O=C1CC[C@H](N2Cc3c(OCc4ccc(CN5CCOCC5)cc4)cccc3C2=O)C(=O)N1 CHEMBL3989927 DC50 1.7 nM
O=C1CCC(N2Cc3cc(C4CCN(Cc5csc(-c6ccccc6)n5)CC4)ccc3C2=O)C(=O)N1 CHEMBL5094460 EC50 39.0 nM
O=C1CCC(N2Cc3cc(C4CCN(Cc5nc(-c6ccccc6)c[nH]5)CC4)ccc3C2=O)C(=O)N1 CHEMBL5086132 EC50 43.0 nM
Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O CHEMBL43452 AC50 50.0 nM
COc1c(C2=CCN(Cc3ccccc3)CC2)ccc2c1CN(C1CCC(=O)NC1=O)C2=O CHEMBL5422767 AC50 66.0 nM
O=C1CCC(N2Cc3cccc(OCc4ccc(CN5CCOCC5)cc4)c3C2)C(=O)N1 CHEMBL5400126 DC50 90.0 nM
CO[C@H]1CC[C@H](CN2CCC(c3ccc4c(c3Cl)CN(C3CCC(=O)NC3=O)C4=O)CC2)CC1 CHEMBL5399912 AC50 130.0 nM
CC(C)(C)c1cccc(CN2CCC(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)c1 CHEMBL5088556 EC50 140.0 nM
O=C1CCC(N2Cc3ccccc3C2=O)C(=O)N1 CHEMBL304572 DC50 193.0 nM
CN(C)S(=O)(=O)c1cccc(CN2CCC(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)c1 CHEMBL5072327 EC50 220.0 nM
O=C1CCC(N2Cc3cc(C4=CCN(Cc5ccccc5)CC4)ccc3C2=O)C(=O)N1 CHEMBL5088587 EC50 250.0 nM
CC(C)Oc1cccc(CN2CCC(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)n1 CHEMBL5077358 EC50 320.0 nM