Cc1ccc(C(Nc2c(Nc3cccc(C(=O)N(C)C)c3O)c(=O)c2=O)C2(C)CCCO2)o1 CHEMBL3979652 pIC50 1.995 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3c(C(F)(F)F)cccc3s2)cc(OC)c1OC CHEMBL4637126 pIC50 39.81 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3c(Br)cccc3s2)cc(OC)c1OC CHEMBL4638895 IC50 80.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3c(F)cccc3s2)cc(OC)c1OC CHEMBL4632425 IC50 110.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2cccc(Cl)c2Cl)cc(OC)c1OC CHEMBL4647701 IC50 120.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2cc(Cl)ccc2Cl)cc(OC)c1OC CHEMBL4646569 IC50 130.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3c(Cl)cccc3s2)cc(OC)c1OC CHEMBL4646120 IC50 130.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2ccccc2Cl)cc(OC)c1OC CHEMBL4645971 IC50 140.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2ccccc2Br)cc(OC)c1OC CHEMBL4640388 IC50 160.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2ccc(Cl)cc2Cl)cc(OC)c1OC CHEMBL4648997 IC50 160.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3cc(Cl)ccc3s2)cc(OC)c1OC CHEMBL4641681 IC50 170.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3c(C)cccc3s2)cc(OC)c1OC CHEMBL4639692 IC50 250.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3cccc(Cl)c3s2)cc(OC)c1OC CHEMBL4638493 IC50 260.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3ccc(Cl)cc3s2)cc(OC)c1OC CHEMBL4640319 IC50 270.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2nc3ccccc3s2)cc(OC)c1OC CHEMBL4642230 IC50 300.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2cc(Cl)cc(Cl)c2)cc(OC)c1OC CHEMBL4647206 IC50 310.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2cccc(Br)c2)cc(OC)c1OC CHEMBL4645763 IC50 350.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2ccc(Cl)c(Cl)c2)cc(OC)c1OC CHEMBL4649351 IC50 350.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2cccc(Cl)c2)cc(OC)c1OC CHEMBL4635707 IC50 410.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2cc(C)ccc2C)cc(OC)c1OC CHEMBL4639114 IC50 610.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2ccccc2F)cc(OC)c1OC CHEMBL4644133 IC50 620.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2ccccc2C(F)(F)F)cc(OC)c1OC CHEMBL4639996 IC50 640.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2ccccc2C)cc(OC)c1OC CHEMBL4640657 IC50 790.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2cccc(F)c2)cc(OC)c1OC CHEMBL4640101 IC50 840.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3Cc2cc3ccccc3s2)cc(OC)c1OC CHEMBL4633183 IC50 900.0 nM
COc1cc(C(=O)N[C@@H]2C[C@H]3CCC[C@@H](C2)N3CC(=O)Nc2ccccc2C#N)cc(OC)c1OC CHEMBL4632989 IC50 930.0 nM