C[C@H](CCCC(C)(C)O)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C CHEMBL4788348 EC50 0.032 nM
C[C@H](CCCC(C)(C)O)[C@H]1CC[C@H]2[C@H]3[C@H](CC[C@]12C)[C@@]1(C)CC[C@H](O)CC1=C[C@]3(O)C(F)(F)F CHEMBL4779254 EC50 0.102 nM
COc1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cc1 CHEMBL3262896 pIC50 0.2239 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 CHEMBL3560809 IC50 0.409 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)c2ccccc2)CC1 CHEMBL3560864 IC50 0.62 nM
Cc1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cc1 CHEMBL3560888 IC50 1.02 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2ccc(Cl)cc2)CC1 CHEMBL3560331 IC50 1.03 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)C2=Cc3ccccc3CC2)CC1 CHEMBL3560117 IC50 1.15 nM
O=C(/C=C/c1ccc(Cl)c(Cl)c1)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 CHEMBL3561364 IC50 1.17 nM
CC(CO)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C CHEMBL4788277 EC50 1.3 nM
Cc1cc(CN2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)ccc1F CHEMBL3561756 IC50 1.5 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1 CHEMBL3561399 IC50 1.66 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2ccc(Cl)c(Cl)c2)CC1 CHEMBL3560041 IC50 1.72 nM
N#Cc1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cc1 CHEMBL3560453 IC50 1.74 nM
Cc1ccc(CN2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cc1 CHEMBL3561255 IC50 1.77 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 CHEMBL3560732 IC50 1.88 nM
CCCCN1CCN(C(=O)/C=C/c2ccc(Br)cc2)CC1 CHEMBL3560464 IC50 2.1 nM
C[C@H](CCCC(C)(C)O)[C@H]1CC[C@H]2[C@@H]3[C@@H](O)C=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C CHEMBL3311219 EC50 2.1 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2cc(F)cc(F)c2)CC1 CHEMBL3560573 IC50 2.21 nM
CCC(C)N1CCN(C(=O)/C=C/c2ccc(Br)cc2)CC1 CHEMBL3561798 IC50 2.23 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2cccc(F)c2)CC1 CHEMBL3560897 IC50 2.61 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2ccccc2)CC1 CHEMBL1704801 IC50 2.8 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)CCc2ccccc2)CC1 CHEMBL3560820 IC50 3.27 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1 CHEMBL3561859 IC50 3.43 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1 CHEMBL1580410 IC50 3.59 nM
COc1cc(CN2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cc(OC)c1 CHEMBL3560415 IC50 3.64 nM
C[C@H](CCCC(C)(C)O)[C@H]1CC[C@H]2[C@H]3[C@H](CC[C@]12C)[C@@]1(C)CC[C@H](O)CC1=C[C@@]3(O)C(F)(F)F CHEMBL4757291 EC50 4.1 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)C2CCCC2)CC1 CHEMBL3560365 IC50 4.41 nM
O=C(COc1ccc2ccccc2c1)N1CCN(C(=O)Cc2ccccc2)CC1 CHEMBL3262876 pIC50 4.898 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)c2ccc3c(c2)CCO3)CC1 CHEMBL3262895 IC50 5.0 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2ccc(Cl)cc2C(F)(F)F)CC1 CHEMBL3561495 IC50 5.23 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 CHEMBL3561390 IC50 5.48 nM
CCCCC(=O)N1CCN(C(=O)/C=C/c2ccc(Br)cc2)CC1 CHEMBL3561208 IC50 5.62 nM
CC(C)c1ccc(CN2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cc1 CHEMBL3561719 IC50 5.92 nM
Cc1cc(C)cc(CN2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)c1 CHEMBL3559986 IC50 6.4 nM
Cc1ccc(S(=O)(=O)N2CCN(C(=O)/C=C/c3ccc(F)cc3)CC2)cc1 CHEMBL3559987 IC50 7.67 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2ccccc2Br)CC1 CHEMBL3560529 IC50 8.01 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2ccc(Cl)cc2F)CC1 CHEMBL3561484 IC50 8.11 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2ccc(F)cc2C(F)(F)F)CC1 CHEMBL3561739 IC50 8.18 nM
CC(C)(C)c1ccc(CN2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cc1 CHEMBL3559757 IC50 9.36 nM
COc1ccc(/C=C/C(=O)N2CCN(S(=O)(=O)c3ccc(Br)cc3)CC2)cc1 CHEMBL3561084 IC50 9.58 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2cccc(Cl)c2)CC1 CHEMBL3560763 IC50 11.5 nM
COc1ccc(S(=O)(=O)N2CCN(C(=O)/C=C/c3ccc(F)cc3)CC2)cc1 CHEMBL3560467 IC50 12.1 nM
CC(C)(C)c1ccc(S(=O)(=O)N2CCN(C(=O)/C=C/c3ccc(F)cc3)CC2)cc1 CHEMBL3560404 IC50 12.4 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2ccccc2)CC1 CHEMBL3559792 IC50 12.5 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3ccc(Cl)c(C)c3)CC2)cc1 CHEMBL3262892 pIC50 12.88 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2ccc([N+](=O)[O-])cc2)CC1 CHEMBL3560431 IC50 12.9 nM
CC(C)(C)c1ccc(CSc2cnn(C(C)(C)C)c(=O)c2Cl)cc1 CHEMBL225963 IC50 13.85 nM
O=C(/C=C/c1ccc(Cl)c(Cl)c1)N1CCN(Cc2ccc(Cl)cc2)CC1 CHEMBL3559855 IC50 14.3 nM
CCOc1ccc(/C=C/C(=O)N2CCN(S(=O)(=O)c3ccc(Br)cc3)CC2)cc1 CHEMBL3561444 IC50 14.3 nM
CCN1CCN(C(=O)/C=C/c2ccc(Br)cc2)CC1 CHEMBL3560691 IC50 15.8 nM
O=C(/C=C/c1ccc(Cl)cc1)N1CCN(C(=O)c2ccc3c(c2)CCO3)CC1 CHEMBL3262894 pIC50 15.85 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)c2ccc3occc3c2)CC1 CHEMBL5401247 IC50 16.0 nM
Cc1ccc(/C=C/C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1F CHEMBL3262883 pIC50 16.98 nM
COC(=O)c1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc(OC)cc3)CC2)cc1 CHEMBL3262890 pIC50 16.98 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2cccc(Br)c2)CC1 CHEMBL3560750 IC50 17.5 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3ccc4c(c3)CCO4)CC2)cc1 CHEMBL3262891 IC50 18.0 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2ccc(F)cc2)CC1 CHEMBL3560941 IC50 18.5 nM
Cc1ccc(/C=C/C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1 CHEMBL3262880 IC50 19.0 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3ccc(N(C)C)cc3)CC2)cc1 CHEMBL3262889 IC50 19.0 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2ccccc2F)CC1 CHEMBL3559845 IC50 19.4 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2cccc(F)c2)CC1 CHEMBL3561498 IC50 19.6 nM
COc1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc4c(c3)OC(F)(F)O4)CC2)cn1 CHEMBL5421607 IC50 20.7 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)Cc2ccccc2)CC1 CHEMBL3262879 pIC50 20.89 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1 CHEMBL3560607 IC50 21.2 nM
O=C(/C=C/c1ccccc1)N1CCN(Cc2ccc(F)cc2)CC1 CHEMBL3561640 IC50 21.6 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2cc(Cl)ccc2Cl)CC1 CHEMBL3561698 IC50 21.9 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2ccc3[nH]ncc3c2)CC1 CHEMBL5424378 IC50 22.0 nM
O=C(/C=C/c1ccc(Cl)c(Cl)c1)N1CCN(C(=O)Cc2ccccc2)CC1 CHEMBL3262882 pIC50 23.99 nM
CCCc1ccc(S(=O)(=O)N2CCN(C(=O)/C=C/c3ccc(F)cc3)CC2)cc1 CHEMBL3561833 IC50 24.1 nM
CC(C)c1ccc(S(=O)(=O)N2CCN(C(=O)/C=C/c3ccc(F)cc3)CC2)cc1 CHEMBL3560877 IC50 24.3 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)N2CCC2)CC1 CHEMBL5406913 IC50 25.7 nM
O=C(COc1ccc(Br)cc1)N1CCN(C(=O)Cc2ccccc2)CC1 CHEMBL3262877 IC50 28.0 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)Cc2ccccc2)CC1 CHEMBL3560082 IC50 28.7 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)c2cccc(B(O)O)c2)CC1 CHEMBL3560195 IC50 28.7 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(Cc2ccccc2F)CC1 CHEMBL3560274 IC50 28.7 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1 CHEMBL3262881 pIC50 28.84 nM
COc1ncc(C(=O)N2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cn1 CHEMBL5399120 IC50 29.4 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3cccc(C)c3)CC2)cc1 CHEMBL3262884 pIC50 29.51 nM
COc1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cn1 CHEMBL5395781 IC50 30.0 nM
COc1ncc(C(=O)N2CCN(C(=O)/C=C/c3ccc4c(c3)OC(F)(F)O4)CC2)cn1 CHEMBL5394700 IC50 31.3 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3ccc(OC)cc3)CC2)cc1 CHEMBL3262888 IC50 32.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)OC2CC2)CC1 CHEMBL5405057 IC50 33.3 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)C2CCOCC2)CC1 CHEMBL5414588 IC50 39.0 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3ccc(C)cc3)CC2)cc1 CHEMBL3262887 pIC50 39.81 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3ccc(C)c(C)c3)CC2)cc1 CHEMBL3262893 pIC50 43.65 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cnc3c(c2)OCCO3)CC1 CHEMBL5439756 IC50 45.1 nM
CC(C)(C)c1ccc(S(=O)(=O)N2CCN(C(=O)/C=C/c3ccc(Cl)c(Cl)c3)CC2)cc1 CHEMBL3560209 IC50 46.8 nM
N#Cc1ccccc1S(=O)(=O)N1CCN(C(=O)/C=C/c2ccc(F)cc2)CC1 CHEMBL3560541 IC50 48.2 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2cccc3ccccc23)CC1 CHEMBL3559902 IC50 49.7 nM
CC(CO)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3[C@@H](O)C=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C CHEMBL4776911 EC50 51.0 nM
COc1cccc(S(=O)(=O)N2CCN(C(=O)/C=C/c3ccc(F)cc3)CC2)c1 CHEMBL3561230 IC50 52.1 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cncnc2)CC1 CHEMBL5397313 IC50 52.4 nM
COc1ccc(C(=O)N2CCCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cn1 CHEMBL5402356 IC50 54.6 nM
CC(C)(C)C(O)C(=O)N1CCN(C(=O)/C=C/c2ccc3c(c2)OC(F)(F)O3)CC1 CHEMBL5412445 IC50 58.0 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)c2ccc3[nH]ccc3c2)CC1 CHEMBL5438584 IC50 60.5 nM
CC(C)(O)C(=O)N1CCN(C(=O)/C=C/c2ccc3c(c2)OC(F)(F)O3)CC1 CHEMBL5400278 IC50 65.0 nM
O=C(/C=C/c1ccc(Br)cc1F)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1 CHEMBL3559896 IC50 65.5 nM
COCCOc1ncc(C(=O)N2CCN(C(=O)/C=C/c3ccc4c(c3)OC(F)(F)O4)CC2)cn1 CHEMBL5395361 IC50 66.0 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3ccc(Br)cc3)CC2)cc1 CHEMBL3262886 pIC50 67.61 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cnc3[nH]ncc3c2)CC1 CHEMBL5400459 IC50 70.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cnc(C(F)(F)F)nc2)CC1 CHEMBL5395357 IC50 70.1 nM
O=C(/C=C/c1ccc(F)cc1)N1CCN(S(=O)(=O)c2cccs2)CC1 CHEMBL3560506 IC50 81.0 nM
COc1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2C)cn1 CHEMBL5405959 IC50 81.8 nM
COc1ccc(/C=C/C(=O)N2CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)cc1 CHEMBL3262885 pIC50 97.72 nM
O=C(/C=C/c1ccccc1)N1CCN(Cc2ccc(Cl)cc2)CC1 CHEMBL3561800 IC50 98.4 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cnc3[nH]ccc3c2)CC1 CHEMBL5431534 IC50 103.0 nM
CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3[C@H](O)C=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C CHEMBL497207 EC50 104.88 nM
Cc1ncc(C(=O)N2CCN(C(=O)/C=C/c3ccc4c(c3)OC(F)(F)O4)CC2)cn1 CHEMBL5435007 IC50 105.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)C2(c3ccccc3)CC2)CC1 CHEMBL5430675 IC50 110.0 nM
O=C(CCc1ccc(F)cc1)N1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1 CHEMBL3559877 IC50 113.0 nM
COc1ccc(C(=O)N2CC3(CN(C(=O)/C=C/c4ccc(Br)cc4)C3)C2)cn1 CHEMBL5425366 IC50 122.8 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cnc(N3CCC3)nc2)CC1 CHEMBL5425720 IC50 129.0 nM
COc1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc4c(c3)OC(F)(F)O4)CC2)nc1 CHEMBL5413510 IC50 131.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cnc(OC3CCOCC3)nc2)CC1 CHEMBL5422521 IC50 135.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cnc(OC3CCCC3)nc2)CC1 CHEMBL5395113 IC50 158.0 nM
O=C(/C=C/c1ccc(Cl)cc1F)N1CCN(S(=O)(=O)c2ccccc2)CC1 CHEMBL3561595 IC50 184.0 nM
Cc1ccccc1/C=C/C(=O)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1 CHEMBL3559978 IC50 187.0 nM
CC(C(=O)N1CCN(C(=O)/C=C/c2ccc3c(c2)OC(F)(F)O3)CC1)C1COC1 CHEMBL5412345 IC50 200.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)c2cnc(N3CC[C@H](O)C3)nc2)CC1 CHEMBL5423746 IC50 207.0 nM
O=C(/C=C/c1ccc(Br)cc1)N1CCN(C(=O)c2ccc3[nH]cnc3c2)CC1 CHEMBL5394888 IC50 214.0 nM
COc1ccc(C(=O)N2CCN(C(=O)CCc3ccc(Br)cc3)CC2)cn1 CHEMBL5402708 IC50 221.0 nM
COC1CC(C(=O)N2CCN(C(=O)/C=C/c3ccc4c(c3)OC(F)(F)O4)CC2)C1 CHEMBL5423491 IC50 225.0 nM
COc1cnc(C(=O)N2CCN(C(=O)/C=C/c3ccc4c(c3)OC(F)(F)O4)CC2)cn1 CHEMBL5416074 IC50 230.0 nM
O=C(/C=C/c1ccccc1F)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1 CHEMBL3561130 IC50 252.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)N2CCOCC2)CC1 CHEMBL5415152 IC50 253.0 nM
O=C(COc1ccc(Cl)cc1)N1CCN(C(=O)Cc2ccccc2)CC1 CHEMBL1305842 pIC50 309.03 nM
O=C(/C=C/c1ccccc1C(F)(F)F)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1 CHEMBL3561867 IC50 310.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)C2COC2)CC1 CHEMBL5400812 IC50 354.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)N2CC3(CC(O)C3)C2)CC1 CHEMBL5432988 IC50 439.0 nM
O=C(/C=C/c1ccc2c(c1)OC(F)(F)O2)N1CCN(C(=O)C2CCOCC2)CC1 CHEMBL5419703 IC50 467.0 nM
O=C(c1ccc(Br)cc1)N1CCN(Cc2ccc(Cl)cc2)CC1 CHEMBL3561875 IC50 478.0 nM
COc1ccc(C(=O)N2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC23CC3)cn1 CHEMBL5434815 IC50 498.0 nM
COc1ccc(C(=O)N2CCN(C(=O)/C=C(\C)c3ccc(Br)cc3)CC2)cn1 CHEMBL5426423 IC50 562.0 nM
Cc1ccccc1C#Cc1ccc(CCC(=O)O)cc1 CHEMBL449588 IC50 582.5 nM
O=C(/C=C/c1ccccc1)N1CCN(S(=O)(=O)c2ccc(F)cc2)CC1 CHEMBL1557734 IC50 626.0 nM
Cn1cnc(C(=O)N2CCN(C(=O)/C=C/c3ccc4c(c3)OC(F)(F)O4)CC2)c1 CHEMBL5413214 IC50 739.0 nM
O=C(/C=C/c1cc(Br)ccc1F)N1CCN(S(=O)(=O)c2ccc(Br)cc2)CC1 CHEMBL3560891 IC50 743.0 nM
COc1ccc(C(=O)NC2CCN(C(=O)/C=C/c3ccc(Br)cc3)CC2)cn1 CHEMBL5411108 IC50 865.0 nM