Cc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)ccc2n1 CHEMBL4070633 IC50 2.8 nM
CCc1cnn2c(NCc3ccc[n+]([O-])c3)cc(N3CCCC[C@H]3CCO)nc12 CHEMBL2103840 IC50 7.0 nM
Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1ccc2ncccc2c1 CHEMBL4063330 IC50 12.0 nM
CN1CCC[C@H]1COc1ccc(Nc2cc(-n3cnc4ncccc43)ncn2)nc1 CHEMBL3975567 IC50 14.0 nM
c1cnc2ncn(-c3cc(Nc4ccc(OCCN5CCCCC5)cn4)ncn3)c2c1 CHEMBL3937369 IC50 15.0 nM
Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1ccc2nc(OCCN3CCCC3)ccc2c1 CHEMBL4087666 pIC50 18.62 nM
Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1ccc2nc(OCCN)ccc2c1 CHEMBL4102297 IC50 26.0 nM
CN(C)CCOc1ccc(Nc2cc(-n3cnc4ncccc43)ncn2)nc1 CHEMBL3911352 IC50 28.0 nM
Cc1ccc2ncn(-c3cc(Nc4ccc(OCCN(C)C)cn4)ncn3)c2c1 CHEMBL3964729 IC50 39.0 nM
CN1CCC[C@@H]1COc1ccc(Nc2cc(-n3cnc4ccccc43)ncn2)nc1 CHEMBL3972065 IC50 45.0 nM
Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1ccc2ccncc2c1 CHEMBL4069552 IC50 51.0 nM
CN1CCC[C@H]1COc1ccc(Nc2cc(-n3cnc4ccccc43)ncn2)nc1 CHEMBL3953713 IC50 55.0 nM
c1ccc2c(c1)ncn2-c1cc(Nc2ccc(OCCN3CCCCC3)cn2)ncn1 CHEMBL3928361 IC50 57.0 nM
CN(C)CCOc1ccc(Nc2cc(-n3cnc4ccccc43)ncn2)nc1 CHEMBL3919811 IC50 80.0 nM
CCC(=O)NCCOc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCO5)ccc3C)ccc2n1 CHEMBL4070302 pIC50 114.82 nM
CN(C)CCCOc1ccc(Nc2cc(-n3cnc4ccccc43)ncn2)nc1 CHEMBL3983798 IC50 165.0 nM
CN(C)CCCc1ccc(Nc2cc(-n3cnc4ccccc43)ncn2)nc1 CHEMBL3901185 IC50 198.0 nM
Cc1ccc(NC(=O)c2ccc3c(c2)OCCO3)cc1NC(=O)c1ccc2c(c1)CCCN2 CHEMBL4096048 IC50 220.0 nM
c1ccc2c(c1)ncn2-c1cc(Nc2ccc(OCCN3CCOCC3)cn2)ncn1 CHEMBL3900925 IC50 295.0 nM
Cc1ccc2cc(C(=O)Nc3cc(NC(=O)c4ccc5c(c4)OCCC5)ccc3C)ccc2n1 CHEMBL4077078 pIC50 446.68 nM
CN1CCN(c2ccc(Nc3cc(-n4cnc5ccccc54)ncn3)nc2)CC1 CHEMBL3919459 IC50 450.0 nM
CN(C)C1CCN(c2ccc(Nc3cc(-n4cnc5ccccc54)ncn3)nc2)CC1 CHEMBL3946252 IC50 610.0 nM
CC(C)(C)c1cnc(CSc2cnc(NC(=O)N3CCNCC3)s2)o1 CHEMBL3967087 IC50 750.0 nM
CN(C)CCOc1ccc(Nc2cc(-n3cnc4cccnc43)ncn2)nc1 CHEMBL3936187 IC50 760.0 nM
c1ccc(Nc2cc(-n3cnc4ccccc43)ncn2)nc1 CHEMBL3944589 IC50 842.0 nM
CN1CCC(Oc2ccc(Nc3cc(-n4cnc5ccccc54)ncn3)nc2)CC1 CHEMBL3955977 IC50 884.0 nM