CCn1c(=O)c2ccccc2n(Cc2nnc(-c3ccc(F)c(O)c3F)s2)c1=O CHEMBL5411903 Ki 0.6 nM
CCn1c(=O)c(C)cn(Cc2nnc(-c3ccc(F)c(O)c3F)s2)c1=O CHEMBL5307400 Ki 0.7 nM
CCn1c(=O)c2c(n(Cc3nnc(-c4ccc(F)c(O)c4F)s3)c1=O)CCC2 CHEMBL5417980 Ki 0.8 nM
CCn1c(=O)c(C)cn(Cc2cnc(-c3ccc(F)c(O)c3F)s2)c1=O CHEMBL5405782 Ki 1.0 nM
CCn1c(=O)ccn(Cc2nnc(-c3ccc(F)c(O)c3F)s2)c1=O CHEMBL5418605 Ki 2.0 nM
CCn1c(=O)ccn(Cc2cnc(-c3ccc(F)c(O)c3F)s2)c1=O CHEMBL5429503 Ki 2.6 nM
O=c1ccn(Cc2cnc(-c3ccc(F)c(O)c3F)s2)c(=O)n1CC1CC1 CHEMBL5423975 Ki 3.0 nM
CCn1c(=O)cc(C)n(Cc2nnc(-c3ccc(F)c(O)c3F)s2)c1=O CHEMBL5394877 Ki 3.6 nM
O=c1ccn(Cc2cnc(-c3ccc(F)c(O)c3F)s2)c(=O)n1CC(F)(F)F CHEMBL5405439 IC50 4.0 nM
Cn1c(=O)ccn(Cc2nnc(-c3ccc(F)c(O)c3F)s2)c1=O CHEMBL5414092 Ki 4.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3cc(F)cc(O)c3Cl)s2)c1=O CHEMBL5394361 IC50 9.0 nM
Cc1cc(O)c(Cl)c(-c2ncc(Cn3ccc(=O)n(C)c3=O)s2)c1 CHEMBL5418452 IC50 18.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3cc(O)c(F)cc3F)s2)c1=O CHEMBL5424281 IC50 19.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3cccc(O)c3F)s2)c1=O CHEMBL5423890 IC50 23.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3ccc(F)c(O)c3Cl)s2)c1=O CHEMBL5414113 IC50 30.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3cccc(O)c3Cl)s2)c1=O CHEMBL5422335 IC50 48.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3ccc(F)c(O)c3)s2)c1=O CHEMBL5408952 IC50 97.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3cc(O)cc(F)c3)s2)c1=O CHEMBL5415759 IC50 97.0 nM
O=C(Nc1cccc2ncn(Cc3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5395506 IC50 100.0 nM
O=C(Nc1cccc2ncn(CC3CC3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5397286 IC50 100.0 nM
COc1ccccc1Cn1cnc2cccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c1=O CHEMBL5397292 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccc(F)cc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5405454 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccc(OC(F)(F)F)cc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5433430 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccccc3F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5430396 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cccc(F)c3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5425794 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccc(C(F)(F)F)nc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5429126 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5409199 IC50 100.0 nM
O=C(Nc1ncsc1C(=O)NCCc1ccccc1C(F)(F)F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5407026 IC50 100.0 nM
O=C(Nc1ncsc1C(=O)NCc1ccccc1C(F)(F)F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5405504 IC50 100.0 nM
O=C(Nc1ncsc1C(=O)NCc1ccccc1OC(F)(F)F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5408341 IC50 100.0 nM
O=C(Nc1ncsc1C(=O)NC1(c2ccc(F)cc2)CC1)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5425997 IC50 100.0 nM
Cc1nsc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c1C(=O)NCc1ccccc1F CHEMBL5420097 IC50 100.0 nM
O=C(Nc1scnc1C(=O)NCc1ccccc1F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5426934 IC50 100.0 nM
COc1ccccc1CCn1cnc2cccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c1=O CHEMBL5395069 IC50 100.0 nM
O=C(Nc1cc(Cl)sc1C(=O)NCCc1ccccc1OC(F)(F)F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5410205 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cccc(C(F)(F)F)c3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5423086 IC50 100.0 nM
N#Cc1cccc(Cn2cnc3cccc(NC(=O)c4cc(Cl)c(O)c(Cl)c4)c3c2=O)c1 CHEMBL5419894 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cccc(OC(F)(F)F)c3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5415032 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccc(OC(F)(F)F)cc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5429968 IC50 100.0 nM
CS(=O)(=O)c1ccccc1Cn1cnc2cccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c1=O CHEMBL5420215 IC50 100.0 nM
CC(C)(C)CCn1cnc2cccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c1=O CHEMBL5421316 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccc(OCCO)cc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5437607 IC50 100.0 nM
CC(C)(C)CCn1cnc2cccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c1=O CHEMBL5436217 IC50 100.0 nM
CC(C)(C)n1ccc(Cn2cnc3cccc(NC(=O)c4cc(Cl)c(O)c(Cl)n4)c3c2=O)n1 CHEMBL5403172 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccc(N4CCS(=O)(=O)CC4)cc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5395375 IC50 100.0 nM
N#Cc1ccccc1Cn1cnc2cccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c1=O CHEMBL5431821 IC50 100.0 nM
O=C(Nc1cccnc1C(=O)NCc1ccccc1OC(F)(F)F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5407358 IC50 100.0 nM
O=C(Nc1cccc2nc(C(F)(F)F)n(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5417715 IC50 100.0 nM
CC(C)(C)CCNC(=O)c1ccccc1NC(=O)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5426273 IC50 100.0 nM
O=C(Nc1cccc2ncn(C3(c4ccccc4F)CC3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5396658 IC50 100.0 nM
O=C(Nc1cnccc1C(=O)NCc1ccccc1OC(F)(F)F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5434503 IC50 100.0 nM
CC(c1ccccc1OC(F)(F)F)n1cnc2cccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c1=O CHEMBL5411521 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccn(-c4ccccc4)n3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5429505 IC50 100.0 nM
O=C(Nc1ccc(OCCO)cc1C(=O)NCc1ccccc1OC(F)(F)F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5438729 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cccnc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5409499 IC50 100.0 nM
O=C(Nc1ccc(Cl)c2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5400119 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ccccc3OC(F)(F)F)cnc12 CHEMBL5401817 IC50 100.0 nM
O=C(Nc1ccnc2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5401989 IC50 100.0 nM
Cc1ccc2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c2c1NC(=O)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5407748 IC50 100.0 nM
O=C(Nc1ccnc2[nH]c(=O)n(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5425130 IC50 100.0 nM
O=C(Nc1csc2ncn(Cc3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5400824 IC50 100.0 nM
O=C(Nc1csc2ncn(Cc3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5402307 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cnn4ccccc34)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5433237 IC50 100.0 nM
O=C(Nc1csc2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5433549 IC50 100.0 nM
O=C(Nc1csc2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5440523 IC50 100.0 nM
Cn1ccc(-c2ccccc2Cn2cnc3cccc(NC(=O)c4cc(Cl)c(O)c(Cl)c4)c3c2=O)n1 CHEMBL5422285 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccccc3-c3ccccn3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5438723 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ccccc3-c3ccccn3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5395467 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3ccccc3OC(F)(F)F)c(C(F)(F)F)nc12 CHEMBL5419052 IC50 100.0 nM
Cn1c(=O)n(Cc2ccccc2OC(F)(F)F)c(=O)c2c(NC(=O)c3cc(Cl)c(O)c(Cl)n3)cccc21 CHEMBL5420561 IC50 100.0 nM
Cc1nsc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c1C(=O)NCc1ccccc1F CHEMBL5414301 IC50 100.0 nM
Cc1nsc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c1C(=O)N[C@@H](C)c1ccccc1F CHEMBL5399220 IC50 100.0 nM
O=C(Nc1cccc2nc(C(F)(F)F)n(C3CC3c3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5415821 IC50 100.0 nM
Cn1nc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ccccc3OC(F)(F)F)cnc21 CHEMBL5429030 IC50 100.0 nM
O=C(Nc1cccc2ncn([C@H]3CC[C@@H]3c3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5436398 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cccnc3Cl)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5427317 IC50 100.0 nM
O=C(Nc1cccc2ncn(C(CN3CCOCC3)c3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5396981 IC50 100.0 nM
O=C(Nc1sc(C(F)(F)F)nc1C(=O)NCc1ccccc1OC(F)(F)F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5402660 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cccnc3Cl)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5421244 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ncccc3F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5398292 IC50 100.0 nM
Cc1ccc2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c2c1NC(=O)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5403856 IC50 100.0 nM
O=C(Nc1ccc(F)c2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5405884 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cccnc3F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5397519 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3cccnc3F)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5421584 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ncccc3F)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5431104 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3cccnc3C(F)(F)F)c(C)nc12 CHEMBL5429787 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3cccnc3C(F)(F)F)c(C)nc12 CHEMBL5412141 IC50 100.0 nM
O=C(Nc1cccc2ncn(Cc3ncccc3Cl)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5423106 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ncccc3C(F)(F)F)c(C)nc12 CHEMBL5436106 IC50 100.0 nM
Cc1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c(=O)n1Cc1ncccc1C(F)(F)F CHEMBL5416441 IC50 100.0 nM
Cc1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c(=O)n1C(C)c1ccccc1OC(F)(F)F CHEMBL5424401 IC50 100.0 nM
Cc1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c(=O)n1Cc1ccccc1C(F)(F)F CHEMBL5430947 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3nn(C)c4ccccc34)c(C)nc12 CHEMBL5437897 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ccccc3C(F)(F)F)c(C)nc12 CHEMBL5425384 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3ncccc3C(F)(F)F)c(C(F)F)nc12 CHEMBL5418907 IC50 100.0 nM
Cc1nc2c(Cl)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c(=O)n1Cc1ncccc1C(F)(F)F CHEMBL5411931 IC50 100.0 nM
Cc1nc2c(Cl)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c(=O)n1Cc1ncccc1C(F)(F)F CHEMBL5409271 IC50 100.0 nM
Cc1nc2c(Cl)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c(=O)n1Cc1ccccc1C(F)(F)F CHEMBL5413196 IC50 100.0 nM
[2H]C([2H])([2H])c1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c(=O)n1Cc1ccccc1C(F)(F)F CHEMBL5418415 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3ncccc3Cl)c(C)nc12 CHEMBL5400961 IC50 100.0 nM
Cc1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c(=O)n1[C@@H](C)c1ccccc1OC(F)(F)F CHEMBL5426835 IC50 100.0 nM
Cc1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c(=O)n1[C@H](C)c1ccccc1OC(F)(F)F CHEMBL5402107 IC50 100.0 nM
O=C(Nc1cccc2ncn([C@@H]3CC[C@H]3c3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5416475 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ncccc3C(F)(F)F)c(C(F)F)nc12 CHEMBL5422016 IC50 100.0 nM
[2H]C([2H])([2H])c1nc2c(C)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c(=O)n1Cc1ccccc1C(F)(F)F CHEMBL5412096 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ccccc3C(F)(F)F)c(C(F)F)nc12 CHEMBL5412804 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3ncccc3F)c(C)nc12 CHEMBL5419216 IC50 100.0 nM
[2H]C([2H])([2H])c1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c(=O)n1Cc1ccccc1C(F)(F)F CHEMBL5421460 IC50 100.0 nM
Cn1nc(CNC(=O)c2ncsc2NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2ccccc21 CHEMBL5426094 IC50 100.0 nM
O=C(Nc1scnc1C(=O)NCc1cccc(F)c1)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5433659 IC50 100.0 nM
O=C(Nc1scnc1C(=O)NCc1ccccc1C(F)(F)F)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5429805 IC50 100.0 nM
Cc1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c(=O)n1Cc1nn(C)c2ccccc12 CHEMBL5409131 IC50 100.0 nM
O=C(Nc1scnc1C(=O)NCc1ncccc1C(F)(F)F)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5418089 IC50 100.0 nM
[2H]C([2H])(c1ccccc1C(F)(F)F)n1c(C)nc2c(C)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c1=O CHEMBL5403127 IC50 100.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n([C@@H]3CC[C@H]3c3ccccc3)c(C)nc12 CHEMBL5406249 IC50 100.0 nM
Cc1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c(=O)n1[C@H]1CC[C@@H]1c1ccccc1 CHEMBL5399143 IC50 100.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3ccc(Cl)c(O)c3)s2)c1=O CHEMBL5423215 IC50 117.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3cc(O)cc(C(F)(F)F)c3)s2)c1=O CHEMBL5396531 IC50 118.0 nM
Cn1c(=O)ccn(Cc2nnc(-c3cccc(O)c3)s2)c1=O CHEMBL5428422 IC50 176.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3cc(O)ccc3F)s2)c1=O CHEMBL5396549 IC50 397.0 nM
O=C(Nc1cccc2ncn(Cc3ccncc3F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5421633 IC50 500.0 nM
O=C(Nc1cccc2ncn(Cc3cocn3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5413478 IC50 500.0 nM
O=C(Nc1ncsc1C(=O)NCC1CCC(F)(F)CC1)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5398685 IC50 500.0 nM
CC(C)(C)n1ccc(Cn2cnc3cccc(NC(=O)c4cc(Cl)c(O)c(Cl)c4)c3c2=O)n1 CHEMBL5427557 IC50 500.0 nM
Cn1ccc(Cn2cnc3cccc(NC(=O)c4cc(Cl)c(O)c(Cl)c4)c3c2=O)n1 CHEMBL5397057 IC50 500.0 nM
CS(=O)(=O)c1cccc(Cn2cnc3cccc(NC(=O)c4cc(Cl)c(O)c(Cl)c4)c3c2=O)c1 CHEMBL5419316 IC50 500.0 nM
CS(=O)(=O)c1ccccc1Cn1cnc2cccc(NC(=O)c3cc(Cl)c(O)c(Cl)n3)c2c1=O CHEMBL5434612 IC50 500.0 nM
O=C(Nc1cccc2ncn(Cc3cccnc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5420979 IC50 500.0 nM
Cn1nc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ccccc3)cnc21 CHEMBL5423891 IC50 500.0 nM
O=C(Nc1cccc2ncn([C@@H]3C[C@H]3c3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5439133 IC50 500.0 nM
Cn1nc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3ccccc3OC(F)(F)F)cnc21 CHEMBL5425558 IC50 500.0 nM
O=C(NC1CCCC1C(=O)NCc1ccccc1OC(F)(F)F)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5438627 IC50 500.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3ccccc3OC(F)(F)F)c(CF)nc12 CHEMBL5406423 IC50 500.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ncccc3Cl)c(C)nc12 CHEMBL5437149 IC50 500.0 nM
O=C(Nc1scnc1C(=O)NCc1cccc(C(F)(F)F)n1)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5440483 IC50 500.0 nM
Cc1nc2c(F)ccc(NC(=O)c3cc(Cl)c(O)c(Cl)c3)c2c(=O)n1Cc1cccc(C(F)(F)F)n1 CHEMBL5421209 IC50 500.0 nM
O=C(Nc1scnc1C(=O)NCc1cccc(C(F)(F)F)n1)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5402646 IC50 500.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3cccc(C(F)(F)F)n3)c(C)nc12 CHEMBL5405234 IC50 500.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3cccc(C(F)(F)F)n3)c(C)nc12 CHEMBL5416634 IC50 500.0 nM
Cn1c(=O)ccn(Cc2cc(-c3cccc(O)c3)on2)c1=O CHEMBL5413959 IC50 510.0 nM
Cn1c(=O)ccn(Cc2cc(-c3cccc(O)c3)no2)c1=O CHEMBL5436438 IC50 562.0 nM
Cn1c(=O)ccn(Cc2cnc(-c3cncc(O)c3)s2)c1=O CHEMBL5434049 IC50 644.0 nM
Cn1c(=O)ccn(Cc2ncc(-c3cccc(O)c3)s2)c1=O CHEMBL5423248 IC50 652.0 nM
O=C(Nc1cccc2ncn(Cc3cc[nH]c(=O)c3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5413418 IC50 1000.0 nM
O=C(Nc1cccc2ncn(Cc3nncs3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5418442 IC50 1000.0 nM
O=C(Nc1cccc2ncn(Cc3ccncc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5432384 IC50 1000.0 nM
O=C(Nc1cccc2ncn(C3(c4ccccc4)CC3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5415521 IC50 1000.0 nM
O=C(Nc1ncsc1C(=O)NCc1ccccc1F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5423244 IC50 1000.0 nM
O=C(Nc1ncsc1C(=O)NCc1ccc(F)cc1F)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5406196 IC50 1000.0 nM
CN1CCN(c2ccc(Cn3cnc4cccc(NC(=O)c5cc(Cl)c(O)c(Cl)c5)c4c3=O)cc2)CC1 CHEMBL5423062 IC50 1000.0 nM
O=C(Nc1cccc2ncnc(NCc3ccccc3OC(F)F)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5438147 IC50 1000.0 nM
CS(=O)(=O)c1ccc(Cn2cnc3cccc(NC(=O)c4cc(Cl)c(O)c(Cl)c4)c3c2=O)cc1 CHEMBL5410536 IC50 1000.0 nM
O=C(Nc1cccc2ncn(Cc3cccc(OC(F)(F)F)c3)c(=O)c12)c1ccc(Cl)c(O)c1Cl CHEMBL5406067 IC50 1000.0 nM
O=C(Nc1cccc2ncn(Cc3ccccc3N3CCS(=O)(=O)CC3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5401673 IC50 1000.0 nM
Cn1nc(NC(=O)c2cc(Cl)c(O)c(Cl)c2)c2c(=O)n(Cc3ccccc3)cnc21 CHEMBL5426496 IC50 1000.0 nM
O=C(Nc1cccc2nc(C(F)(F)F)n(C3CC3c3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5420111 IC50 1000.0 nM
O=C(Nc1cccc2ncn([C@@H]3C[C@H]3c3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5399593 IC50 1000.0 nM
O=C(Nc1cccc2ncn([C@H]3C[C@@H]3c3ccccc3)c(=O)c12)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5437370 IC50 1000.0 nM
O=C(NCc1ccccc1OC(F)(F)F)C1CCCCN1C(=O)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5424978 IC50 1000.0 nM
O=C(Nc1nccc2ncn(Cc3ccccc3OC(F)(F)F)c(=O)c12)c1cc(Cl)c(O)c(Cl)c1 CHEMBL5402917 IC50 1000.0 nM
O=C(N[C@@H]1CCCC[C@H]1C(=O)NCc1ccccc1OC(F)(F)F)c1cc(Cl)c(O)c(Cl)n1 CHEMBL5428675 IC50 1000.0 nM
Cc1ccc(NC(=O)c2cc(Cl)c(O)c(Cl)n2)c2c(=O)n(Cc3ncccc3F)c(C)nc12 CHEMBL5416567 IC50 1000.0 nM