O=C(Nc1ccc(OC(F)(F)F)cc1)NC1CCN(C(=O)C(F)(F)F)CC1 CHEMBL1257517 IC50 0.4 nM
Cc1ccc(S(=O)(=O)N2CCC(NC(=O)Nc3ccc(OC(F)(F)F)cc3)CC2)cc1 CHEMBL1257759 IC50 0.4 nM
O=C(Nc1ccc(OC(F)(F)F)cc1)NC1CCN(S(=O)(=O)c2ccc(C(F)(F)F)cc2)CC1 CHEMBL3642246 IC50 0.4 nM
CN(C)c1cccc2c(S(=O)(=O)N3CCC(NC(=O)Nc4ccc(OC(F)(F)F)cc4)CC3)cccc12 CHEMBL1257880 IC50 0.8 nM
COC(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL3642245 IC50 0.9 nM
NC(=O)C(SCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C1CCCC1 CHEMBL4741234 IC50 0.94 nM
COC(=O)c1cccc(C(=O)N2CCC(CNC(=O)NC34CC5CC(CC(C5)C3)C4)CC2)c1 CHEMBL215121 IC50 1.1 nM
COC(=O)c1ccc(C(=O)N2CCC(CNC(=O)NC34CC5CC(CC(C5)C3)C4)CC2)cc1 CHEMBL215908 IC50 1.1 nM
O=C(NC1CCN(C(=O)C(F)(F)F)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL217758 IC50 1.1 nM
COC(=O)c1ccc(C(=O)N2CCC(NC(=O)NC34CC5CC(CC(C5)C3)C4)CC2)cc1 CHEMBL215999 IC50 1.1 nM
O=C(NC1CCN(C(=O)c2ccccn2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL215161 IC50 1.2 nM
O=C(NC1CCN(C(=O)c2ccccc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL216016 IC50 1.3 nM
CS(=O)(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL1668935 IC50 1.4 nM
O=C(NC1CCN(C(=O)c2ccncc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL214179 IC50 1.7 nM
COC(=O)c1ccccc1C(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL214644 IC50 1.7 nM
COC(=O)c1ccccc1C(=O)N1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL384280 IC50 1.8 nM
O=C(NCC1CCN(C(=O)C(F)(F)F)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL214127 IC50 1.8 nM
O=C(NC1CCN(C(=O)c2cccnc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL214128 IC50 2.1 nM
CCCC(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL215125 IC50 2.64 nM
COC(=O)CCCC(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL214505 IC50 2.7 nM
CCC(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL214943 IC50 3.19 nM
O=C(NCC1CCN(C(=O)c2ccccc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL214883 IC50 3.2 nM
O=C(NC1CCN(C(=O)c2ccc(C(=O)O)cc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL386384 IC50 3.3 nM
COC(=O)CCCC(=O)N1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL384075 IC50 3.4 nM
CC(C)(C)OC(=O)N1CCC(NC(=O)NC2CCCCC2)CC1 CHEMBL3640214 IC50 4.3 nM
CC(SC(C(N)=O)C1CCCC1)c1cccc(C(F)(F)F)c1 CHEMBL4761537 IC50 4.7 nM
O=C(NC1CCN(C(=O)c2ccccc2)CC1)NC1CCN(C(=O)c2ccccc2)CC1 CHEMBL3642240 IC50 4.8 nM
CC(=O)N1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL215025 IC50 5.0 nM
O=C(NCC1CCN(C(=O)c2ccncc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL215069 IC50 5.4 nM
COC(=O)CCC(=O)N1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL217711 IC50 6.2 nM
CCCC(=O)N1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL214675 IC50 6.7 nM
O=C(NCC1CCN(C(=O)c2cccnc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL425436 IC50 7.3 nM
O=C(NCC1CCN(C(=O)c2ccccn2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL386855 IC50 7.6 nM
O=C(NC1CCN(Cc2ccccc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL387034 IC50 8.4 nM
CCC(=O)N1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL215874 IC50 8.7 nM
COC(=O)CCC(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL215827 IC50 9.0 nM
NC(=O)C(SCc1cc(Br)cc(Br)c1)C1CCCC1 CHEMBL4759724 IC50 9.0 nM
NC(=O)C(SCc1ccc(Cl)c(OC(F)(F)F)c1)C1CCCC1 CHEMBL4778376 IC50 10.0 nM
O=C(NC1CCN(C(=O)c2cccc(C(=O)O)c2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL385946 IC50 10.1 nM
NC(=O)C(SCc1ccc(F)c(C(F)(F)F)c1)C1CCCC1 CHEMBL4744212 IC50 10.1 nM
NC(=O)C(SCc1cc(Cl)cc(Cl)c1)C1CCCC1 CHEMBL4785066 IC50 11.0 nM
CC(=O)N1CCC(NC(=O)Nc2ccc(OC(F)(F)F)cc2)CC1 CHEMBL1668934 IC50 11.5 nM
O=C(NCC1CCN(C(=O)c2ccc(C(=O)O)cc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL387280 IC50 11.8 nM
NC(=O)C(SCCc1cccc(C(F)(F)F)c1)C1CCCC1 CHEMBL4758328 IC50 14.0 nM
CC(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL436774 IC50 14.5 nM
NC(=O)C(SCc1cccc(C(F)(F)F)c1)C1CCCC1 CHEMBL4791944 IC50 16.0 nM
Cc1cc(C)cc(CSC(C(N)=O)C2CCCC2)c1 CHEMBL4790572 IC50 18.0 nM
NC(=O)C(SCc1cccc(C(F)(F)F)c1)C1CCCCC1 CHEMBL4777339 IC50 19.0 nM
NC(=O)C(SCc1cccc(C(F)(F)F)c1)SCc1cccc(C(F)(F)F)c1 CHEMBL4779655 IC50 23.0 nM
NC(=O)C(SCc1cccc(OC(F)(F)F)c1)C1CCCC1 CHEMBL4751272 IC50 26.0 nM
CC(=O)N1CCC(NC(=O)NC2CCCCCC2)CC1 CHEMBL1668928 IC50 27.6 nM
CC(C)CC(SCc1cccc(C(F)(F)F)c1)C(N)=O CHEMBL4741225 IC50 28.0 nM
O=C(CC12CC3CC(CC(C3)C1)C2)NC1CCN(C(=O)C(F)(F)F)CC1 CHEMBL3642244 IC50 28.3 nM
CCCCC(SCc1cccc(C(F)(F)F)c1)C(N)=O CHEMBL4750146 IC50 29.0 nM
NC(=O)C(SCc1cccc([N+](=O)[O-])c1)C1CCCC1 CHEMBL4756934 IC50 32.0 nM
NC(=O)C(SCc1ccc2ccccc2c1)C1CCCC1 CHEMBL4753260 IC50 33.0 nM
O=C(O)CCCC(=O)N1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL215820 IC50 41.6 nM
CCCCCCCCCCCCNC(=O)NC1CCNCC1 CHEMBL3640213 IC50 42.5 nM
O=C(NCC1CCN(C(=O)c2cccc(C(=O)O)c2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL437328 IC50 43.6 nM
CCCCCCNC(=O)NC1CCCCC1 CHEMBL3661351 IC50 70.0 nM
CC(C)c1ccc(NC(=O)NC2CCCCC2)cc1 CHEMBL1360431 IC50 70.0 nM
O=C(O)CCCC(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL426340 IC50 72.8 nM
O=C(Nc1ccc2[nH]ccc2c1)NC1CCCCC1 CHEMBL3640216 IC50 87.0 nM
CC(C)C(SCc1cccc(C(F)(F)F)c1)C(N)=O CHEMBL4800559 IC50 88.0 nM
O=C(NC1CCCCCCC1)NC1CCCCC1 CHEMBL1330191 IC50 90.0 nM
O=C(NC1CCCCCCCCCCC1)NC1CCCCC1 CHEMBL3661369 IC50 100.0 nM
O=C(NC1CCCCC1)OC1C2CC3CC(C2)CC1C3 CHEMBL3661318 IC50 100.0 nM
O=C(NCC1CCCCC1)Nc1cccc(Cl)c1 CHEMBL2031928 IC50 100.0 nM
O=C(NC1CCCCC1)NC1C2CC3CC(C2)CC1C3 CHEMBL1609005 IC50 100.0 nM
O=C(NC12CC3CC(CC(C3)C1)C2)NC12CC3CC(CC(C3)C1)C2 CHEMBL3263303 IC50 100.0 nM
CCCCCCNC(=O)Nc1ccc(C(C)C)cc1 CHEMBL3661396 IC50 100.0 nM
CC1CCC(NC(=O)NC2CCCCC2)CC1 CHEMBL3661360 IC50 100.0 nM
O=C(NC1CCCCC1)NC1CC2CCC1C2 CHEMBL3661370 IC50 100.0 nM
CCCCCCCCCNC(=O)NC1CCCCC1 CHEMBL3661354 IC50 100.0 nM
CCCCCCCCCCNC(=O)NC1CCCCC1 CHEMBL67158 IC50 100.0 nM
O=C(NC(=O)c1ccc(Cl)cc1)NC1CCCCC1 CHEMBL3661400 IC50 100.0 nM
O=C(NCCC1=CCCCC1)NC1CCCCC1 CHEMBL1533919 IC50 100.0 nM
N#Cc1ccc(NC(=O)NC2CCCCC2)cc1 CHEMBL3661383 IC50 100.0 nM
O=C(NC1CCCCCC1)NC1CCCCC1 CHEMBL3661368 IC50 100.0 nM
O=C(NC1CCCCC1)OCc1ccc(-c2ccccc2)cc1 CHEMBL3661317 IC50 100.0 nM
O=C(Nc1nnn[nH]1)NC1CCCCC1 CHEMBL3661365 IC50 100.0 nM
O=C(NC1CCCCC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL242255 IC50 100.0 nM
C[C@H](NC(=O)NC1CCCCC1)c1ccccc1 CHEMBL3661373 IC50 100.0 nM
O=C(NC1CCCCC1)NC1CCCc2ccccc21 CHEMBL3661379 IC50 100.0 nM
O=C(NCCCc1ccccc1)NC12CC3CC(CC(C3)C1)C2 CHEMBL2031923 IC50 100.0 nM
O=C(Nc1ccc(OC(F)(F)F)cc1)NC1CCCCC1 CHEMBL2031931 IC50 100.0 nM
O=C(NC1CCCCC1)OCc1cccc2ccccc12 CHEMBL3661320 IC50 100.0 nM
O=C(Nc1ccc(Oc2ccccc2)cc1)NC1CCCCC1 CHEMBL2098452 IC50 100.0 nM
O=C(NCCC1CCCCC1)NC1CCCCC1 CHEMBL3661363 IC50 100.0 nM
CCCCCCCNC(=O)NC1CCCCC1 CHEMBL3661353 IC50 100.0 nM
O=C(O)CCCCCCCCCCCNC(=O)NC1CCCCC1 CHEMBL3661356 IC50 100.0 nM
O=C(NCC1CCCCC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL3661375 IC50 100.0 nM
CC(C)(C)C1CCC(NC(=O)NC2CCCCC2)CC1 CHEMBL3661367 IC50 100.0 nM
CC(C)c1ccc(NC(=O)NCC2CCCCC2)cc1 CHEMBL2031927 IC50 100.0 nM
CC1CCCCC1NC(=O)NC1CCCCC1 CHEMBL3661361 IC50 100.0 nM
CCCCCCCCCCCCNC(=O)NC1CCCCC1 CHEMBL3661355 IC50 100.0 nM
O=C(NC1CCCCCCCCCCC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL3661391 IC50 100.0 nM
CCCCCCCCCCCCCNC(=O)NC1CCCCC1 CHEMBL3661357 IC50 100.0 nM
CC(C)C(SCc1ccc(Br)cc1)C(N)=O CHEMBL4791378 IC50 100.0 nM
CC(C)(C)CC(C)(C)NC(=O)NC1C2CC3CC(C2)CC1C3 CHEMBL3661329 IC50 110.0 nM
O=C(Nc1ccc(Br)cc1)NC1CCCCC1 CHEMBL3661387 IC50 110.0 nM
NC(=O)C(SCc1ccc(Br)cc1)c1ccccc1 CHEMBL4765145 IC50 110.0 nM
O=C(NCC1CCN(Cc2ccccc2)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL215146 IC50 112.0 nM
O=C(Nc1ccc(Cl)cc1)Nc1ccc(Cl)c(Cl)c1 CHEMBL1076347 IC50 120.0 nM
O=C(Nc1ccc(I)cc1)NC1CCCCC1 CHEMBL1231797 IC50 120.0 nM
CCCCCCCCNC(=O)NC1CCCCC1 CHEMBL3661337 IC50 120.0 nM
CC1CCC(C(C)C)C(OC(=O)NC2CCCCC2)C1 CHEMBL3661319 IC50 120.0 nM
O=C(NCC1CCCCC1)Nc1ccc2ccccc2c1 CHEMBL3661381 IC50 130.0 nM
O=C(NC1CCCCC1)OC1CCCCC1 CHEMBL3657188 IC50 130.0 nM
O=C(Nc1c2ccccc2nc2ccccc12)NC1CCCCC1 CHEMBL3661380 IC50 140.0 nM
CC(C)(C)OC(=O)NCCNC(=O)NC1CCCCC1 CHEMBL3661349 IC50 140.0 nM
CC(C)C(SCc1ccc(Cl)cc1Cl)C(N)=O CHEMBL4783157 IC50 140.0 nM
NC(=O)C(SCc1cccc(C(F)(F)F)c1)c1ccccc1 CHEMBL4762042 IC50 140.0 nM
Cc1cccc(C(O)C2OC2c2ccc(-c3ccccc3)cc2)c1 CHEMBL3661411 IC50 150.0 nM
O=C(Nc1ccncc1)NC1CCCCC1 CHEMBL3661378 IC50 150.0 nM
CCCC(SCc1cccc(C(F)(F)F)c1)C(N)=O CHEMBL4748684 IC50 150.0 nM
O=C(NC1CCCCC1)NC1CCCCC1 CHEMBL1458 IC50 160.0 nM
O=C(NCC1CCCCC1)NC1CCCCC1 CHEMBL3661362 IC50 160.0 nM
CCCCCCc1ccc(NC(=O)NC2CCCCC2)cc1 CHEMBL2031932 IC50 160.0 nM
O=C(NCCc1ccccc1)NC1CCCCC1 CHEMBL193888 IC50 160.0 nM
O=C(NC1CCN(C(=O)c2ccccc2C(=O)O)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL214884 IC50 161.2 nM
Cc1ccc(NC(=O)NC2CCCCC2)cc1 CHEMBL3661382 IC50 170.0 nM
O=C(O)CCC(=O)N1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL386455 IC50 174.5 nM
CC(NC(=O)NC1CCCCC1)C1C2CC3CC(C2)CC1C3 CHEMBL3661371 IC50 180.0 nM
Cc1cccc(C)c1NC(=O)NC1CCCCC1 CHEMBL3661372 IC50 180.0 nM
CCCCCCCCNC(=O)Nc1cccc(Cl)c1 CHEMBL3661339 IC50 180.0 nM
O=C(NC1CCCCC1)OCCCCc1ccc([N+](=O)[O-])cc1 CHEMBL3657193 IC50 180.0 nM
O=C(Nc1cccc(Cl)c1)NC1CCCCC1 CHEMBL192293 IC50 190.0 nM
O=C(NCc1ccc(Cl)cc1)NC1CCCCC1 CHEMBL3661385 IC50 190.0 nM
Cc1cccc(C(=O)C2OC2c2ccc(-c3ccccc3)cc2)c1 CHEMBL3661410 IC50 190.0 nM
N#Cc1cccc(CSC(C(N)=O)C2CCCC2)c1 CHEMBL4762164 IC50 193.0 nM
O=C(c1ccccc1)C1OC1c1ccc(-c2ccccc2)cc1 CHEMBL3661417 IC50 200.0 nM
O=C(NCCc1ccc(Cl)cc1)NC1CCCCC1 CHEMBL3661386 IC50 200.0 nM
C=C(C)CCOC(=O)NC1CCCCC1 CHEMBL3657192 IC50 220.0 nM
COc1ccc(NC(=O)NC2CCCCC2)cc1 CHEMBL191968 IC50 230.0 nM
CC(C)(C)c1ccc(NC(=O)NC2CCCCC2)cc1 CHEMBL2029374 IC50 230.0 nM
CCCCCCCCNC(=O)NCCCCCC CHEMBL3661335 IC50 240.0 nM
CCCCCCCCCCCCCCNC(=O)NC1CCCCC1 CHEMBL3661358 IC50 240.0 nM
CCCCCCNC(=O)Nc1cccc(Cl)c1 CHEMBL3661331 IC50 250.0 nM
O=C(O)CCC(=O)N1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL385348 IC50 254.5 nM
O=C(Nc1ccc(Cl)c(Cl)c1)Nc1ccc(Cl)c(Cl)c1 CHEMBL10835 IC50 260.0 nM
CCCCCCCCCCCCNC(=O)NCC(C)C CHEMBL3661343 IC50 260.0 nM
CC(=O)c1ccc(NC(=O)NC2CCCCC2)cc1 CHEMBL3661384 IC50 270.0 nM
CC(=O)N1CCC(NC(=O)CC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL3642242 IC50 275.1 nM
CCCNC(=O)Nc1cccc2ccccc12 CHEMBL3661398 IC50 280.0 nM
NC(=O)C(SCc1ccc(Cl)cc1Cl)c1ccccc1 CHEMBL4800165 IC50 280.0 nM
O=NC(c1ccccc1)C1OC1c1ccccc1 CHEMBL3661402 IC50 290.0 nM
O=C(NCCCc1ccccc1)NC1CCCCC1 CHEMBL1231909 IC50 290.0 nM
CCCCCCCCCCNC(=O)Nc1cccc(Cl)c1 CHEMBL3661341 IC50 300.0 nM
O=C(c1ccccc1)C1OC1c1ccc(F)cc1 CHEMBL3661416 IC50 300.0 nM
O=C(c1ccccc1)C1OC1c1ccccc1 CHEMBL1733373 IC50 300.0 nM
[O-][S+](c1ccccc1)C1OC1c1ccccc1 CHEMBL3661403 IC50 310.0 nM
NC(=O)C(SCc1ccc([N+](=O)[O-])cc1)C1CCCC1 CHEMBL4758098 IC50 315.0 nM
O=C(NC1CCCCC1)Oc1ccccc1CO CHEMBL3657189 IC50 320.0 nM
O=C(NC1CCCCC1)OCc1c2ccccc2cc2ccccc12 CHEMBL3661321 IC50 330.0 nM
O=C(NC1CCCCC1)OCCCCC1CCCCC1 CHEMBL3657191 IC50 340.0 nM
O=C(NC1CCCCC1)Oc1ccc2ccccc2c1 CHEMBL77250 IC50 350.0 nM
O=C(Nc1ccc([N+](=O)[O-])cc1)NC1CCCCC1 CHEMBL3661390 IC50 360.0 nM
CC(=O)c1cccc(CSC(C(N)=O)C2CCCC2)c1 CHEMBL4759940 IC50 384.0 nM
NC(=O)C(SCc1cc(F)cc(F)c1)C1CCCC1 CHEMBL4795572 IC50 399.0 nM
O=C(Nc1ccc(Cl)cc1)NC1CCCCC1 CHEMBL11405 IC50 400.0 nM
O=C(NCC1CCN(C(=O)c2ccccc2C(=O)O)CC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL214735 IC50 407.1 nM
O=C(CC1CCCCC1)NC1CCCCC1 CHEMBL3661325 IC50 420.0 nM
NC(=O)C(SCc1ccc(C(=O)NCc2ccccc2C(F)(F)F)cc1)C1CCCC1 CHEMBL4756126 IC50 422.0 nM
O=C(Nc1ccc(F)cc1)NC1CCCCC1 CHEMBL1573741 IC50 430.0 nM
CC(C)C(SCc1ccc(C(C)(C)C)cc1)C(N)=O CHEMBL4762926 IC50 430.0 nM
NC(=O)C(SCc1cccc(C(=O)NCc2ccccc2C(F)(F)F)c1)C1CCCC1 CHEMBL4785232 IC50 433.0 nM
NC(=O)C(SCc1c(F)cccc1F)C1CCCC1 CHEMBL4797034 IC50 441.0 nM
O=C(Nc1ccc2nc[nH]c2c1)NC1CCCCC1 CHEMBL3642236 IC50 457.0 nM
C(=NC1CCCCC1)=NC1CCCCC1 CHEMBL162598 IC50 470.0 nM
CCCCCCCCNC(=O)OC CHEMBL3657186 IC50 480.0 nM
O=C(Nc1cccc2ccccc12)NC1CCCCC1 CHEMBL1713120 IC50 480.0 nM
CC(C)c1ccc(NC(=O)NCCc2ccccc2)cc1 CHEMBL3661395 IC50 480.0 nM
CC(C)(C)c1ccc(CS[C@H](C(N)=O)c2ccccc2)cc1 CHEMBL4758730 IC50 480.0 nM
NC(=O)C(SCc1ccnc(Cl)c1)C1CCCC1 CHEMBL4752449 IC50 493.0 nM
CC(C)(C)OC(=O)n1cc(CSC(C(N)=O)C2CCCC2)c2ccccc21 CHEMBL4752183 IC50 500.0 nM
NC(=O)C(SCc1ccc(OC(F)(F)F)cc1)c1ccccc1 CHEMBL4795018 IC50 500.0 nM
O=C(NCC1CCCCC1)Nc1ccccc1 CHEMBL3661376 IC50 530.0 nM
O=C(NCCCc1ccccc1)Nc1ccccc1 CHEMBL1413197 IC50 550.0 nM
O=C(NCCc1cnc[nH]1)NC1CCCCC1 CHEMBL3661364 IC50 550.0 nM
O=C(NC1CCCCC1)NC1CCNCC1 CHEMBL3642238 IC50 561.7 nM
CCCCCCNC(=O)Nc1ccc2ccccc2c1 CHEMBL3661330 IC50 570.0 nM
CCCCCCCCNC(=O)Nc1ccccc1 CHEMBL3661338 IC50 580.0 nM
O=C(NCCCCc1ccccc1)NC1CCCCC1 CHEMBL3661377 IC50 580.0 nM
CCCCCCCCCCNC(=O)Nc1ccccc1 CHEMBL3661340 IC50 610.0 nM
CCCCN1CCC(CNC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL386044 IC50 613.0 nM
CCCCCCCCCCCCNC(=O)Nc1ccc2[nH]ccc2c1 CHEMBL3640215 IC50 639.1 nM
CCCCCCCCCCCCNC(=O)NCCCC CHEMBL3661345 IC50 640.0 nM
CC(C)(C)c1ccc(CSC(C(N)=O)c2ccccc2)cc1 CHEMBL4785633 IC50 640.0 nM
CC(C)C(SCc1ccc(OC(F)(F)F)cc1)C(N)=O CHEMBL4765067 IC50 670.0 nM
O=C(CCCCc1ccccc1)NC1CCCCC1 CHEMBL3661327 IC50 680.0 nM
CCCCCCCCNC(=O)NCCC CHEMBL3661332 IC50 680.0 nM
CC(C)(C)c1ccc(CS[C@@H](C(N)=O)c2ccccc2)cc1 CHEMBL4748651 IC50 680.0 nM
CCCCCCCCNC(=O)NCCCCC CHEMBL3661333 IC50 720.0 nM
OC(c1ccccc1)C1OC1c1ccc(-c2ccccc2)cc1 CHEMBL3661406 IC50 720.0 nM
CCCCCCCCCCCNC(=O)NCCCC CHEMBL3661342 IC50 740.0 nM
NC(=O)C(SCC1CCCCC1)C1CCCC1 CHEMBL4799024 IC50 773.0 nM
CCCN1CCC(NC(=O)NC23CC4CC(CC(C4)C2)C3)CC1 CHEMBL215168 IC50 809.0 nM
NC(=O)C(SCc1cccc(C(=O)O)c1)C1CCCC1 CHEMBL4793637 IC50 839.0 nM
O=C(c1ccccc1)C1OC1c1cccc2ccccc12 CHEMBL3661418 IC50 850.0 nM
CC(C(=O)O)c1ccc(CSC(C(N)=O)C2CCCC2)cc1 CHEMBL4753889 IC50 899.0 nM
CCCCCNC(=O)NC1CCCCC1 CHEMBL3661350 IC50 920.0 nM
O=C(CC1CCCNC1)NC12CC3CC(CC(C3)C1)C2 CHEMBL3642248 IC50 960.0 nM
COc1ccc(CCNC(=O)NC2CCCCC2)cc1OC CHEMBL1568999 IC50 1000.0 nM
CCCNC(=O)NC1CCCCCCCCCCC1 CHEMBL3661328 IC50 1000.0 nM