CCc1ccc(OC(F)(F)F)cc1CC(=O)N1CCc2cc(-c3cn(CC)c4ncnc(N)c34)ccc21 CHEMBL5279578 EC50 37.0 nM
CCc1ccc(OC(F)(F)F)cc1CC(=O)N1CCc2cc(-c3nn(CC)c4ncnc(N)c34)ccc21 CHEMBL5286788 EC50 95.0 nM
Cc1cc(C)n(CC(=O)N2CCc3c2ccc(-c2cn(C)c4ncnc(N)c24)c3F)n1 CHEMBL2441346 IC50 99.0 nM
Cc1[nH]c2ccc(Cl)cc2c1-c1ccnc(Nc2ccc(N3CCN(C)CC3)cc2)n1 CHEMBL1802782 IC50 100.0 nM
Cc1[nH]c2ccccc2c1-c1ccnc(Nc2cccnc2)n1 CHEMBL1802629 IC50 100.0 nM
CCn1cc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc21 CHEMBL4281823 IC50 116.0 nM
C[C@]12O[C@H](C[C@]1(O)CO)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)CNC4=O CHEMBL603469 Kd 120.0 nM
CS(=O)(=O)CCCOc1cccc2c1ccn2-c1ccnc(N[C@H]2CC[C@H](C(=O)N3CCC(O)CC3)CC2)n1 CHEMBL2425628 Kd 120.0 nM
Cc1[nH]c2ccccc2c1-c1ccnc(Nc2ccc(F)cc2)n1 CHEMBL1802778 IC50 150.0 nM
COc1cc(Nc2ncc(F)c(Nc3ccc4c(n3)NC(=O)C(C)(C)O4)n2)cc(OC)c1OC CHEMBL475251 Kd 180.0 nM
N#Cc1cnc2cnc(NCc3cccnc3)cc2c1Nc1ccc(F)c(Cl)c1 CHEMBL200381 IC50 250.0 nM
NC(=O)Nc1sc(-c2ccc(F)cc2)cc1C(N)=O CHEMBL257167 IC50 250.0 nM
Cn1cc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(Cl)c2)c2c(N)ncnc21 CHEMBL2171122 IC50 291.0 nM
Cc1[nH]c2ccccc2c1-c1ccnc(Nc2cccc(Cl)c2)n1 CHEMBL1802769 IC50 300.0 nM
CC(=O)Cn1cc(-c2cnc(N)c3c(-c4ccc(NC(=O)Nc5cccc(C)c5)cc4)csc23)cn1 CHEMBL5271785 IC50 306.0 nM
Cn1cc(-c2ccc3c(c2F)CCN3C(=O)Cc2cccc(C(F)(F)F)n2)c2c(N)ncnc21 CHEMBL2441342 IC50 359.0 nM
CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4c(c5c6ccccc6n2c5c31)C(=O)NC4 CHEMBL388978 Kd 360.0 nM
COCCO[C@H]1CC[C@H](n2nc(-c3ccc(Nc4nc5cc(Cl)cc(F)c5o4)cc3)c3c(N)ncnc32)CC1 CHEMBL5266620 IC50 364.0 nM
CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)NC4CCN(C)CC4)cc3OC)nc2N1C1CCCC1 CHEMBL513909 Kd 460.0 nM
Nc1ncc(-c2nnn(CCCO)n2)cc1-c1cc2cc(NC(=O)Nc3ccc(Cl)c(C(F)(F)F)c3)ccc2o1 CHEMBL5267979 IC50 475.0 nM
Cc1[nH]c2ccccc2c1-c1ccnc(Nc2ccc(Cl)cc2)n1 CHEMBL1802630 IC50 600.0 nM
O=C1Nc2cc(Br)ccc2/C1=C1/Nc2ccccc2/C1=N\O CHEMBL409450 IC50 600.0 nM
CCN(CC)CCNC(=O)c1c(C)[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c1C CHEMBL535 Kd 670.0 nM
Cn1cc(-c2ccc3c(c2)CCN3C(=O)Cc2cccc(C(F)(F)F)c2)c2c(N)ncnc21 CHEMBL2171124 IC50 696.0 nM
O=C1NCc2c1c1c3ccccc3n3c1c1c2c2ccccc2n1C1CCC3O1 CHEMBL1802486 IC50 750.0 nM
Cc1cccc(CC(=O)N2CCc3c2ccc(-c2cn(C)c4ncnc(N)c24)c3F)n1 CHEMBL2441340 IC50 905.0 nM
Cn1c(Nc2ccc(C(F)(F)F)cc2)nc2cc(Oc3ccnc(-c4ncc(C(F)(F)F)[nH]4)c3)ccc21 CHEMBL558752 Kd 950.0 nM
Cn1cc(-c2cnc(N)c3c(-c4ccc5c(c4)CCN5C(=O)Cc4ccccc4)csc23)cn1 CHEMBL2171132 IC50 978.0 nM
CN1C(=O)[C@@H](N2CCc3cn(Cc4ccccc4)nc3C2=O)COc2ccccc21 CHEMBL4088216 pIC50 1000.0 nM
CN1C(=O)[C@@H](N2CCc3c(nn(Cc4ccccc4)c3Br)C2=O)COc2ccccc21 CHEMBL4549667 pIC50 1000.0 nM
CN1C(=O)[C@@H](N2CCc3cn(CC4CCS(=O)(=O)CC4)nc3C2=O)COc2ccccc21 CHEMBL4097778 pIC50 1000.0 nM