O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1ccco1 CHEMBL48848 EC50 9.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cccs1 CHEMBL50374 EC50 12.0 nM
N#Cc1cccc(C(=O)Nc2c(C(O)(C(F)(F)F)C(F)(F)F)ccc3ccccc23)c1 CHEMBL49806 EC50 12.0 nM
CCC(=O)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL50760 EC50 15.0 nM
CC(=O)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL299167 EC50 18.0 nM
Cc1cccc(C(=O)Nc2c(C(O)(C(F)(F)F)C(F)(F)F)ccc3ccccc23)c1 CHEMBL300958 EC50 23.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cnco1 CHEMBL48797 EC50 24.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cccc(F)c1 CHEMBL49787 EC50 44.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1ccccc1 CHEMBL51071 EC50 44.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)C1CCC1 CHEMBL47170 EC50 45.0 nM
CC(C)=CC(=O)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL300969 EC50 46.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1ccc(Br)cc1 CHEMBL298866 EC50 47.0 nM
CC(C)CCC(=O)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL49116 EC50 49.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cccnc1 CHEMBL49076 EC50 60.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1ccc(F)cc1 CHEMBL48291 EC50 70.0 nM
C/C=C/C(=O)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL49153 EC50 72.0 nM
Cc1ccc(C(=O)Nc2c(C(O)(C(F)(F)F)C(F)(F)F)ccc3ccccc23)cc1 CHEMBL296954 EC50 76.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cccc(Br)c1 CHEMBL298383 EC50 80.0 nM
O=C(CC1CCCC1)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL45937 EC50 81.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cccc(C(F)(F)F)c1 CHEMBL298970 EC50 84.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cccc(Cl)c1 CHEMBL301296 EC50 98.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cccc([N+](=O)[O-])c1 CHEMBL295458 EC50 117.0 nM
CCCC(=O)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL49797 EC50 131.0 nM
CC(=O)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2c(O)cccc12 CHEMBL49701 EC50 137.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1ccc(I)cc1 CHEMBL51460 EC50 154.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1ccc(C(F)(F)F)cc1 CHEMBL48801 EC50 160.0 nM
COc1cccc(C(=O)Nc2c(C(O)(C(F)(F)F)C(F)(F)F)ccc3ccccc23)c1 CHEMBL48765 EC50 185.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1ccc(Cl)c(Cl)c1 CHEMBL46244 EC50 194.0 nM
COCC(=O)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL45749 EC50 213.0 nM
O=C(Nc1ccc(Cl)cc1)Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12 CHEMBL48174 EC50 276.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cc(Cl)cc(Cl)c1 CHEMBL49348 EC50 306.0 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1cnc2ccccc2n1 CHEMBL301591 EC50 317.0 nM
CC(Cl)(Cl)[C@@H](NC(=O)c1ccc(Cl)cc1)N/C(=N/C#N)Nc1cccnc1 CHEMBL239512 Log EC50 338.84 nM
COc1ccc(C(=O)Nc2c(C(O)(C(F)(F)F)C(F)(F)F)ccc3ccccc23)cc1 CHEMBL48615 EC50 417.0 nM
C[C@](O)(C(=O)Nc1ccc(C(=O)c2ccccc2)cc1)C(F)(F)F CHEMBL18861 Log EC50 436.52 nM
CC(Cl)(Cl)C(NC(=O)c1ccc(Cl)cc1)N/C(=N/C#N)Nc1ccc(Cl)nc1 CHEMBL239514 Log EC50 457.09 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)C1CCCC1 CHEMBL49191 EC50 495.0 nM
CC(Cl)(Cl)C(NC(=O)c1ccc(Br)cc1)N/C(=N/C#N)Nc1ccc(Cl)nc1 CHEMBL391369 Log EC50 537.03 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)c1ccc(Cl)cc1 CHEMBL296931 EC50 570.0 nM
CC(Cl)(Cl)C(NC(=O)c1ccc(Cl)cc1)N/C(=N/C#N)Nc1cncc(Br)c1 CHEMBL393831 Log EC50 645.65 nM
O=C(Nc1c(C(O)(C(F)(F)F)C(F)(F)F)ccc2ccccc12)C1CC1 CHEMBL296840 EC50 751.0 nM
Cc1cncc(N/C(=N\C#N)NC(NC(=O)c2ccc(Cl)cc2)C(C)(Cl)Cl)c1 CHEMBL238883 Log EC50 758.58 nM
CC(Cl)(Cl)C(NC(=O)c1cccc(Cl)c1)N/C(=N/C#N)Nc1cncc(Br)c1 CHEMBL241199 Log EC50 776.25 nM
CC(Cl)(Cl)C(NC(=O)c1cc(Cl)cc(Cl)c1)N/C(=N/C#N)Nc1ccc(Cl)nc1 CHEMBL239119 Log EC50 812.83 nM
CC(Cl)(Cl)C(NC(=O)c1ccc(I)cc1)N/C(=N/C#N)Nc1ccc(Cl)nc1 CHEMBL239121 Log EC50 891.25 nM
Cc1ccc(C(=O)NC(N/C(=N/C#N)Nc2ccc(Cl)nc2)C(C)(Cl)Cl)cc1 CHEMBL239128 Log EC50 912.01 nM
CC(Cl)(Cl)C(NC(=O)c1ccc(F)cc1)N/C(=N/C#N)Nc1cncc(Br)c1 CHEMBL393424 Log EC50 954.99 nM