O=c1[nH]c2c(S(=O)(=O)c3ccccc3)csc2c(=O)n1O CHEMBL361962 IC50 0.023 nM
O=c1[nH]c2c(-c3ccccc3)csc2c(=O)n1O CHEMBL361011 IC50 0.028 nM
O=c1[nH]c2c(Cc3ccccc3)coc2c(=O)n1O CHEMBL183133 IC50 0.061 nM
O=c1[nH]c2c(sc3ccccc32)c(=O)n1O CHEMBL359533 IC50 0.062 nM
O=c1[nH]c2sccc2c(=O)n1O CHEMBL361350 IC50 0.101 nM
Cc1ccc(-c2coc3c(=O)n(O)c(=O)[nH]c23)cc1 CHEMBL182381 IC50 0.128 nM
O=c1[nH]c2c(-c3ccc(-c4ccccc4)cc3)coc2c(=O)n1O CHEMBL364591 IC50 0.136 nM
Cc1csc2[nH]c(=O)n(O)c(=O)c12 CHEMBL183792 IC50 0.145 nM
O=c1[nH]c2sc3c(c2c(=O)n1O)CCCC3 CHEMBL362842 IC50 0.157 nM
O=c1[nH]c2ccccc2c(=O)n1O CHEMBL183852 IC50 0.16 nM
O=c1[nH]c2cccc(Cl)c2c(=O)n1O CHEMBL182687 IC50 0.185 nM
O=c1[nH]c2cc(-c3ccccc3)sc2c(=O)n1O CHEMBL183062 IC50 0.202 nM
COc1cccc(-c2coc3c(=O)n(O)c(=O)[nH]c23)c1 CHEMBL185325 IC50 0.215 nM
NC(=O)c1ccc(-c2cccc(Cn3c(=O)n(O)c(=O)c4sccc43)c2)cc1 CHEMBL181962 IC50 0.226 nM
COc1ccc(-c2coc3c(=O)n(O)c(=O)[nH]c23)cc1 CHEMBL359747 IC50 0.23 nM
O=c1[nH]c2c(oc3ccccc32)c(=O)n1O CHEMBL181766 IC50 0.257 nM
CC(C)(C)c1cc2[nH]c(=O)n(O)c(=O)c2s1 CHEMBL360615 IC50 0.258 nM
O=c1[nH]c2c(-c3ccccc3)coc2c(=O)n1O CHEMBL183539 IC50 0.276 nM
O=c1c2sccc2n(CC2COc3ccccc3O2)c(=O)n1O CHEMBL361546 IC50 0.292 nM
O=c1[nH]c2c(-c3ccc(Br)cc3)coc2c(=O)n1O CHEMBL180566 IC50 0.327 nM
O=c1c2sccc2n(Cc2cccc(Br)c2)c(=O)n1O CHEMBL185322 IC50 0.55 nM
CC(=O)Nc1cccc(-c2cccc(Cn3c(=O)n(O)c(=O)c4sccc43)c2)c1 CHEMBL182077 IC50 0.556 nM
O=c1c2ccsc2n(Cc2ccccc2)c(=O)n1O CHEMBL182974 IC50 2.0 nM
COc1cc(Cn2c(=O)n(O)c(=O)c3c(C)csc32)cc2c1OCO2 CHEMBL182519 IC50 3.04 nM
Cc1csc2c1c(=O)n(O)c(=O)n2Cc1ccccc1 CHEMBL181709 IC50 3.99 nM
Cc1csc2c1c(=O)n(O)c(=O)n2C CHEMBL181637 IC50 4.62 nM
COc1ccc(-n2c(=O)n(O)c(=O)c3c(C)csc32)cc1 CHEMBL362205 IC50 8.45 nM
Cc1csc2c(=O)n(O)c(=O)n(Cc3cccc(-c4ccc(C(N)=O)cc4)c3)c12 CHEMBL181907 IC50 30.2 nM
O=C(O)C(=O)CC(=O)c1ccc(-c2ccc(OC(F)(F)F)cc2)s1 CHEMBL182756 IC50 310.0 nM
COc1ccc(-c2ccc(Cl)c(C(=O)CC(=O)C(=O)O)c2)cc1 CHEMBL182748 IC50 570.0 nM
O=C(O)C(=O)CC(=O)c1ccc(-c2ccc(Cl)c(F)c2)s1 CHEMBL361960 IC50 900.0 nM
O=C(O)C(=O)CC(=O)c1ccc(-c2ccc(Cl)cc2)o1 CHEMBL183027 IC50 980.0 nM