C[C@@H](CC1CCCCC1)OC(=O)C1CCCN1C#N CHEMBL180839 IC50 580.0 nM
CCNc1nc(C#N)nc2c1ncn2-c1cc(F)cc(F)c1 CHEMBL567134 pIC50 645.65 nM