FC1(F)CC(Nc2nc(NC3CC(F)(F)C3)nc(-c3cccc(C(F)(F)F)n3)n2)C1 CHEMBL4280772 IC50 3.0 nM
C[C@@H](Nc1nc(N[C@H](C)C2CC2)nc(-c2cccc(Cl)n2)n1)C1CC1 CHEMBL4278420 IC50 4.0 nM
O[C@@]1(C(F)(F)F)CCN(c2nc(Nc3ccnc(C(F)(F)F)c3)nc(-c3cccc(C(F)(F)F)n3)n2)C1 CHEMBL5415614 IC50 4.78 nM
C[C@H](Nc1nc(N2C(=O)OC[C@@H]2[C@H](C)F)c2cc[nH]c2n1)c1cn(-c2ccc(Cl)cc2)cn1 CHEMBL4463644 IC50 6.0 nM
Cc1cc([C@@H](C)Nc2nc(N3C(=O)OC[C@@H]3C(C)C)c3cc[nH]c3n2)ncc1-c1ccnc(C(F)(F)F)c1 CHEMBL4439421 IC50 6.0 nM
FC1(F)CCC(Nc2nc(NC3CCC(F)(F)C3)nc(-c3cccc(Cl)n3)n2)C1 CHEMBL4280132 IC50 6.0 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCCCCC2 CHEMBL4753099 IC50 6.1 nM
C[C@@H](Nc1nc(N[C@H](C)C(F)(F)F)nc(-c2cccc(Cl)n2)n1)C(F)(F)F CHEMBL4279047 IC50 7.0 nM
C[C@H](Nc1nc(N[C@@H](C)C(F)(F)F)nc(-c2cccc(Cl)n2)n1)C(F)(F)F CHEMBL4278845 IC50 7.0 nM
OCC(O)CNc1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)c2)n1 CHEMBL5405494 IC50 7.0 nM
CC(Nc1nc(NC(C)C(F)(F)F)nc(-c2cccc(Cl)n2)n1)C(F)(F)F CHEMBL4283785 IC50 8.0 nM
OCC(CO)Nc1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)c2)n1 CHEMBL5428697 IC50 8.0 nM
CC(C)(O)CNc1nc(Nc2ccnc(C(F)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL3989908 IC50 9.0 nM
FC1(F)CCC(Nc2nc(NC3CCC(F)(F)C3)nc(-c3cccc(C(F)(F)F)n3)n2)C1 CHEMBL4277352 IC50 9.0 nM
FC1(F)CCC(Nc2nc(NC3CCC(F)(F)CC3)nc(-c3cccc(C(F)(F)F)n3)n2)CC1 CHEMBL4288840 IC50 9.0 nM
OC[C@@H](O)CNc1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)c2)n1 CHEMBL5430339 IC50 9.0 nM
CC1(C)CNc2nc(nc(-c3cccc(C(F)(F)F)n3)n2)Nc2cc(cc(C(F)(F)F)c2)CCCCO1 CHEMBL4787510 IC50 9.6 nM
OC1CCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)c3)n2)C1 CHEMBL5441137 IC50 10.0 nM
FC(F)(F)c1cccc(-c2nc3nc(n2)Nc2cc(Cl)cc(c2)CCCCOCCN3)n1 CHEMBL4800354 IC50 12.2 nM
FC(F)(F)c1cccc(-c2nc(NCC3CC3)nc(NCC3CC3)n2)n1 CHEMBL4292293 IC50 13.0 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCC/C=C/C2 CHEMBL4796025 IC50 13.8 nM
C[C@@H](Nc1nc(N[C@H](C)C2CC2)nc(-c2cccc(C(F)(F)F)n2)n1)C1CC1 CHEMBL4278828 IC50 14.0 nM
CCC(Nc1nc(NC(CC)C2CC2)nc(-c2cccc(Cl)n2)n1)C1CC1 CHEMBL4282989 IC50 14.0 nM
C=CCOC(C)(C)CNc1nc(Nc2cccc(C(F)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4754521 IC50 15.5 nM
FC(F)(F)c1cc2cc(c1)OC/C=C\CCCNc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)N2 CHEMBL4786020 IC50 17.4 nM
CC1CNc2nc(nc(-c3cccc(C(F)(F)F)n3)n2)Nc2cc(cc(C(F)(F)F)c2)CCCCO1 CHEMBL4762400 IC50 17.7 nM
FC(F)(F)c1cc2cc(c1)OC/C=C\CCNc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)N2 CHEMBL4753744 IC50 18.4 nM
Fc1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCOCCCC2 CHEMBL4783076 IC50 18.6 nM
CC(C)Nc1nc(Nc2ccnc(C(F)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4448857 IC50 19.0 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCCCCCC2 CHEMBL4782070 IC50 19.9 nM
FC1(F)CCC(Nc2nc(NC3CCC(F)(F)CC3)nc(-c3cccc(Cl)n3)n2)CC1 CHEMBL4289692 IC50 22.0 nM
Cc1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCOCCCC2 CHEMBL4746278 IC50 22.2 nM
O=C(Nc1cccc(C(F)(F)F)c1)Nc1cc(S(=O)(=O)NC2CC2)ccc1-c1ccsc1 CHEMBL3392845 IC50 23.0 nM
OC1CCCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)c3)n2)C1 CHEMBL5397750 IC50 23.0 nM
O[C@@H]1CCCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)c3)n2)C1 CHEMBL5433752 IC50 24.0 nM
O[C@H]1CCCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)c3)n2)C1 CHEMBL5410201 IC50 25.0 nM
CC(C)(O)CNc1nc(Nc2cccc(C(F)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4756154 IC50 26.0 nM
CC1(C)CNc2nc(nc(-c3cccc(C(F)(F)F)n3)n2)Nc2cc(cc(C(F)(F)F)c2)OCCCO1 CHEMBL4756939 IC50 27.4 nM
Fc1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCOC/C=C\C2 CHEMBL4750012 IC50 29.5 nM
OC[C@H](O)CNc1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)c2)n1 CHEMBL5432152 IC50 31.0 nM
CC(C)(C)ONc1nc(Nc2ccnc(C(F)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4456102 IC50 31.69 nM
OC1CCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)c3)n2)CC1 CHEMBL5406499 IC50 32.0 nM
FC(F)(F)c1cccc(-c2nc3nc(n2)Nc2cc(Cl)cc(c2)C/C=C\COCCN3)n1 CHEMBL4790341 IC50 36.0 nM
CNc1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)c2)n1 CHEMBL5401153 IC50 37.0 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCCCCCCC2 CHEMBL4739900 IC50 37.2 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCCCC/C=C/C2 CHEMBL4781074 IC50 37.6 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCCC/C=C/C2 CHEMBL4751821 IC50 37.6 nM
Cc1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCOC/C=C\C2 CHEMBL4779519 IC50 37.9 nM
O[C@@H]1CCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)n3)n2)C1 CHEMBL5418738 IC50 38.0 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCOC/C=C\C2 CHEMBL4793173 IC50 39.9 nM
Cc1ccc(Cl)cc1NC(=O)Nc1cc(NC(=O)c2ccccc2)ccc1N1CCCC1 CHEMBL4536525 IC50 41.0 nM
FC(F)(F)c1cc2cc(c1)OCCCCCCNc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)N2 CHEMBL4793042 IC50 45.5 nM
CC(C)(C)Nc1nc(NC(C)(C)C)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4284907 IC50 46.0 nM
C=CCOC(C)(C)CNc1nc(Nc2ccccc2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4761041 IC50 46.0 nM
COc1ccc(F)c(-c2nc(N[C@H](C)C3CC3)nc(N[C@H](C)C3CC3)n2)c1 CHEMBL4290152 IC50 50.0 nM
C[C@@H](Nc1nc(NCC(C)(C)O)nc(-c2cccc(C(F)(F)F)n2)n1)C1CC1 CHEMBL4280581 IC50 50.0 nM
CC(O)CNc1nc(N[C@H](C)C2CC2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4282029 IC50 50.0 nM
C[C@@H](Nc1nc(NC2(c3ccccc3)CC2)nc(-c2cccc(C(F)(F)F)n2)n1)C1CC1 CHEMBL4292196 IC50 50.0 nM
CC(C)CNc1nc(NC2CCOCC2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4280463 IC50 50.0 nM
FC1(F)CCCC1Nc1nc(NC2CCCC2(F)F)nc(-c2cccc(Cl)n2)n1 CHEMBL4281900 IC50 50.0 nM
CC[C@H](Nc1nc(N[C@@H](CC)C(F)(F)F)nc(-c2cccc(Cl)n2)n1)C(F)(F)F CHEMBL4284624 IC50 50.0 nM
FC1(F)CCC(Nc2nc(NC3CCC(F)(F)C3)nc(-c3ccnc(C(F)(F)F)n3)n2)C1 CHEMBL4288431 IC50 50.0 nM
CC[C@H](Nc1nc(N[C@H](CC)C(F)(F)F)nc(-c2cccc(Cl)n2)n1)C(F)(F)F CHEMBL4286718 IC50 50.0 nM
FC1(F)CCC(Nc2nc(Nc3ccnc(-c4ccccc4)c3)nc(-c3cccc(C(F)(F)F)n3)n2)CC1 CHEMBL4284814 IC50 50.0 nM
C[C@@H](Nc1nc(NCCOc2ccccc2)nc(-c2cccc(C(F)(F)F)n2)n1)C1CC1 CHEMBL4277498 IC50 50.0 nM
C[C@@H](Nc1nc(N[C@H](C)C2CC2)nc(-c2nccc(C(F)(F)F)n2)n1)C1CC1 CHEMBL4285495 IC50 50.0 nM
FC1(F)CC(Nc2nc(NC3CC(F)(F)C3)nc(-c3cccc(OC(F)(F)F)n3)n2)C1 CHEMBL4289797 IC50 50.0 nM
FC1(F)CCC(Nc2nc(NC3CCC(F)(F)CC3)nc(-c3nccc(C(F)(F)F)n3)n2)CC1 CHEMBL4288632 IC50 50.0 nM
C[C@@H](Nc1nc(N[C@H](C)C(F)(F)F)nc(-c2ccnc(C(F)(F)F)n2)n1)C(F)(F)F CHEMBL4282694 IC50 50.0 nM
CC[C@H](Nc1nc(N[C@@H](CC)C(F)(F)F)nc(-n2ccc(C(F)(F)F)n2)n1)C(F)(F)F CHEMBL4289800 IC50 50.0 nM
FC(F)c1ccnc(-c2nc(NC3CC(F)(F)C3)nc(NC3CC(F)(F)C3)n2)n1 CHEMBL4281625 IC50 50.0 nM
CC(COC(C)C)Nc1nc(N[C@H](C)C2CC2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4286667 IC50 50.0 nM
CC(C)(O)CNc1nc(Nc2cc(F)cc(C#N)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4281594 IC50 50.0 nM
CC(CC#N)Nc1nc(Nc2ccnc(C(C)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4290554 IC50 50.0 nM
CC(C)(C#N)CNc1nc(Nc2ccnc(C(C)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4278435 IC50 50.0 nM
CC(C)(C)Nc1nc(Nc2ccnc(C(C)(F)F)c2)nc(-c2nccc(C(F)(F)F)n2)n1 CHEMBL4282925 IC50 50.0 nM
CC(C)Nc1nc(Nc2ccnc(C(C)(F)F)c2)nc(-c2nccc(C(F)(F)F)n2)n1 CHEMBL4284203 IC50 50.0 nM
CC(C)(O)CNc1nc(Nc2cc(F)cc(F)c2)nc(-c2nccc(C(F)(F)F)n2)n1 CHEMBL4277108 IC50 50.0 nM
FC(F)(F)c1cc2cc(c1)OCCCCCNc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)N2 CHEMBL4786533 IC50 51.0 nM
FC(F)(F)c1cccc(Nc2nc(Nc3ccccc3)nc(Nc3cccc(C(F)(F)F)c3)n2)c1 CHEMBL5394948 IC50 53.0 nM
CC(C)Nc1cc(Nc2cc(C(F)(F)F)ccn2)nc(-c2ccccc2)c1 CHEMBL4514677 IC50 54.6 nM
OC1CCCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)n3)n2)C1 CHEMBL5406543 IC50 56.0 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCCCCC2 CHEMBL4794091 IC50 60.9 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCCOCCCC2 CHEMBL4784873 IC50 64.4 nM
FC(F)(F)c1cccc(Nc2nc(Nc3cccc(C(F)(F)F)c3)nc(N3CCCCC3)n2)c1 CHEMBL5422550 IC50 66.0 nM
O[C@H]1CCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)n3)n2)C1 CHEMBL5407241 IC50 71.0 nM
OCC(CO)Nc1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)n2)n1 CHEMBL5397296 IC50 81.0 nM
CC(C)(O)CNc1nc(Nc2ccccc2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4790929 IC50 98.2 nM
FC1(F)CCC(Nc2nc(NC3CCN(c4ccccn4)C3)nc(-c3cccc(C(F)(F)F)n3)n2)C1 CHEMBL4289977 IC50 100.0 nM
FC1(F)CCC(Nc2nc(NC3CCN(c4ncccn4)C3)nc(-c3cccc(C(F)(F)F)n3)n2)C1 CHEMBL4282071 IC50 100.0 nM
CC(C)(O)CNc1nc(Nc2cccc(Cl)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4294615 IC50 100.0 nM
FC1(F)CCC(Nc2nc(NC3CCC(F)(F)CC3)nc(-c3ccnc(C(F)(F)F)n3)n2)CC1 CHEMBL4294396 IC50 100.0 nM
Fc1ccc([C@H]2C[C@@H](Nc3nc(N[C@H]4C[C@@H](c5ccc(F)cc5)C4)nc(-c4cccc(C(F)(F)F)n4)n3)C2)cc1 CHEMBL4291957 IC50 100.0 nM
C[C@@H](Nc1nc(N[C@H](C)C2CC2)nc(-n2cc(I)cn2)n1)C1CC1 CHEMBL4293859 IC50 100.0 nM
CC(F)(F)c1nc(-c2nc(NC3CCC(F)(F)CC3)nc(NC3CCC(F)(F)CC3)n2)cs1 CHEMBL4294387 IC50 100.0 nM
CC(C)(O)CNc1nc(NC2CCC(F)(F)CC2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4281385 IC50 100.0 nM
CC(C)(O)CNc1nc(Nc2ccnc(C#N)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4280325 IC50 100.0 nM
FC1(F)CCC(Nc2nc(NC3CCC(F)(F)CC3)nc(-n3cc(Cl)cn3)n2)CC1 CHEMBL4285024 IC50 100.0 nM
FC(F)c1ccnc(-c2nc(NC3CCC(F)(F)CC3)nc(NC3CCC(F)(F)CC3)n2)n1 CHEMBL4294544 IC50 100.0 nM
CC[C@H](Nc1nc(N[C@@H](CC)C(F)(F)F)nc(-c2ccnc(C(F)(F)F)n2)n1)C(F)(F)F CHEMBL4283760 IC50 100.0 nM
C[C@@H](Nc1nc(NC2C3CC4CC(C3)CC2C4)nc(-c2cccc(C(F)(F)F)n2)n1)C1CC1 CHEMBL4278414 IC50 100.0 nM
FC1(F)CCC(Nc2nc(NC3CCOCC3)nc(-c3cccc(C(F)(F)F)n3)n2)CC1 CHEMBL4292464 IC50 100.0 nM
C[C@@H](Nc1nc(NCC(C)(C)C#N)nc(-c2cccc(C(F)(F)F)n2)n1)C1CC1 CHEMBL4278807 IC50 100.0 nM
O=C(c1ccccc1)N1CCC(Nc2nc(NC3CCC(F)(F)C3)nc(-c3cccc(C(F)(F)F)n3)n2)C1 CHEMBL4283985 IC50 100.0 nM
FC1(F)CC2(CC(Nc3nc(NC4CC5(C4)CC(F)(F)C5)nc(-c4cccc(Cl)n4)n3)C2)C1 CHEMBL4285110 IC50 100.0 nM
CS(=O)(=O)N1CCC(Nc2nc(NC3CCC(F)(F)CC3)nc(-c3cccc(C(F)(F)F)n3)n2)CC1 CHEMBL4284068 IC50 100.0 nM
CC(CC#N)Nc1nc(NC(C)CC#N)nc(-c2cccc(Cl)n2)n1 CHEMBL4288016 IC50 100.0 nM
CC(C)(C)OC(=O)N1CCC(Nc2nc(NC3CCC(F)(F)CC3)nc(-c3cccc(C(F)(F)F)n3)n2)CC1 CHEMBL4277506 IC50 100.0 nM
FC1(F)CCC(Nc2nc(NC3CCN(Cc4ccccc4)C3)nc(-c3cccc(C(F)(F)F)n3)n2)C1 CHEMBL4294899 IC50 100.0 nM
C[C@H](Nc1cc(N[C@@H](C)C2CC2)nc(-c2cccc(C(F)(F)F)n2)n1)C1CC1 CHEMBL4286947 IC50 100.0 nM
CC(C)(C)Nc1nc(Nc2ccccc2)nc(-c2ccccc2)n1 CHEMBL5438535 IC50 100.0 nM
OC1CCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)n3)n2)C1 CHEMBL5429258 IC50 104.0 nM
O=C1OCCCCCNc2nc(nc(-c3cccc(C(F)(F)F)n3)n2)Nc2cc1cc(C(F)(F)F)c2 CHEMBL4782130 IC50 104.6 nM
CC(C)(O)CNc1nc(Nc2ccnc(C(F)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL3989931 IC50 123.6 nM
O=C(O)C1CCCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)c3)n2)C1 CHEMBL5405111 IC50 159.0 nM
OCC(O)CNc1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)n2)n1 CHEMBL5411897 IC50 160.0 nM
CC1(C)CCNc2nc(nc(-c3cccc(C(F)(F)F)n3)n2)Nc2cc(cc(C(F)(F)F)c2)CCCCO1 CHEMBL4748664 IC50 182.3 nM
CC(C)(O)CNc1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)c2)n1 CHEMBL5416375 IC50 193.0 nM
FC(F)(F)c1cc(Nc2nc(Nc3cccc(C(F)(F)F)n3)nc(N3CCCCC3)n2)ccn1 CHEMBL5425240 IC50 231.0 nM
O=S(=O)(NC1CC1)c1ccc(-c2ccsc2)c(Nc2nc3cc(Br)ccc3[nH]2)c1 CHEMBL4634103 IC50 260.0 nM
CC1CNc2nc(nc(-c3cccc(C(F)(F)F)n3)n2)Nc2cc(cc(C(F)(F)F)c2)C/C=C\CO1 CHEMBL4748497 IC50 266.7 nM
CC(C)(O)CNc1nc(Nc2ccnc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)n2)n1 CHEMBL5437453 IC50 287.0 nM
[2H]C([2H])([2H])C([2H])(C([2H])([2H])[2H])C([2H])([2H])Nc1nc(Nc2ccnc(C(F)(F)F)c2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4454958 IC50 360.0 nM
OC1CCCN(c2nc(Nc3ccnc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)n3)n2)C1 CHEMBL5425277 IC50 371.0 nM
CC1(C)CNc2nc(nc(-c3cccc(C(F)(F)F)n3)n2)Nc2cc(cc(C(F)(F)F)c2)C/C=C\CO1 CHEMBL4762182 IC50 396.0 nM
FC(F)(F)c1cccc(Nc2nc(Nc3cccc(C(F)(F)F)c3)nc(N3CCNCC3)n2)c1 CHEMBL5411497 IC50 423.0 nM
CN(C)c1nc(Nc2cccc(C(F)(F)F)c2)nc(Nc2cccc(C(F)(F)F)c2)n1 CHEMBL5412348 IC50 493.0 nM
O=S(=O)(NC1CC1)c1ccc(-c2ccsc2)c(Nc2nc3ccc(Br)c(Br)c3[nH]2)c1 CHEMBL4643441 IC50 650.0 nM
CC(C)(O)CNc1nc(Nc2ccncc2)nc(-c2cccc(C(F)(F)F)n2)n1 CHEMBL4788410 IC50 663.4 nM
FC(F)(F)c1cc2cc(c1)Nc1nc(nc(-c3cccc(C(F)(F)F)n3)n1)NCC/C=C/C2 CHEMBL4753020 IC50 683.5 nM
O=C1NCCCCNc2nc(nc(-c3cccc(C(F)(F)F)n3)n2)Nc2cc1cc(C(F)(F)F)c2 CHEMBL4784579 IC50 699.0 nM
O=S(=O)(NC1CC1)c1ccc(-c2ccsc2)c(Nc2nc3cc(F)ccc3[nH]2)c1 CHEMBL4646777 IC50 730.0 nM
FC(F)(F)c1cccc(Nc2nc(Nc3cccc(C(F)(F)F)c3)nc(NC3CCCNC3)n2)c1 CHEMBL5431662 IC50 769.0 nM
NC1CCCN(c2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)c3)n2)C1 CHEMBL5406596 IC50 909.0 nM
Cc1cc(C)c2[nH]c(Nc3cc(S(=O)(=O)NC4CC4)ccc3-c3ccsc3)nc2c1 CHEMBL4639434 IC50 960.0 nM
CN1CCC(Nc2nc(Nc3cccc(C(F)(F)F)c3)nc(Nc3cccc(C(F)(F)F)c3)n2)CC1 CHEMBL5437900 IC50 989.0 nM
