Fc1ccn([C@H]2C[C@H](c3cc(O[C@H]4C[C@@H](n5cccn5)C4)ncn3)C2)n1 CHEMBL5090501 IC50 0.3 nM
c1ccc([C@H]2CN(c3cc(O[C@H]4C[C@@H](n5cccn5)C4)ncn3)CCO2)cc1 CHEMBL5092963 IC50 0.4 nM
Fc1cnn([C@H]2C[C@H](c3cc(O[C@H]4C[C@@H](n5cccn5)C4)ncn3)C2)c1 CHEMBL5075747 IC50 0.6 nM
Clc1ccn([C@H]2C[C@H](c3cc(O[C@H]4C[C@@H](n5cccn5)C4)ncn3)C2)n1 CHEMBL5081977 IC50 2.0 nM
Fc1ccc(CCOc2cc(N3CCCOCC3)ncn2)cc1 CHEMBL5093558 IC50 3.0 nM
c1ccc([C@H]2CN(c3cc(O[C@H]4C[C@@H](c5ncco5)C4)ncn3)CCO2)cc1 CHEMBL5085396 IC50 5.0 nM
O=C(Nc1ccn(-c2ccnc(F)c2)n1)C1(c2ccccc2F)CC1 CHEMBL5081193 IC50 5.0 nM
Cc1ccnn1CCCOc1cc(N2CCCCC2)ncn1 CHEMBL5091893 IC50 7.0 nM
Cc1ccnn1CCCOc1cc(N2CCOC(C(F)(F)F)C2)ncn1 CHEMBL5079831 IC50 7.0 nM
Cc1ccnn1CCCOc1cc(N2CCOC(c3ccccc3)C2)ncn1 CHEMBL5088572 IC50 7.0 nM
c1ccc([C@H]2CN(c3cc(O[C@H]4C[C@@H](n5ccnn5)C4)ncn3)CCO2)cc1 CHEMBL5091423 IC50 9.0 nM
c1ccc([C@H]2CN(c3cc(O[C@H]4C[C@@H](c5nnco5)C4)ncn3)CCO2)cc1 CHEMBL5082929 IC50 9.0 nM
c1cnn([C@H]2C[C@@H](Oc3cc([C@H]4C[C@H](n5cccn5)C4)ncn3)C2)c1 CHEMBL5084780 IC50 10.0 nM
Fc1ccc(CCOc2cc(N3CCOCC3)ncn2)cc1 CHEMBL5084384 IC50 12.0 nM
O=C(Nc1ccn(-c2ccccc2)n1)C1(c2ccccc2F)CC1 CHEMBL5169448 IC50 12.0 nM
c1ccc([C@H]2CN(c3cc(O[C@H]4C[C@@H](c5ccccc5)C4)ncn3)CCO2)cc1 CHEMBL5084868 IC50 15.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2c(F)cccc2F)CC1 CHEMBL5185729 IC50 17.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2ccccc2F)CC1 CHEMBL5203823 IC50 18.0 nM
O=C(Nc1ccn(-c2ncns2)n1)C1(c2ccccc2F)CC1 CHEMBL5206398 IC50 18.0 nM
O=C(Nc1ccn(-c2ccccc2)n1)C1(c2ccccc2)CC1 CHEMBL5204141 IC50 20.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2ccccc2)CC1 CHEMBL5172768 IC50 22.0 nM
O=C(Nc1ccn(-c2ccc(F)nc2)n1)C1(c2ccccc2F)CC1 CHEMBL5185644 IC50 23.0 nM
O=C(Nc1ccn(-c2ccncn2)n1)C1(c2ccccc2F)CC1 CHEMBL5205200 IC50 30.0 nM
C[C@H](C(=O)Nc1ccn(-c2ccccc2)n1)c1ccccc1 CHEMBL5199478 IC50 38.0 nM
COc1cc(-n2ccc(NC(=O)C3(c4ccccc4F)CC3)n2)ccn1 CHEMBL5194186 IC50 50.0 nM
CN(C)c1cc(OCCc2ccc(F)cc2)ncn1 CHEMBL5080503 IC50 60.0 nM
CN(c1cc(OCCc2ccc(F)cc2)ncn1)C1CCOC1 CHEMBL5077819 IC50 60.0 nM
O=C(Cc1ccccc1F)Nc1ccn(-c2ccccc2)n1 CHEMBL5190392 IC50 60.0 nM
O=C(Cc1ccccc1)Nc1ccn(-c2ccccc2)n1 CHEMBL5200554 IC50 70.0 nM
Fc1ccc(CCOc2cc(N3CCCCC3)ncn2)cc1 CHEMBL5088321 IC50 80.0 nM
O=C(Nc1ccn(-c2ccncc2)n1)C1(c2ccccc2F)CC1 CHEMBL5174762 IC50 80.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2ccc(F)cc2)CC1 CHEMBL5204609 IC50 100.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2ccccc2Cl)CC1 CHEMBL5202816 IC50 110.0 nM
N#Cc1ccc(C2(C(=O)Nc3ccn(-c4cncc(F)c4)n3)CC2)cc1 CHEMBL5192322 IC50 110.0 nM
Cc1ccnn1CCCOc1cc(N2CCOC3(COC3)C2)ncn1 CHEMBL5087669 IC50 120.0 nM
Cc1ccnn1CCOc1cc(N2CCCCC2)ncn1 CHEMBL5094213 IC50 140.0 nM
Cc1ccnn1CCCOc1cc(N2CCOC(c3ccnn3C)C2)ncn1 CHEMBL5094005 IC50 140.0 nM
O=C(Nc1ccn(-c2ccccc2)n1)C1(c2ccccc2)CC1(F)F CHEMBL5182190 IC50 140.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2cccc(F)c2F)CC1 CHEMBL5188173 IC50 140.0 nM
COc1cccc(C2(C(=O)Nc3ccn(-c4cncc(F)c4)n3)CC2)c1 CHEMBL5200718 IC50 170.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2cc(F)ccc2F)CC1 CHEMBL5202203 IC50 170.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2cccc(F)c2)CC1 CHEMBL5190417 IC50 190.0 nM
c1cnn([C@H]2C[C@@H](Oc3cc([C@H]4C[C@@H](n5cccn5)C4)ncn3)C2)c1 CHEMBL5084617 IC50 210.0 nM
C[C@@H](C(=O)Nc1ccn(-c2ccccc2)n1)c1ccccc1 CHEMBL5194918 IC50 210.0 nM
Fc1ccc(CCOc2cc(N3CCCCCC3)ncn2)cc1 CHEMBL5079994 IC50 230.0 nM
Cc1ccnn1CCCOc1cc(N2C3COCC2C3)ncn1 CHEMBL5094745 IC50 230.0 nM
O=C(Nc1ccn(-c2ccccc2)n1)C1(c2ccccc2)COC1 CHEMBL5202062 IC50 260.0 nM
O=C(Cc1ccccc1F)Nc1nc(-c2ccccc2)cs1 CHEMBL5178289 IC50 280.0 nM
CC(C)(C(=O)Nc1ccn(-c2ccccc2)n1)c1ccccc1 CHEMBL5174196 IC50 300.0 nM
N#Cc1cccc(C2(C(=O)Nc3ccn(-c4cncc(F)c4)n3)CC2)c1 CHEMBL5202263 IC50 310.0 nM
O=C(Nc1ccn(-c2cncc(F)c2)n1)C1(c2ccc(Cl)cc2)CC1 CHEMBL5207495 IC50 340.0 nM
Cc1ccccc1C1(C(=O)Nc2ccn(-c3cncc(F)c3)n2)CC1 CHEMBL5190980 IC50 400.0 nM
Fc1ccc(CCOc2cc(N3CCCC3)ncn2)cc1 CHEMBL5082781 IC50 430.0 nM
Fc1ccc(CCOc2cc(N3CCCCC3)ccn2)cc1 CHEMBL5083459 IC50 440.0 nM
O=C(Cc1ccccc1)Nc1nc(-c2ccccc2)cs1 CHEMBL2403494 IC50 500.0 nM
COc1ccc(C2(C(=O)Nc3ccn(-c4cncc(F)c4)n3)CC2)cc1 CHEMBL5170748 IC50 640.0 nM
CC[C@@H](C(=O)Nc1ccn(-c2ccccc2)n1)c1ccccc1 CHEMBL5201832 IC50 650.0 nM
O=C(Cc1ccccc1F)Nc1cnn(-c2ccccc2)n1 CHEMBL5181945 IC50 900.0 nM
CC1(C)CC1(C(=O)Nc1ccn(-c2ccccc2)n1)c1ccccc1 CHEMBL5177661 IC50 900.0 nM