NC(=O)c1ccc(-c2cccc(Cn3c(=O)n(O)c(=O)c4sccc43)c2)cc1 CHEMBL181962 IC50 0.003 nM
CC(=O)Nc1cccc(-c2cccc(Cn3c(=O)n(O)c(=O)c4sccc43)c2)c1 CHEMBL182077 IC50 0.004 nM
O=c1[nH]c2sc3c(c2c(=O)n1O)CCCC3 CHEMBL362842 IC50 0.009 nM
O=c1[nH]c2c(S(=O)(=O)c3ccccc3)csc2c(=O)n1O CHEMBL361962 IC50 0.01 nM
O=c1c2sccc2n(CC2COc3ccccc3O2)c(=O)n1O CHEMBL361546 IC50 0.011 nM
O=c1[nH]c2c(-c3ccccc3)csc2c(=O)n1O CHEMBL361011 IC50 0.012 nM
O=c1[nH]c2cccc(Cl)c2c(=O)n1O CHEMBL182687 IC50 0.014 nM
Cc1csc2[nH]c(=O)n(O)c(=O)c12 CHEMBL183792 IC50 0.014 nM
COc1cc(Cn2c(=O)n(O)c(=O)c3c(C)csc32)cc2c1OCO2 CHEMBL182519 IC50 0.018 nM
O=c1[nH]c2c(-c3ccc(-c4ccccc4)cc3)coc2c(=O)n1O CHEMBL364591 IC50 0.023 nM
O=c1[nH]c2sccc2c(=O)n1O CHEMBL361350 IC50 0.025 nM
Cc1csc2c1c(=O)n(O)c(=O)n2Cc1ccccc1 CHEMBL181709 IC50 0.028 nM
COc1cccc(-c2coc3c(=O)n(O)c(=O)[nH]c23)c1 CHEMBL185325 IC50 0.031 nM
COc1ccc(-c2coc3c(=O)n(O)c(=O)[nH]c23)cc1 CHEMBL359747 IC50 0.034 nM
COc1ccc(-n2c(=O)n(O)c(=O)c3c(C)csc32)cc1 CHEMBL362205 IC50 0.035 nM
O=c1[nH]c2c(Cc3ccccc3)coc2c(=O)n1O CHEMBL183133 IC50 0.038 nM
O=c1[nH]c2c(sc3ccccc32)c(=O)n1O CHEMBL359533 IC50 0.043 nM
O=c1c2sccc2n(Cc2cccc(Br)c2)c(=O)n1O CHEMBL185322 IC50 0.072 nM
O=c1[nH]c2c(-c3ccc(Br)cc3)coc2c(=O)n1O CHEMBL180566 IC50 0.076 nM
O=c1[nH]c2ccccc2c(=O)n1O CHEMBL183852 IC50 0.079 nM
Cc1ccc(-c2coc3c(=O)n(O)c(=O)[nH]c23)cc1 CHEMBL182381 IC50 0.082 nM
CC(C)(C)c1cc2[nH]c(=O)n(O)c(=O)c2s1 CHEMBL360615 IC50 0.135 nM
O=c1[nH]c2c(-c3ccccc3)coc2c(=O)n1O CHEMBL183539 IC50 0.143 nM
O=c1[nH]c2cc(-c3ccccc3)sc2c(=O)n1O CHEMBL183062 IC50 0.146 nM
O=c1c2ccsc2n(Cc2ccccc2)c(=O)n1O CHEMBL182974 IC50 0.23 nM
O=c1[nH]c2c(oc3ccccc32)c(=O)n1O CHEMBL181766 IC50 0.285 nM
Cc1csc2c1c(=O)n(O)c(=O)n2C CHEMBL181637 IC50 0.338 nM
Cc1csc2c(=O)n(O)c(=O)n(Cc3cccc(-c4ccc(C(N)=O)cc4)c3)c12 CHEMBL181907 IC50 1.08 nM
CC(=O)Nc1cccc2c(=O)n(O)c(=O)[nH]c12 CHEMBL3617199 IC50 38.0 nM
COc1ccc(-c2ccc(Cl)c(C(=O)CC(=O)C(=O)O)c2)cc1 CHEMBL182748 IC50 190.0 nM
O=c1[nH]c2cc(Nc3ccccc3)ccc2c(=O)n1O CHEMBL3617197 IC50 230.0 nM
O=C1c2cccc3cccc(c23)C(=O)N1O CHEMBL1207029 IC50 300.0 nM
O=C(O)C(=O)CC(=O)c1cc(-c2ccccc2)ccc1Cl CHEMBL188067 IC50 330.0 nM
O=C(O)C(=O)CC(=O)c1ccc(-c2ccc(Cl)cc2)cc1Cl CHEMBL183257 IC50 410.0 nM
O=C(O)C(=O)CC(=O)c1ccc(-c2ccc(OC(F)(F)F)cc2)s1 CHEMBL182756 IC50 440.0 nM
O=C(O)C(=O)CC(=O)c1ccc(-c2ccc(Cl)c(F)c2)s1 CHEMBL361960 IC50 570.0 nM
O=c1cc(-c2ccccc2)[nH]c(=O)n1O CHEMBL3617203 IC50 630.0 nM
O=C1c2cccc3c(Cl)ccc(c23)C(=O)N1O CHEMBL1415852 IC50 700.0 nM