Cc1ncccc1NC(=O)c1ccc2c(c1)CC[C@@H]1C[C@@](O)(CCC(F)(F)F)CC[C@@]21Cc1ccccc1 CHEMBL3647441 IC50 1.1 nM
Cc1ncccc1NC(=O)c1ccc2c(c1)C(=O)C[C@@H]1C[C@@](O)(C(F)(F)F)CC[C@@]21Cc1ccccc1 CHEMBL3647443 IC50 1.1 nM
Cc1ccncc1NC(=O)c1ccc2c(c1)CC[C@@H]1C[C@@](O)(C(F)(F)F)CC[C@@]21Cc1ccccc1 CHEMBL3647442 IC50 1.3 nM
Cc1c(NC(=O)c2ccc3c(c2)CC[C@@H]2C[C@@](O)(C(F)(F)F)CC[C@@]32Cc2ccccc2)ccc[n+]1[O-] CHEMBL3647445 IC50 2.1 nM
Cc1ncccc1NC(=O)c1ccc2c(c1)C=C[C@@H]1C[C@@](O)(C(F)(F)F)CC[C@@]21Cc1ccccc1 CHEMBL3647447 IC50 2.8 nM
Cc1cnc(NC(=O)c2ccc3c(c2)CC[C@@H]2C[C@@](O)(C(F)(F)F)CC[C@@]32Cc2ccccc2)c(C)n1 CHEMBL3647440 IC50 4.0 nM
C[C@]12C=CC(=O)C=C1CC[C@@H]1[C@@H]2[C@@H](O)C[C@@]2(C)[C@H]1CC[C@]2(O)C(=O)CO CHEMBL131 IC50 4.2 nM
Cc1ncccc1NC(=O)c1ccc2c(c1)CC[C@@H]1C[C@@](O)(C(F)F)CC[C@@]21Cc1ccccc1 CHEMBL3647446 IC50 4.3 nM
Cc1ncccc1NC(=O)c1ccc2c(c1)[C@H](O)C[C@@H]1C[C@@](O)(C(F)(F)F)CC[C@@]21Cc1ccccc1 CHEMBL3647444 IC50 7.0 nM
CCS(=O)(=O)c1cc2cc(C[C@](O)(CC(C)(C)c3ccc(F)cc3C(N)=O)C(F)(F)F)[nH]c2cn1 CHEMBL3358954 IC50 23.0 nM
Cc1ncccc1NC(=O)c1ccc2c(c1)CC[C@@H]1C[C@@](OP(=O)(O)O)(C(F)(F)F)CC[C@@]21Cc1ccccc1 CHEMBL3137316 IC50 60.0 nM
COc1c(O)cc2c(c1O)[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1OC2=O CHEMBL273019 IC50 208.0 nM
Cc1ncc(NC(=O)c2ccc3c(c2)CC[C@@H]2C[C@@](O)(CCC(F)(F)F)CC[C@@]32Cc2ccccc2)c(C)n1 CHEMBL3647448 IC50 291.0 nM
CCOC(=O)C1=C(C)NC2S/C(=C\c3ccc(N4CCOCC4)cc3)C(=O)N2C1c1cccs1 CHEMBL5282465 IC50 560.0 nM
C=CCOc1ccc(C2C(C(=O)OCC)=C(C)NC3S/C(=C\c4ccc(N5CCOCC5)cc4)C(=O)N32)cc1 CHEMBL5289737 IC50 600.0 nM
CCOC(=O)C1=C(C)N=c2s/c(=C\c3ccc(N4CCOCC4)cc3)c(=O)n2C1c1ccccc1 CHEMBL2391027 IC50 860.0 nM