Cc1cc(N2CCc3sccc3C2)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4250878 EC50 20.0 nM
Cc1cc(N2CCc3ccsc3C2)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4238783 EC50 20.0 nM
Cc1cc2c(s1)CN(c1cc(C)c(NC(=O)CC(C)(C)C)c(C)c1)CC2 CHEMBL4250403 EC50 30.0 nM
Cc1cc(N2CCn3cccc3C2)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4247074 EC50 34.0 nM
Cc1ccc2c(c1)CCCCN2c1cc(C)c(NC(=O)CC(C)(C)C)c(C)c1 CHEMBL4247002 EC50 40.0 nM
O=C1c2ccccc2C(Cc2ccnc(F)c2)(Cc2ccnc(F)c2)c2ccccc21 CHEMBL343822 IC50 48.0 nM
CCOC(=O)Nc1cc(F)c(NCc2ccc(C(F)(F)F)cc2)c(F)c1N CHEMBL5185685 EC50 50.0 nM
O=C1c2ccccc2C(Cc2ccncc2)(Cc2ccncc2)c2ccccc21 CHEMBL342375 IC50 55.0 nM
CC[C@H](C(=O)Nc1ccccc1N1CCCC1)c1ccccc1 CHEMBL2164048 IC50 70.0 nM
CCCCCCC(=O)Nc1ccc2c(ccn2Cc2ccc(C(F)(F)F)cc2)c1 CHEMBL4545892 EC50 80.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(OC)c1 CHEMBL2163658 IC50 120.0 nM
Cc1cc(N2CCc3sc(C(F)(F)F)cc3C2)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4246596 EC50 120.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(F)cc1 CHEMBL2164068 IC50 130.0 nM
Cc1cc(N2CCC(=O)CC2)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4128096 EC50 130.0 nM
Cc1cc(N2CCCCc3cc(Cl)ccc32)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4250839 EC50 140.0 nM
O=C1c2ccccc2C(Cc2ccnnc2)(Cc2c(F)cncc2F)c2ccccc21 CHEMBL4465132 IC50 160.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1 CHEMBL1464225 IC50 163.0 nM
O=C(Cc1cccc(Cl)c1)Nc1ccccc1N1CCCC1 CHEMBL2163660 EC50 170.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(F)c(F)c1 CHEMBL2164062 IC50 170.0 nM
O=C1c2ccccc2C(Cc2c(F)cncc2F)(Cc2c(F)cncc2F)c2ccccc21 CHEMBL4471453 IC50 200.0 nM
CCC(C(=O)Nc1ccc(N2CCCC2)cc1)c1ccccc1 CHEMBL2163667 IC50 210.0 nM
Cc1cc(N2CCC(c3cccc(F)c3)CC2)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4125892 EC50 220.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(Cl)c1 CHEMBL2163659 IC50 240.0 nM
Cc1cc(N2CCCCc3cc(F)ccc32)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4246564 EC50 250.0 nM
CC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1 CHEMBL2164049 IC50 260.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(Cl)cc1 CHEMBL2163662 IC50 280.0 nM
Cc1cc(N2CCc3sc(C#N)cc3C2)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4246239 EC50 290.0 nM
Cc1csc2c1CN(c1cc(C)c(NC(=O)CC(C)(C)C)c(C)c1)CC2 CHEMBL4244768 EC50 300.0 nM
CCCC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1 CHEMBL2164054 IC50 320.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(C)c1 CHEMBL2164066 IC50 330.0 nM
O=C(Nc1ccccc1N1CCCC1)C1CCc2ccccc21 CHEMBL2164055 IC50 330.0 nM
Cc1cc(CN2CCCc3ccccc32)cc(C)c1NC(=O)CC(C)(C)C CHEMBL4126113 EC50 330.0 nM
O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccccc1N1CCCC1 CHEMBL1572950 EC50 350.0 nM
CCOC(=O)Nc1ccc(NCc2ccc(F)cc2)cc1N CHEMBL41355 EC50 350.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(F)c1 CHEMBL2164064 IC50 360.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(OC)cc1 CHEMBL2163661 IC50 380.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1cccc(C(F)(F)F)c1 CHEMBL2163657 IC50 390.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccccc1F CHEMBL2163664 IC50 440.0 nM
CCC(C(=O)Nc1ccccc1N1CCCC1)c1ccc(Cl)c(Cl)c1 CHEMBL2164069 IC50 470.0 nM
O=C(Cc1cccc(F)c1)Nc1ccccc1N1CCCC1 CHEMBL2164065 EC50 490.0 nM
Cc1cc(CC2(Cc3ccnc(C)c3)c3ccccc3C(=O)c3ccccc32)ccn1 CHEMBL4447214 IC50 540.0 nM
CC(C)(C)CC(=O)Nc1ccc2c(ccn2Cc2ccc(C(F)(F)F)cc2)c1 CHEMBL4457044 EC50 630.0 nM
C[C@H](NC(=O)/C=C/c1ccccc1)c1cccc(N2CCOCC2)c1 CHEMBL317935 EC50 690.0 nM
O=C(Cc1ccc(F)cc1)Nc1ccccc1N1CCCC1 CHEMBL1415708 EC50 700.0 nM
O=C(Cc1ccccc1)Nc1ccccc1N1CCCC1 CHEMBL1448089 EC50 743.0 nM
O=C(Cc1ccc(Cl)cc1)Nc1ccccc1N1CCCC1 CHEMBL2163663 EC50 800.0 nM
O=C(Cc1ccccc1Cl)Nc1ccccc1N1CCCC1 CHEMBL2163656 EC50 950.0 nM
[2H]c1cc(NC(=O)OCC)c(N)c(F)c1NCc1ccc(C(F)(F)F)cc1 CHEMBL5186399 EC50 980.0 nM
O=C(Nc1ccccc1N1CCCC1)C(F)c1ccccc1 CHEMBL2164050 EC50 990.0 nM
C#CCN(Cc1ccc(F)cc1)c1ccc(NC(=O)OCC)c(N)c1 CHEMBL5174234 EC50 990.0 nM