N#Cc1ccc2c(c1)CN(S(=O)(=O)c1cccs1)[C@H](Cc1ccccc1)CN2Cc1c[nH]cn1 CHEMBL351706 IC50 1.3 nM
N#Cc1ccc(Cn2cncc2CN2CCN(c3cccc(Cl)c3)C(=O)C2)cc1 CHEMBL279433 Ki 1.6 nM
O=C(Cc1ccncc1)N1CCN([C@H]2c3ccc(Cl)cc3CCc3cccnc32)CC1 CHEMBL66699 IC50 1.9 nM
Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4cc5cc(NC(=O)c6ccc(N(CCCl)CCCl)cc6)ccc5o4)cn3C)cn2C)cc1C(=O)NCCC(=N)N CHEMBL554247 IC50 15.0 nM
Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4nc5cc(NC(=O)c6ccc(N(CCCl)CCCl)cc6)ccc5[nH]4)cn3C)cn2C)cc1C(=O)NCCC(=N)N CHEMBL552690 IC50 15.0 nM
Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4cc5cc(NC(=O)c6ccc(N(CCCl)CCCl)cc6)ccc5[nH]4)cn3C)cn2C)cc1C(=O)NCCC(=N)N CHEMBL554353 IC50 15.0 nM
Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4cc5cc(N(CCCl)CCCl)ccc5o4)cn3C)cn2C)cc1C(=O)NCCC(=N)N CHEMBL540313 IC50 15.0 nM
Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4cc5cc(NC(=O)c6ccc(N(CCCl)CCCl)cc6)ccc5n4C)cn3C)cn2C)cc1C(=O)NCCC(=N)N CHEMBL554189 IC50 15.0 nM
Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4cc5cc(N(CCCl)CCCl)ccc5n4C)cn3C)cn2C)cc1C(=O)NCCC(=N)N CHEMBL552863 IC50 20.0 nM
Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC(=O)c4cc5cc(N(CCCl)CCCl)ccc5[nH]4)cn3C)cn2C)cc1C(=O)NCCC(=N)N CHEMBL536328 IC50 20.0 nM
COc1nc(-c2cccc3c2OCCO3)ccc1Nc1ccc(CN(C)C)cc1 CHEMBL4456044 Kd 51.0 nM
NC(=O)N1CCC(CC(=O)N2CCC([C@H]3c4ncc(Br)cc4CCc4cc(Cl)cc(Br)c43)CC2)CC1 CHEMBL298734 IC50 70.0 nM
O=C(CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)NCC1(c2ccccc2)CCC1 CHEMBL326352 IC50 88.0 nM
COC(=O)[C@H](CCSC)CC(=O)c1cc(CNC[C@@H](N)CS)ccc1-c1ccccc1 CHEMBL5171806 IC50 100.0 nM
O=C(CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)NCC1(c2ccccc2)CC1 CHEMBL407445 IC50 180.0 nM
CC(C)(CNC(=O)CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)c1ccccc1 CHEMBL431440 IC50 180.0 nM
N#CC(CNC(=O)CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)c1ccccc1 CHEMBL115943 IC50 190.0 nM
Cn1cc(NC(=O)c2cc(NC(=O)c3cc(NC=O)cn3C)cn2C)cc1C(=O)NCCC(=N)N CHEMBL11252 IC50 200.0 nM
C[C@H](CNC(=O)CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)c1ccccc1 CHEMBL115669 IC50 300.0 nM
CC(CNC(=O)CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)c1ccccc1 CHEMBL324827 IC50 310.0 nM
O=C(CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)NCC1(c2ccccc2)CCCC1 CHEMBL326127 IC50 330.0 nM
CCC(CNC(=O)CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)c1ccccc1 CHEMBL112512 IC50 400.0 nM
C[C@@H](CNC(=O)CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1)c1ccccc1 CHEMBL114281 IC50 570.0 nM
C[C@H](Cc1ccccc1)NC(=O)CN(Cc1ccc(OCc2ccccc2)cc1)C(=O)[C@H](Cc1c[nH]cn1)NC(=O)OCc1ccccc1 CHEMBL325073 IC50 710.0 nM
COc1ccc2nc3c(c(C)nn3[C@H]3CN(Sc4ccccc4[N+](=O)[O-])C[C@@H](CO[Si](C)(C)C(C)(C)C)O3)c(Cl)c2c1 CHEMBL304462 IC50 1000.0 nM