O=C(C[C@H](NCC1CC1)c1ccccc1)N1CCCOc2ccccc21 CHEMBL4456545 EC50 1.0 nM
C[C@H](C(=O)NC1COc2ccc(F)cc2C1O)c1ccccc1 CHEMBL4446583 EC50 1.205 nM
C[C@H](C(=O)N[C@@H]1Cc2ccccc2[C@H]1S(C)(=O)=O)c1ccc(F)cc1 CHEMBL5285249 EC50 6.0 nM
C[C@H](C(=O)NC1COc2ccccc2C1S(C)(=O)=O)c1ccc(F)cc1 CHEMBL4556629 EC50 6.9 nM
C[C@H](C(=O)N[C@H]1COc2ccccc2[C@@H]1S(C)(=O)=O)c1ccc(F)cc1 CHEMBL5266235 EC50 7.0 nM
C[C@H](C(=O)N[C@@H]1CCc2ccccc2[C@H]1S(C)(=O)=O)c1ccc(F)cc1 CHEMBL5280256 EC50 28.0 nM
O=C(NCc1ccccc1F)C1c2ccccc2CC(=O)N1CC1CC1 CHEMBL4443735 EC50 29.2 nM
C[C@H](C(=O)N[C@H]1Cc2ccccc2[C@@H]1S(C)(=O)=O)c1ccc(F)cc1 CHEMBL5288955 EC50 38.0 nM
C[C@H](C(=O)NC1Cc2ccccc2C1)c1ccc(F)cc1 CHEMBL5286456 EC50 55.0 nM
CCc1nc2c(o1)CC(c1ccc(C)cc1C)CC2=O CHEMBL4174742 IC50 63.0 nM
c1ccc(C(NCCNC(c2ccccc2)c2ccccc2)c2ccccc2)cc1 CHEMBL1387826 EC50 64.0 nM
Cc1cc(N2C(=O)c3cccc(Cl)c3C2=O)c(F)cc1NC(=O)c1occc1C CHEMBL4798021 EC50 98.0 nM
Cc1ccc2c(c1)C(=O)N(c1cc(C)c(NC(=O)c3occc3C)cc1F)C2=O CHEMBL4777502 EC50 106.0 nM
CNCC[C@H](NCC(=O)N1CCCc2ccccc21)c1ccccc1 CHEMBL4535940 pEC50 109.65 nM
CNC[C@@H](OCC(=O)N1CCCc2ccccc21)c1ccccc1 CHEMBL5272418 EC50 110.0 nM
C[C@H](C(=O)NC1Cc2ccccc2C1)c1ccccc1 CHEMBL5291195 EC50 113.0 nM
Cc1cc(N2C(=O)c3cccc(F)c3C2=O)c(F)cc1NC(=O)c1occc1C CHEMBL4764083 EC50 114.0 nM
O=C(Nc1ccc(Oc2ccc(Cl)cn2)c(Cl)c1)c1ccccn1 CHEMBL4162576 EC50 148.0 nM
O=C(Cc1ccc(Cl)cc1)NC1Cc2ccccc2C1 CHEMBL5281755 EC50 156.0 nM
Cc1cc(NC(=O)c2occc2C)c(F)cc1N1C(=O)c2ccccc2C1=O CHEMBL4745982 EC50 180.0 nM
Cc1ccoc1C(=O)Nc1cc(F)c(N2C(=O)c3cccc(Cl)c3C2=O)c(F)c1F CHEMBL4787053 EC50 201.0 nM
O=C(CNC(c1ccccc1)c1ccccc1)N1CCCc2ccccc21 CHEMBL4575681 pEC50 218.78 nM
Cc1ccoc1C(=O)Nc1c(F)cc(N2C(=O)c3ccccc3C2=O)c(F)c1F CHEMBL4799902 EC50 302.0 nM
Cc1cc(N2C(=O)C3=C(CCCC3)C2=O)c(F)cc1NC(=O)c1occc1C CHEMBL4792152 EC50 372.0 nM
Cc1cc(N2C(=O)C3=C(CCCC3)C2=O)c(F)cc1NC(=O)c1ccco1 CHEMBL4760570 EC50 377.0 nM
Cc1cc(N2C(=O)C3=C(CCCC3)C2=O)c(F)cc1NC(=O)c1ccc(Cl)o1 CHEMBL4797971 EC50 400.0 nM
Cc1ccoc1C(=O)Nc1cc(F)c(N2C(=O)c3cccc(F)c3C2=O)c(F)c1F CHEMBL4746530 EC50 487.0 nM
COc1cc(F)c(-c2c(C)nn3c(C(F)(F)F)cc(C)nc23)c(F)c1 CHEMBL4168668 EC50 600.0 nM
COc1ccc(C(=O)Nc2cc(OC(F)(F)F)ccc2-n2cncn2)cc1OC CHEMBL4176971 pIC50 630.96 nM
COc1ccc(-c2c(C)nn3c(C(F)(F)F)cc(C)nc23)c(F)c1F CHEMBL4160748 EC50 649.0 nM
CCc1nn2c(C(F)(F)F)cc(C)nc2c1-c1cc(F)c(OC)cc1F CHEMBL4446107 EC50 740.0 nM
COc1cc(F)c(-c2noc(-c3cc(Cl)ccc3-n3cncn3)n2)c(F)c1OC CHEMBL5171986 pIC50 794.33 nM
COc1cc(-c2noc(-c3cc(Cl)ccc3-n3cncn3)n2)cc(F)c1OC CHEMBL5190992 pIC50 794.33 nM
COc1cc(OCC(=O)Nc2cc(OC(F)(F)F)ccc2-n2cncn2)ccc1OC1COC1 CHEMBL5202961 pIC50 812.83 nM
N[C@](CC1c2ccccc2Oc2ccccc21)(C(=O)O)[C@H]1C[C@@H]1C(=O)O CHEMBL432038 Ki 990.0 nM