C[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4789123 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4762957 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(Cl)c(Cl)c1 CHEMBL4781404 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cccnn3c2=O)cc1Cl CHEMBL4785963 EC50 1.0 nM
Cc1cc([C@H](C)NC(=O)Cn2nc3cccnn3c2=O)ccc1Cl CHEMBL4759611 EC50 1.0 nM
Cc1cc(Cl)ccc1[C@H](C)NC(=O)Cn1nc2cccnn2c1=O CHEMBL4748681 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(Cl)cc1 CHEMBL4786371 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(C2CC2)c(F)c1 CHEMBL4757480 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cccnn3c2=O)cc1F CHEMBL4753587 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(OC(F)(F)F)c(F)c1 CHEMBL4745096 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccc(Cl)nn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4796254 EC50 1.0 nM
Cc1ccc2nn(CC(=O)N[C@@H](C)c3ccc(Cl)cc3)c(=O)n2n1 CHEMBL4792732 EC50 1.0 nM
Cc1cnn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc2c1 CHEMBL4760528 EC50 1.0 nM
Cc1cnn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)nc2c1 CHEMBL4792356 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(Cl)cnn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4754476 EC50 1.0 nM
O=C(Cn1nc2cccnn2c1=O)N[C@H](c1ccc(Cl)c(F)c1)C1CC1 CHEMBL4798509 EC50 1.0 nM
CC[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4762121 EC50 1.0 nM
CC(C)[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4790080 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccc(C3CC3)nn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4750718 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(NC3COC3)ccnn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4746822 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(N3CCOCC3)cnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4740519 EC50 1.0 nM
CC(C(=O)N[C@@H](C)c1ccc(Cl)c(F)c1)n1nc2cccnn2c1=O CHEMBL4740228 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cnccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4746108 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cnc(C)cn3c2=O)cc1 CHEMBL4763362 EC50 1.0 nM
Cc1cn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)nc2cn1 CHEMBL4745668 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(NC3COC3)nccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4757619 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(C(F)F)nccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4783815 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ccncn3c2=O)cc1 CHEMBL4791843 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cc(C)nc(C)n3c2=O)cc1 CHEMBL4754384 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(N3CCNCC3)nccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4756937 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(N3CCN(C)CC3)nccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4745432 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ncccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4787308 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ncccn2c1=O)c1ccc(Cl)c(Cl)c1 CHEMBL4784153 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ncccn3c2=O)cc1Cl CHEMBL4760812 EC50 1.0 nM
Cc1cc(Cl)ccc1[C@H](C)NC(=O)Cn1nc2ncccn2c1=O CHEMBL4744169 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ncccn3c2=O)cc1F CHEMBL4792515 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ncccn2c1=O)c1ccc(OC(F)(F)F)c(F)c1 CHEMBL4757742 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ncccn2c1=O)c1ccc(C2CC2)c(F)c1 CHEMBL4751886 EC50 1.0 nM
Cc1cnc2nn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)c(=O)n2c1 CHEMBL4799144 EC50 1.0 nM
COc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(C)cc3)nc2n1 CHEMBL4751720 EC50 1.0 nM
COc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)cc3)nc2n1 CHEMBL4800487 EC50 1.0 nM
Cc1cnc2nn(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)c(=O)n2c1 CHEMBL4797724 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ncc(F)cn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4747431 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ncc(F)cn2c1=O)c1ccc(Cl)cc1 CHEMBL4749705 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ncc(F)cn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4764666 EC50 1.0 nM
COc1cnc2nn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)c(=O)n2c1 CHEMBL4740491 EC50 1.0 nM
Cc1cnc2nn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)c(F)c3)c(=O)n2c1 CHEMBL4759991 EC50 1.0 nM
Cc1cc(C)n2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)cc3)nc2n1 CHEMBL4793463 EC50 1.0 nM
CC(C(=O)N[C@@H](C)c1ccc(Cl)c(F)c1)n1nc2ncccn2c1=O CHEMBL4757506 EC50 1.0 nM
Cc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)nc2n1 CHEMBL4791551 EC50 1.0 nM
Cc1ccnc2nn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)c(=O)n12 CHEMBL4790498 EC50 1.0 nM
Cc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc2n1 CHEMBL4742901 EC50 1.0 nM
C[C@H](NC(=O)[C@@H](C)n1nc2ncccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4761321 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ccccn3c2=O)cc1 CHEMBL4750143 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4756787 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccccn2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL4762206 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4743612 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccccn2c1=O)c1ccc(OC(F)F)c(F)c1 CHEMBL4753547 EC50 1.0 nM
Cc1cc(Cl)ccc1[C@H](C)NC(=O)Cn1nc2ccccn2c1=O CHEMBL4764290 EC50 1.0 nM
Cc1ncc([C@H](C)NC(=O)Cn2nc3cc(Cl)ccn3c2=O)cc1F CHEMBL4750692 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ccc(Br)cn3c2=O)cc1 CHEMBL4743199 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cccc(Br)n3c2=O)cc1 CHEMBL4741806 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)C(C)n2nc3ccccn3c2=O)cc1 CHEMBL4743938 EC50 1.0 nM
COc1ccc2nn(CC(=O)N[C@@H](C)c3ccc(C)cc3)c(=O)n2c1 CHEMBL4785283 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3c(Cl)cccn3c2=O)cc1 CHEMBL4751203 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3c(F)cccn3c2=O)cc1 CHEMBL4795078 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cccc(F)n3c2=O)cc1 CHEMBL4798029 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccc(F)cn2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL4756137 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(C#N)ccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4751304 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cccc(N3CCN(C)CC3)n2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4751259 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cccc(N3CCN(C)CC3)n2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4742673 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(N3CCOCC3)ccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4786573 EC50 1.0 nM
COC1CCN(c2ccn3c(=O)n(CC(=O)N[C@@H](C)c4ccc(OC(F)(F)F)cc4)nc3c2)CC1 CHEMBL4752993 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(N3CCC[C@@H](O)C3)ccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4744340 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(N3CCC[C@H](O)C3)ccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4754503 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(NC3COC3)ccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4756431 EC50 1.0 nM
CC(C(=O)N[C@@H](C)c1ccc(Cl)c(F)c1)n1nc2ccccn2c1=O CHEMBL4764506 EC50 1.0 nM
CC(NC(=O)Cn1nc2ccccn2c1=O)c1ccc(OC(F)F)cc1 CHEMBL4777673 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3c(N)cccn3c2=O)cc1 CHEMBL4783739 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3c(NC(=O)OC(C)(C)C)cccn3c2=O)cc1 CHEMBL4745487 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(OC3COC3)ccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4758375 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(N3CCC(O)CC3)ccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4764839 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(N3CCC34CNC4)cccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4756392 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(C3CC3)cnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4753640 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(Cl)cnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4765018 EC50 1.0 nM
COc1cnn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc2c1 CHEMBL4762651 EC50 1.0 nM
COc1ccnn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc12 CHEMBL4756356 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(C(F)(F)F)ccnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4791193 EC50 1.0 nM
CNc1ccnn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc12 CHEMBL4748076 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(NCC(F)F)ccnn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4792896 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccc(C3CC3)nn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4756243 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2c(C3CC3)ccnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4754735 EC50 1.0 nM
COc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc2n1 CHEMBL4782901 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ncc(C3CC3)cn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4748306 EC50 1.0 nM
Cc1ccnc2nn(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)c(=O)n12 CHEMBL4789252 EC50 1.0 nM
Cc1cc([C@H](C)NC(=O)Cn2nc3ccccn3c2=O)ccc1Cl CHEMBL4762126 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccccn2c1=O)c1ccc(Cl)c(Cl)c1 CHEMBL4744927 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ccccn3c2=O)cc1Cl CHEMBL4800338 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cc(Cl)ccn3c2=O)cc1 CHEMBL4750914 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ccc(C)cn3c2=O)cc1 CHEMBL4780358 EC50 1.0 nM
Cc1ccc2nn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)c(=O)n2c1 CHEMBL4746401 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccc(F)cn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4753388 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccc(F)cn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4754565 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cc(C)ccn3c2=O)cc1 CHEMBL4743662 EC50 1.0 nM
COc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(C)cc3)nc2c1 CHEMBL4764967 EC50 1.0 nM
COc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)nc2c1 CHEMBL4754576 EC50 1.0 nM
COc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc2c1 CHEMBL4742949 EC50 1.0 nM
Cc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc2c1 CHEMBL4799647 EC50 1.0 nM
Cc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)nc2c1 CHEMBL4786542 EC50 1.0 nM
COc1cccc2nn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)c(=O)n12 CHEMBL4750288 EC50 1.0 nM
COc1cccc2nn(CC(=O)N[C@@H](C)c3ccc(Cl)cc3)c(=O)n12 CHEMBL4790949 EC50 1.0 nM
COc1cccc2nn(CC(=O)N[C@@H](C)c3ccc(C)cc3)c(=O)n12 CHEMBL4798385 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccc(F)cn2c1=O)c1ccc(Cl)cc1 CHEMBL4752808 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2cc(Cl)ccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4761154 EC50 1.0 nM
C[C@H](NC(=O)Cn1nc2ccc(C#N)cn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4751501 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ccc(F)cn3c2=O)cc1F CHEMBL4758841 EC50 1.0 nM
CNc1cccn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(C)cc3)nc12 CHEMBL4793093 EC50 1.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3cccc(C)c3c2=O)cc1 CHEMBL4798933 EC50 6.0 nM
Cc1ccc([C@@H](C)NC(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL4788631 EC50 7.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3c(Cl)cccc3c2=O)cc1 CHEMBL4787761 EC50 7.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3c(Cl)cc(Cl)cc3c2=O)cc1 CHEMBL4784744 EC50 7.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3cc(C)ccc3c2=O)cc1 CHEMBL4789079 EC50 7.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3c(C)cc(C)cc3c2=O)cc1 CHEMBL4777495 EC50 7.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3c(C)cccc3c2=O)cc1 CHEMBL4785669 EC50 8.0 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(Cl)c(F)c1 CHEMBL5401670 pEC50 8.71 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL4798863 EC50 9.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3c(F)cccc3c2=O)cc1 CHEMBL4779481 EC50 9.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3c(C)cccc3c2=O)cc1 CHEMBL4789791 EC50 9.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3cccc(C)c3c2=O)cc1 CHEMBL4792561 EC50 9.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(Br)cc1 CHEMBL4776509 EC50 9.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cccnn3c2=O)cc1 CHEMBL4751629 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2cccnn2c1=O)c1ccc(C2CC2)cc1 CHEMBL4744984 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2ccc(N3CCCCC3)nn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4777046 EC50 10.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3cnccn3c2=O)cc1 CHEMBL4786952 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2ncccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4740004 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2ncccn2c1=O)c1ccc(OC(F)F)c(F)c1 CHEMBL4754933 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2ncccn2c1=O)c1ccc(Cl)cc1 CHEMBL4785855 EC50 10.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ncccn3c2=O)cc1 CHEMBL4750043 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2ccccn2c1=O)c1ccc(F)cc1 CHEMBL4762210 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2ccccn2c1=O)c1ccc(-c2ccccc2)cc1 CHEMBL4781160 EC50 10.0 nM
CC(C)Oc1ccc([C@H](C)NC(=O)Cn2nc3ccccn3c2=O)cc1 CHEMBL4762154 EC50 10.0 nM
O=C(Cn1nc2ccccn2c1=O)NC(c1ccc(Cl)cc1)C1CC1 CHEMBL4761733 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2cc(OC3CN(C)C3)ccn2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4745642 EC50 10.0 nM
O=C(Cn1nc2ccc(F)cn2c1=O)NC1(c2ccc(Cl)cc2)CC1 CHEMBL4787820 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2cccc(N3CCNCC3)n2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4755986 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2c(N3CCC34CN(C)C4)cccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4747632 EC50 10.0 nM
Cc1ccc2nn(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)c(=O)n2n1 CHEMBL4792682 EC50 10.0 nM
Cc1ccnn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)c(F)c3)nc12 CHEMBL4744737 EC50 10.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3c(C)ccnn3c2=O)cc1F CHEMBL4778327 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2c(NC3COC3)ccnn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4777214 EC50 10.0 nM
CNc1ccnn2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)nc12 CHEMBL4752829 EC50 10.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nc3ccc(F)cn3c2=O)cc1 CHEMBL4758561 EC50 10.0 nM
C[C@H](NC(=O)Cn1nc2c(N3CCOCC3)cccn2c1=O)c1ccc(Cl)c(F)c1 CHEMBL4799618 EC50 10.0 nM
COc1ccn2c(=O)n(CC(=O)N[C@@H](C)c3c(C)cc(C)cc3C)nc2c1 CHEMBL4754043 EC50 10.0 nM
COc1ccc2nnn(CC(=O)N[C@@H](C)c3ccc(C)cc3)c(=O)c2c1 CHEMBL4780801 EC50 10.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(C)cc3c2=O)cc1 CHEMBL4786722 EC50 10.0 nM
C[C@H](NC(=O)Cn1nnc2ccc(F)cc2c1=O)c1ccc(OC(F)F)cc1 CHEMBL4782619 EC50 10.0 nM
COc1cccc2nnn(CC(=O)N[C@@H](C)c3ccc(C(F)(F)F)cc3F)c(=O)c12 CHEMBL4799483 Ki 11.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(F)cc3c2=O)cc1 CHEMBL4777630 EC50 11.0 nM
COc1cc(C)ccc1[C@H](C)NC(=O)Cn1nnc2ccccc2c1=O CHEMBL4789631 EC50 11.0 nM
Cc1ccc2cnn(CC(=O)N[C@@H](C)c3ccccc3)c(=O)n12 CHEMBL5407185 pEC50 12.59 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(Cl)cc3c2=O)cc1 CHEMBL4778561 EC50 13.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3c(Cl)cccc3c2=O)cc1 CHEMBL4788831 EC50 13.0 nM
C[C@H](NC(=O)Cn1nnc2ccc(F)cc2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL4797857 EC50 13.0 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(Cl)c(Cl)c1 CHEMBL5435834 pEC50 13.49 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(F)cc1Cl CHEMBL4792090 EC50 14.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccccc3c2=O)c(C)c1 CHEMBL4781729 EC50 15.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(C(F)(F)F)cc3c2=O)cc1 CHEMBL4792828 EC50 15.0 nM
COc1cccc2nnn(CC(=O)N[C@@H](C)c3ccc(C(F)(F)F)cc3)c(=O)c12 CHEMBL4789720 EC50 15.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3c(F)cc(C)cc3c2=O)cc1 CHEMBL4797410 EC50 15.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL4779855 EC50 15.0 nM
C[C@H](NC(=O)CNC(=O)c1cccc(Cl)c1)c1ccccc1 CHEMBL3633720 EC50 16.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(F)cc3c2=O)cc1 CHEMBL4795372 EC50 16.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(Cl)cc3c2=O)cc1 CHEMBL4796061 EC50 16.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3c(Cl)cc(Cl)cc3c2=O)cc1 CHEMBL4780038 EC50 16.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3cccc(F)c3c2=O)cc1 CHEMBL4778563 EC50 16.0 nM
COc1cc(C)ccc1[C@H](C)NC(=O)[C@@H](C)n1nnc2ccccc2c1=O CHEMBL4786501 EC50 16.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3cc(Cl)ccc3c2=O)cc1 CHEMBL4778124 EC50 17.0 nM
COc1cccc2nnn(CC(=O)N[C@@H](C)c3ccc(OC(F)F)cc3)c(=O)c12 CHEMBL4783626 EC50 17.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2ncc3sccc3c2=O)cc1 CHEMBL5410300 pEC50 17.78 nM
COc1ccc2nnn(CC(=O)N[C@@H](C)c3ccc(C(F)(F)F)cc3)c(=O)c2c1 CHEMBL4794046 EC50 18.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(OC(F)F)cc1 CHEMBL4790968 EC50 18.0 nM
Cc1ccc2cnn(CC(=O)N[C@@H](C)c3ccc(Br)cc3)c(=O)n12 CHEMBL5438556 pEC50 18.2 nM
Cc1ccc2cnn(CC(=O)N[C@@H](C)c3ccc(F)cc3)c(=O)n12 CHEMBL5417840 pEC50 18.62 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(C)cc3c2=O)cc1 CHEMBL4781651 EC50 19.0 nM
COc1ccc2c(=O)n(CC(=O)N[C@@H](C)c3ccc(C)cc3)nnc2c1 CHEMBL4783071 EC50 19.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(C(F)(F)F)cc1F CHEMBL4791792 EC50 19.0 nM
Cc1cc(C)n2c(=O)n(CC(=O)N[C@@H](C)c3ccccc3)ncc12 CHEMBL5432850 pEC50 19.05 nM
Cc1ccc([C@H](C)NC(=O)Cn2ncc3ccc(C)n3c2=O)cc1 CHEMBL5394347 pEC50 19.5 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(Br)cc1 CHEMBL5403952 pEC50 20.89 nM
O=C(Cn1nnc2ccccc2c1=O)NCCc1ccc(Cl)cc1 CHEMBL4871792 EC50 21.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3sccc3c2=O)cc1 CHEMBL5417548 pEC50 21.38 nM
CC[C@H](NC(=O)Cn1ncc2ccc(C)n2c1=O)c1ccccc1 CHEMBL5411110 pEC50 21.38 nM
C[C@H](NC(=O)Cn1nnc2sccc2c1=O)c1ccc(Cl)cc1 CHEMBL5394715 pEC50 21.88 nM
Cc1ccc2cnn(CC(=O)N[C@@H](C)c3ccc(Cl)cc3)c(=O)n12 CHEMBL5438741 pEC50 21.88 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4779773 EC50 22.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(F)cc1 CHEMBL4792727 EC50 22.0 nM
COc1cccc2nnn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)c(=O)c12 CHEMBL4796493 EC50 22.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(Cl)cc1 CHEMBL4798779 EC50 22.0 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(F)cc1Cl CHEMBL5433281 pEC50 22.39 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(Cl)cc1 CHEMBL5409401 pEC50 22.91 nM
COc1ccc([C@H](C)NC(=O)Cn2ncc3ccc(C)n3c2=O)cc1 CHEMBL5432364 pEC50 23.44 nM
C[C@H](NC(=O)CNC(=O)c1cc(F)cc(Cl)c1)c1ccccc1 CHEMBL3633888 EC50 24.0 nM
Cc1cccc(C(=O)NCC(=O)N[C@@H](C)c2ccccc2)c1 CHEMBL3633878 EC50 24.0 nM
COc1cccc2nnn(CC(=O)N[C@@H](C)c3ccc(C)cc3)c(=O)c12 CHEMBL4778172 EC50 24.0 nM
CCOc1ccc([C@H](C)NC(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL4783081 EC50 24.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(F)cc3c2=O)c(C)c1 CHEMBL4776329 EC50 24.0 nM
Cc1ccccc1[C@H](C)NC(=O)Cn1nnc2ccccc2c1=O CHEMBL4799237 EC50 24.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccccc3c2=O)c(F)c1 CHEMBL4789475 EC50 24.0 nM
CC[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(C)cc1 CHEMBL4869182 EC50 24.0 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(F)c(F)c1 CHEMBL5426183 pEC50 24.55 nM
COc1cccc2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)nnc12 CHEMBL4779884 EC50 25.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3cccc(OC)c3c2=O)cc1 CHEMBL4794908 EC50 26.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3c(F)cccc3c2=O)cc1 CHEMBL4778062 EC50 27.0 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1cccc2ccccc12 CHEMBL5399140 pEC50 27.54 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(F)cc1F CHEMBL5420577 pEC50 27.54 nM
Cc1ccc([C@H](C)NC(=O)Cn2ncc3cccn3c2=O)cc1 CHEMBL5402898 pEC50 27.54 nM
C[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1cccc2ccccc12 CHEMBL5421824 pEC50 27.54 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL5406603 pEC50 28.18 nM
C[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1ccc(Cl)cc1 CHEMBL5397779 pEC50 28.18 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(OC(F)(F)F)cc1F CHEMBL4785741 EC50 29.0 nM
COc1cccc2c(=O)n(CC(=O)N[C@@H](C)c3ccc(C)cc3)nnc12 CHEMBL4783106 EC50 30.0 nM
Cc1ccc(CCNC(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL4875522 EC50 30.0 nM
Cc1ccc([C@H](C)NC(=O)C(C)n2nnc3ccccc3c2=O)cc1 CHEMBL4847108 EC50 30.0 nM
Cc1ccc2cnn(CC(=O)N[C@H](c3ccc(F)cc3)C(C)C)c(=O)n12 CHEMBL5418368 pEC50 30.9 nM
CC[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL4781754 EC50 31.0 nM
C[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1ccc(Br)cc1 CHEMBL5421380 pEC50 31.62 nM
COc1cc(OC)cc(C(=O)NCC(=O)N[C@@H](C)c2ccccc2)c1 CHEMBL3633890 EC50 32.0 nM
COc1cccc(C(=O)NCC(=O)N[C@@H](C)c2ccccc2)c1 CHEMBL3633881 EC50 33.0 nM
COc1cccc2nnn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3F)c(=O)c12 CHEMBL4782204 Ki 33.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL4798667 EC50 33.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1cccc2ccccc12 CHEMBL4874147 EC50 33.0 nM
COc1ccc([C@H](C)NC(=O)Cn2ncc3c(C)cc(C)n3c2=O)cc1 CHEMBL5403066 pEC50 33.11 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(Cl)cc1Cl CHEMBL5437907 pEC50 34.67 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3c(C)cc(C)cc3c2=O)cc1 CHEMBL4795005 EC50 37.0 nM
COc1ccc2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)nnc2c1 CHEMBL4778354 EC50 37.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(C(F)(F)F)cc3c2=O)cc1 CHEMBL4797979 EC50 37.0 nM
C[C@H](NC(=O)Cn1nnc2ccc(F)cc2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4776988 EC50 38.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3c(OC)cccc3c2=O)cc1 CHEMBL4783544 EC50 39.0 nM
C[C@H](NC(=O)CNC(=O)c1cc(Cl)ccc1Cl)c1ccccc1 CHEMBL3633886 EC50 40.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3cccc(F)c3c2=O)cc1 CHEMBL4792174 EC50 41.0 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(F)cc1 CHEMBL5431491 pEC50 41.69 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3cc(C)ccc3c2=O)cc1 CHEMBL4783774 EC50 42.0 nM
COc1cc(OC)cc(C(=O)NNC(=O)Nc2cccc3ccccc23)c1 CHEMBL3633893 EC50 43.0 nM
COc1ccc2nnn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)c(=O)c2c1 CHEMBL4788013 EC50 43.0 nM
Cc1ccc2cnn(CC(=O)N[C@@H](C)c3cccc4ccccc34)c(=O)n12 CHEMBL5395065 pEC50 44.67 nM
C[C@H](NC(=O)CNC(=O)c1cc(Cl)cc(Cl)c1)c1ccccc1 CHEMBL3633887 EC50 46.0 nM
C[C@H](NC(=O)CNC(=O)c1cccc(OC(F)(F)F)c1)c1ccccc1 CHEMBL3633883 EC50 46.0 nM
COc1ccc(CCNC(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL1380104 EC50 46.0 nM
C[C@H](NC(=O)Cn1nnc2sccc2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL5438241 pEC50 46.77 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3sccc3c2=O)cc1 CHEMBL5433669 pEC50 46.77 nM
CC[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1ccccc1 CHEMBL5418797 pEC50 48.98 nM
C[C@H](NC(=O)Cn1nnc2ccc(F)cc2c1=O)c1ccc(OC(F)(F)F)cc1F CHEMBL4780121 EC50 49.0 nM
COc1cccc2c(=O)n(CC(=O)N[C@@H](C)c3ccc(C(F)(F)F)cc3)nnc12 CHEMBL4781805 EC50 50.0 nM
CC[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(OC(F)(F)F)cc1 CHEMBL4783365 EC50 50.0 nM
COc1ccc2c(=O)n(CC(=O)N[C@@H](C)c3ccc(C(F)(F)F)cc3)nnc2c1 CHEMBL4785980 EC50 51.0 nM
COc1ccc([C@H](C)NC(=O)Cn2ncc3sccc3c2=O)cc1 CHEMBL5394251 pEC50 51.29 nM
C[C@H](NC(=O)CNC(=O)c1cccc(Cl)c1Cl)c1ccccc1 CHEMBL3633884 EC50 52.0 nM
C[C@H](NC(=O)CNC(=O)c1cccc(C(F)(F)F)c1)c1ccccc1 CHEMBL3633882 EC50 52.0 nM
COc1cc(C)ccc1[C@H](C)NC(=O)[C@H](C)n1nnc2ccccc2c1=O CHEMBL4778263 EC50 52.0 nM
CC[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccccc1 CHEMBL5435044 pEC50 52.48 nM
Cc1cc(C)n2c(=O)n(CC(=O)N[C@@H](C)c3ccc(Cl)cc3)ncc12 CHEMBL5394567 pEC50 53.7 nM
C[C@H](NC(=O)CNC(=O)c1cccc(F)c1)c1ccccc1 CHEMBL3633880 EC50 54.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccccc1 CHEMBL4786641 EC50 54.0 nM
COc1ccc(C[C@H](C)NC(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL4873905 EC50 54.0 nM
C[C@@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccccc1 CHEMBL4861019 EC50 54.0 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccccc1 CHEMBL5408151 EC50 54.8 nM
C[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1ccc(F)cc1 CHEMBL5397321 pEC50 54.95 nM
C[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL5427962 pEC50 54.95 nM
C[C@H](NC(=O)Cn1nnc2sccc2c1=O)c1ccc(F)cc1 CHEMBL5435655 pEC50 56.23 nM
Cc1ccc2cnn(CC(=O)N[C@@H](C)c3ccc(C(F)(F)F)cc3)c(=O)n12 CHEMBL5429215 pEC50 56.23 nM
COc1ccc([C@H](C)NC(=O)Cn2ncc3cccn3c2=O)cc1 CHEMBL5417091 pEC50 58.88 nM
CC(C)[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1ccccc1 CHEMBL5419423 pEC50 58.88 nM
C[C@H](NC(=O)CNC(=O)c1cccc(C#N)c1)c1ccccc1 CHEMBL3633879 EC50 59.0 nM
O=C(Cn1nnc2ccccc2c1=O)NCCc1cccc(Cl)c1 CHEMBL4861445 EC50 65.0 nM
COc1cccc(C(=O)N[C@@H](C)C(=O)N[C@@H](C)c2ccccc2)c1 CHEMBL3633714 EC50 66.0 nM
O=C(Cn1nnc2ccccc2c1=O)NC1CCCc2ccccc21 CHEMBL1460960 EC50 66.0 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3ccccc3c2=O)c(OC)c1 CHEMBL4792136 EC50 67.0 nM
O=C(Cn1nnc2ccccc2c1=O)NCCc1ccccc1Cl CHEMBL4866435 EC50 68.0 nM
CC(C)[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccccc1 CHEMBL5396468 pEC50 69.18 nM
COc1ccc([C@H](C)NC(=O)Cn2nnc3cc(OC)ccc3c2=O)cc1 CHEMBL4800089 EC50 70.0 nM
CC(C)[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL5409522 pEC50 72.44 nM
Cc1ccc2cnn(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)c(=O)n12 CHEMBL5395516 pEC50 74.13 nM
Cc1ccc([C@H](C)NC(=O)Cn2nnc3ccc(F)cc3c2=O)c(F)c1 CHEMBL4791752 Ki 77.0 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(C(F)(F)F)nc1 CHEMBL4855076 EC50 77.0 nM
C[C@H](NC(=O)CNC(=O)c1cc(Cl)cc(Br)c1)c1ccccc1 CHEMBL3633889 EC50 78.0 nM
CC(NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(Cl)cc1 CHEMBL4860510 EC50 79.0 nM
CC(C)[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1ccc(C(F)(F)F)cc1 CHEMBL5421234 pEC50 83.18 nM
O=C(Cn1nnc2ccccc2c1=O)NCCc1ccc(-c2ccccc2)cc1 CHEMBL4869485 EC50 85.0 nM
Cc1ccc([C@H](C)NC(=O)Cn2ncc3c(C)cc(C)n3c2=O)cc1 CHEMBL5399292 pEC50 89.13 nM
COc1ccc([C@H](C)NC(=O)C(C)n2nnc3ccccc3c2=O)cc1 CHEMBL4871506 EC50 90.0 nM
Cc1cc(C)n2c(=O)n(CC(=O)N[C@@H](C)c3ccc(OC(F)(F)F)cc3)ncc12 CHEMBL5404791 pEC50 93.33 nM
Cc1cc(C)n2c(=O)n(CC(=O)N[C@@H](C)c3ccc(F)cc3)ncc12 CHEMBL5411677 pEC50 93.33 nM
CC(C)[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(F)cc1 CHEMBL5401884 pEC50 109.65 nM
Cc1cccc([C@H](C)NC(=O)Cn2nnc3ccccc3c2=O)c1 CHEMBL4874254 EC50 110.0 nM
C[C@H](NC(=O)Cn1ncc2cccn2c1=O)c1ccccc1 CHEMBL5413318 EC50 111.0 nM
C[C@H](NC(=O)CNC(=O)c1ccc(Cl)cc1)c1ccccc1 CHEMBL3633721 EC50 118.0 nM
Cc1ccc([C@H](C)OC(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL4871591 EC50 119.0 nM
C[C@H](NC(=O)CNC(=O)c1ccccc1Cl)c1ccccc1 CHEMBL3633719 EC50 150.0 nM
Cc1ccc2cnn(CC(=O)N[C@H](c3ccc(C(F)(F)F)cc3)C(C)C)c(=O)n12 CHEMBL5436077 pEC50 158.49 nM
C[C@H](NC(=O)Cn1nnc2ccccc2c1=O)c1ccc(C(F)(F)F)cn1 CHEMBL4857947 EC50 159.0 nM
C[C@H](NC(=O)CNC(=O)c1ccccc1)c1ccccc1 CHEMBL3633718 EC50 162.0 nM
C[C@H](NC(=O)CNC(=O)c1ccc(Cl)c(Cl)c1)c1ccccc1 CHEMBL3633885 EC50 193.0 nM
C[C@H](NC(=O)Cn1ncc2sccc2c1=O)c1ccc(C#N)cc1 CHEMBL5412645 pEC50 269.15 nM
COc1cccc(C(=O)N[C@@H](CO)C(=O)N[C@@H](C)c2ccccc2)c1 CHEMBL3633716 EC50 283.0 nM
C[C@@H](CNC(=O)Cn1nnc2ccccc2c1=O)c1ccccc1 CHEMBL4850747 EC50 288.0 nM
O=C(Cn1nnc2ccccc2c1=O)NCc1ccc(Cl)cc1 CHEMBL1546963 EC50 293.0 nM
COc1cccc(C(=O)N[C@H](C)C(=O)N[C@@H](C)c2ccccc2)c1 CHEMBL3633715 EC50 440.0 nM
CC(NC(=O)CSC(=O)c1ccccc1)c1ccccc1 CHEMBL3633894 EC50 670.0 nM
COc1ccc([C@H](C)NS(=O)(=O)Cn2nnc3ccccc3c2=O)cc1 CHEMBL4847795 EC50 714.0 nM