Cc1ccccc1C#Cc1ccc(CCC(=O)O)cc1 CHEMBL449588 IC50 364.84 nM
O=C(Nc1ccc(Cl)c(Cl)n1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5417806 IC50 500.0 nM
O=C(Nc1ccc(Oc2ccccc2)nc1)N1C2CCC1c1ccnc(F)c1C2 CHEMBL5420624 IC50 500.0 nM
O=C(Nc1cnc(Cl)c(Cl)c1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5427600 IC50 500.0 nM
O=C(Nc1cc(C(F)(F)F)ncc1F)N1[C@H]2CC[C@@H]1c1c[nH]c(=O)cc1C2 CHEMBL5404390 IC50 500.0 nM
O=C(Nc1cnc(-n2nccn2)c(Cl)c1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5437369 IC50 500.0 nM
O=C(Nc1cnc(Cl)cc1F)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5422604 IC50 500.0 nM
O=C(Nc1cc(C(F)(F)F)ncc1F)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5424723 IC50 500.0 nM
O=C(Nc1nc(Cl)c(Cl)cc1F)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5421727 IC50 500.0 nM
Cc1nonc1NC(=O)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5437775 IC50 500.0 nM
O=C(Nc1nnc(-c2ccncc2)s1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5406392 IC50 500.0 nM
O=C(Nc1ncc(C(F)(F)F)cn1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5398106 IC50 500.0 nM
CCc1nnc(NC(=O)N2[C@H]3CC[C@@H]2c2ccnc(F)c2C3)s1 CHEMBL5406035 IC50 500.0 nM
O=C(Nc1cc(Cl)c(C(F)(F)F)cn1)N1C2CCC1c1cncnc1C2 CHEMBL5400228 IC50 500.0 nM
O=C(Nc1nnc(C2CC2)s1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5431825 IC50 500.0 nM
O=C(Nc1ccc2nonc2c1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5433744 IC50 500.0 nM
N#Cc1ccc(NC(=O)N2[C@H]3CC[C@@H]2c2ccnc(F)c2C3)nc1C(F)(F)F CHEMBL5400100 IC50 500.0 nM
O=C(Nc1ccc(OC(F)F)cn1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5402018 IC50 500.0 nM
N#Cc1ccc(NC(=O)N2[C@H]3CC[C@@H]2c2ccnc(F)c2C3)nc1 CHEMBL5413335 IC50 500.0 nM
O=C(Nc1nc(-c2ccccc2)no1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5403385 IC50 500.0 nM
O=C(Nc1nnc(-c2ccccc2)o1)N1[C@H]2CC[C@@H]1c1ccnc(F)c1C2 CHEMBL5407784 IC50 500.0 nM
N#Cc1ccc(NC(=O)N2[C@H]3CC[C@@H]2c2ccnc(F)c2C3)nc1Cl CHEMBL5435598 IC50 500.0 nM
COC(=O)c1cc(NC(=O)N2[C@H]3CC[C@@H]2c2ccnc(F)c2C3)no1 CHEMBL5440522 IC50 500.0 nM