Cc1c(C)c2c(c(C)c1O)CC[C@@](C)(CCCCCCCCCn1ccnc1)O2 CHEMBL524809 ED50 1.0 nM
N#Cc1ccc(COc2ccc(-c3ccn[nH]3)nc2)cc1 CHEMBL5195099 IC50 6.5 nM
N#Cc1cccc(COc2ccc(-c3ccn[nH]3)nc2)c1 CHEMBL5183418 IC50 15.0 nM
Cc1ncsc1CCOc1ccc(-c2ccn[nH]2)cc1 CHEMBL5204432 IC50 17.0 nM
CN(C)C(=O)N1CCC(COc2ccc(-c3ccn[nH]3)nc2)CC1 CHEMBL5174407 IC50 19.0 nM
Fc1ccc(COc2ccc(-c3ccn[nH]3)nc2)cc1 CHEMBL5173608 IC50 21.0 nM
CN(C)S(=O)(=O)N1CCC[C@H](COc2ccc(-c3ccn[nH]3)nc2)C1 CHEMBL5169535 IC50 36.0 nM
CC(=O)N1CCC(COc2ccc(-c3ccn[nH]3)nc2)CC1 CHEMBL5206230 IC50 40.0 nM
Cc1ncsc1CCOc1ccc(-c2ccn[nH]2)nc1 CHEMBL5192170 IC50 44.0 nM
CNC(=O)N1CCC(COc2ccc(-c3ccn[nH]3)nc2)CC1 CHEMBL5172100 IC50 63.0 nM
Cc1ncsc1CCOc1cnc(-c2ccn[nH]2)nc1 CHEMBL5180285 IC50 66.0 nM
CS(=O)(=O)c1cc(O)cc(COc2ccc(-c3ccn[nH]3)nc2)c1 CHEMBL5208981 IC50 69.0 nM
COC(=O)N1CCC(COc2ccc(-c3ccn[nH]3)nc2)CC1 CHEMBL5183091 IC50 73.0 nM
CS(=O)(=O)c1ccc(COc2ccc(-c3ccn[nH]3)nc2)cc1 CHEMBL5195431 IC50 96.0 nM
O=C(C1CC1)N1CCC(COc2ccc(-c3ccn[nH]3)nc2)CC1 CHEMBL5199197 IC50 110.0 nM
CC(=O)N[C@H]1CC[C@@H](COc2ccc(-c3ccn[nH]3)nc2)CC1 CHEMBL5184859 IC50 170.0 nM
CC(=O)N1CCC[C@H](COc2ccc(-c3ccn[nH]3)nc2)C1 CHEMBL5191778 IC50 180.0 nM
CC(=O)N[C@H]1CC[C@H](COc2ccc(-c3ccn[nH]3)nc2)CC1 CHEMBL5203135 IC50 220.0 nM
CS(=O)(=O)c1cccc(COc2ccc(-c3ccn[nH]3)nc2)c1 CHEMBL5205521 IC50 260.0 nM
CCOC(=O)N1CCN(CCOc2ccc(-c3ccn[nH]3)cc2)CC1 CHEMBL5181522 IC50 510.0 nM
CS(=O)(=O)N1CCC(COc2ccc(-c3ccn[nH]3)nc2)CC1 CHEMBL5195609 IC50 640.0 nM
CC(=O)N1CCC[C@@H](COc2ccc(-c3ccn[nH]3)nc2)C1 CHEMBL5192567 IC50 640.0 nM
CS(=O)(=O)N1CCC[C@@H](COc2ccc(-c3ccn[nH]3)nc2)C1 CHEMBL5199278 IC50 710.0 nM
CS(=O)(=O)N1CCC[C@H](COc2ccc(-c3ccn[nH]3)nc2)C1 CHEMBL5189943 IC50 730.0 nM
CC(=O)N1CCN(c2ccc(OCC3COC(Cn4ccnc4)(c4ccc(Cl)cc4Cl)O3)cc2)CC1 CHEMBL157101 Ki 740.0 nM
O=c1cc(-c2ccc(C(F)(F)F)cc2)oc2ccccc12 CHEMBL2130955 IC50 760.0 nM