COc1ccc(-c2c(-c3cc(C(=O)O)ccn3)ncn2C)cc1 CHEMBL3786803 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1-c1ccc(OCC2CC2)cc1 CHEMBL3787664 IC50 100.0 nM
Cc1cc(Cl)ccc1COc1ccnn1-c1cc(C(=O)O)ccn1 CHEMBL3786952 IC50 100.0 nM
CCN(CCN(C)C)C(=O)CNCc1cc(C(=O)O)ccn1 CHEMBL3787669 IC50 100.0 nM
Cc1cc(O)n(-c2cc(C(=O)O)ccn2)n1 CHEMBL4286275 IC50 100.0 nM
Cc1nn(-c2cc(C(=O)O)ccn2)c(O)c1C CHEMBL4292883 IC50 100.0 nM
Cc1nn(-c2cc(C(=O)O)ccn2)c(O)c1-c1ccccc1 CHEMBL4293636 IC50 100.0 nM
CCCc1cc(O)n(-c2cc(C(=O)O)ccn2)n1 CHEMBL4287794 IC50 100.0 nM
O=C(O)c1ccnc(-n2nccc2O)c1 CHEMBL4287317 IC50 100.0 nM
O=C(O)c1ccnc(-n2nccc2OCc2ccc3cn[nH]c3c2)c1 CHEMBL4285840 IC50 100.0 nM
Cn1ncc2ccc(COc3ccnn3-c3cc(C(=O)O)ccn3)cc21 CHEMBL4290631 IC50 100.0 nM
O=C(O)c1ccnc(-n2nccc2OCc2ccc(Cl)cc2OCc2ccccc2)c1 CHEMBL4227526 IC50 100.0 nM
O=C(O)c1ccnc(-n2nc(Cc3cc(Cl)cc(Cl)c3)cc2O)c1 CHEMBL4281922 IC50 100.0 nM
Cn1cnc(-c2cc(-c3c[nH]nn3)ccn2)c1 CHEMBL4281254 IC50 100.0 nM
Fc1c(Cn2cnc(-c3cc(-c4c[nH]nn4)ccn3)c2)cccc1OC(F)(F)F CHEMBL4289127 IC50 100.0 nM
c1ccc(-c2ccccc2CCn2cnc(-c3cc(-c4c[nH]nn4)ccn3)c2)cc1 CHEMBL4292175 IC50 100.0 nM
CC(Cc1ccccc1)n1cnc(-c2cc(-c3c[nH]nn3)ccn2)c1 CHEMBL4291030 IC50 100.0 nM
FC(F)(F)Cn1cnc(-c2cc3[nH]nnc3cn2)c1 CHEMBL4287712 IC50 100.0 nM
Clc1cccc(-n2cnc(-c3cc4[nH]nnc4cn3)c2)c1 CHEMBL4283409 IC50 100.0 nM
Clc1cc(Cl)cc(-n2cnc(-c3cc4[nH]nnc4cn3)c2)c1 CHEMBL4294250 IC50 100.0 nM
Cn1cnc(-c2cc3[nH]nnc3cn2)c1-c1ccc(F)cc1 CHEMBL4286185 IC50 100.0 nM
Cn1cnc(-c2cc3[nH]nnc3cn2)c1-c1ccc(F)cc1OCC1CC1 CHEMBL4289929 IC50 100.0 nM
CCOc1ccccc1CCn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4276861 IC50 100.0 nM
FC(F)(F)c1ccccc1CCn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4278662 IC50 100.0 nM
CC(C)C(c1ccccc1)n1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4293028 IC50 100.0 nM
FC(F)(F)COc1ccccc1Cn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4279214 IC50 100.0 nM
Fc1cccc(Cl)c1CCn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4289631 IC50 100.0 nM
FC(F)(F)c1[nH]nnc1-c1ccnc(-c2cn(CC3CCc4ccccc43)cn2)c1 CHEMBL4289252 IC50 100.0 nM
FC(F)(F)c1ccc(CCn2cnc(-c3cc(-c4nn[nH]c4C(F)(F)F)ccn3)c2)cc1 CHEMBL4285698 IC50 100.0 nM
CCc1ccc(CCn2cnc(-c3cc(-c4nn[nH]c4C(F)(F)F)ccn3)c2)cc1 CHEMBL4287332 IC50 100.0 nM
CC(C)(C)c1ccc(CCn2cnc(-c3cc(-c4nn[nH]c4C(F)(F)F)ccn3)c2)cc1 CHEMBL4281270 IC50 100.0 nM
Fc1cccc2c1CCCC2Cn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4286353 IC50 100.0 nM
Fc1ccc2c(c1)CCCC2Cn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4286728 IC50 100.0 nM
Fc1ccc2c(c1)C(Cn1cnc(-c3cc(-c4nn[nH]c4C(F)(F)F)ccn3)c1)CCC2 CHEMBL4287778 IC50 100.0 nM
Cc1ccc2c(c1)C(Cn1cnc(-c3cc(-c4nn[nH]c4C(F)(F)F)ccn3)c1)CCC2 CHEMBL4291852 IC50 100.0 nM
COc1cccc2c1CCCC2Cn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4294417 IC50 100.0 nM
COc1ccc2c(c1)CCCC2Cn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4277381 IC50 100.0 nM
COc1ccc2c(c1)C(Cn1cnc(-c3cc(-c4nn[nH]c4C(F)(F)F)ccn3)c1)CCC2 CHEMBL4277565 IC50 100.0 nM
COc1cccc2c1C(Cn1cnc(-c3cc(-c4nn[nH]c4C(F)(F)F)ccn3)c1)CCC2 CHEMBL4292396 IC50 100.0 nM
FC(F)(F)c1[nH]nnc1-c1ccnc(-c2cn(CCc3cccc4ccccc34)cn2)c1 CHEMBL4294747 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1Br CHEMBL4278863 IC50 100.0 nM
Cc1ccc(-c2c(-c3cc(C(=O)O)ccn3)ncn2C)cc1O CHEMBL4292111 IC50 100.0 nM
Cc1ccc(-c2c(-c3cc(C(=O)O)ccn3)ncn2C)cc1 CHEMBL4288406 IC50 100.0 nM
CCc1ccc(-c2c(-c3cc(C(=O)O)ccn3)ncn2C)cc1 CHEMBL4288034 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1-c1ccc(C(F)(F)F)cc1 CHEMBL4286983 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1-c1ccc(C2CC2)cc1 CHEMBL4284869 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1-c1cccc(CO)c1 CHEMBL4293936 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1-c1ccc(OC(F)(F)F)cc1 CHEMBL4288145 IC50 100.0 nM
CCOc1ccc(-c2c(-c3cc(C(=O)O)ccn3)ncn2C)cc1 CHEMBL4285443 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1-c1ccc(-n2cccn2)cc1 CHEMBL4286418 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1-c1ccc(Cl)c(Cl)c1 CHEMBL4286705 IC50 100.0 nM
Cn1cnc(-c2cc(C(=O)O)ccn2)c1-c1ccc(Cl)c(C(F)(F)F)c1 CHEMBL4283146 IC50 100.0 nM
CCOc1cc(Cl)ccc1-c1c(-c2cc(C(=O)O)ccn2)ncn1C CHEMBL4277960 IC50 100.0 nM
O=C(O)c1ccnc(-c2cn(CCn3cccn3)cn2)c1 CHEMBL4290028 IC50 100.0 nM
CN(C)CCOCCn1cnc(-c2cc(C(=O)O)ccn2)c1 CHEMBL4279284 IC50 100.0 nM
CN1CCC(n2cnc(-c3cc(C(=O)O)ccn3)c2)CC1 CHEMBL4291702 IC50 100.0 nM
O=C(O)c1ccnc(-c2cn(C3CCNC3)cn2)c1 CHEMBL4286314 IC50 100.0 nM
O=C(O)c1ccnc(-c2cn(CC3CCCN3)cn2)c1 CHEMBL4286674 IC50 100.0 nM
CN(CCn1cnc(-c2cc(C(=O)O)ccn2)c1)CC1CC1 CHEMBL4288025 IC50 100.0 nM
c1cc(-c2nn[nH]n2)cc(-c2cn(CCN3CCCC3)cn2)n1 CHEMBL4283417 IC50 100.0 nM
O=C(O)c1ccnc(-c2cn(CCN3CCc4cc(F)ccc43)cn2)c1 CHEMBL4293359 IC50 100.0 nM
Cc1ccc(OCC2CC2)c(-c2c(-c3cc(C(=O)O)ccn3)ncn2C)c1 CHEMBL4279372 IC50 100.0 nM
Clc1ccc(-c2c(-c3cc(-c4nn[nH]n4)ccn3)ncn2CCc2ccccc2Cl)cc1 CHEMBL4288414 IC50 100.0 nM
CC(C)COc1ccccc1Cn1cnc(-c2cc(-c3nn[nH]n3)ccn2)c1 CHEMBL4283306 IC50 100.0 nM
Cn1cnc(-c2cc(-c3nn[nH]n3)ccn2)c1-c1ccc(F)c(OCC(F)(F)F)c1 CHEMBL4294432 IC50 100.0 nM
Cn1cnc(-c2cc(-c3nn[nH]n3)ccn2)c1-c1ccc(F)c(C(=O)Nc2ccccc2)c1 CHEMBL4294755 IC50 100.0 nM
CC(=O)OCn1nnc(-c2ccnc(-c3cn(Cc4ccccc4Cl)cn3)c2)n1 CHEMBL4290020 IC50 100.0 nM
Fc1ccc(-c2c(-c3cc(-c4nn[nH]n4)ccn3)ncn2Cc2cccc(Cl)c2)c(OCC2CC2)c1 CHEMBL4290366 IC50 100.0 nM
O=C(O)c1ccnc(-n2nccc2Cc2ccccc2)c1 CHEMBL4285977 IC50 1000.0 nM
O=C(O)c1ccnc(-n2ccc(Cc3ccccc3)n2)c1 CHEMBL4284987 IC50 1000.0 nM
Cc1ccc(COc2ccnn2-c2cc(C(=O)O)ccn2)cc1 CHEMBL4228087 IC50 1000.0 nM
CCc1ccc(COc2ccnn2-c2cc(C(=O)O)ccn2)cc1 CHEMBL4227237 IC50 1000.0 nM
Cc1ccc(COc2ccnn2-c2cc(C(=O)O)ccn2)cc1Cl CHEMBL4286133 IC50 1000.0 nM
N#Cc1ccc(COc2ccnn2-c2cc(C(=O)O)ccn2)cc1 CHEMBL4229271 IC50 1000.0 nM
O=C(O)c1ccnc(-n2nccc2OCc2ccc(Cl)cc2OCC2CC2)c1 CHEMBL4225515 IC50 1000.0 nM
O=C(O)c1ccnc(-n2nccc2OCc2ccc(Cl)cc2OCC(F)(F)F)c1 CHEMBL4292430 IC50 1000.0 nM
CCCCOc1cc(Cl)ccc1COc1ccnn1-c1cc(C(=O)O)ccn1 CHEMBL4287296 IC50 1000.0 nM
CC(C)COc1cc(Cl)ccc1COc1ccnn1-c1cc(C(=O)O)ccn1 CHEMBL4281159 IC50 1000.0 nM
O=C(O)c1ccnc(-n2nccc2OCc2ccc(Cl)cc2OCc2ccc(F)cc2)c1 CHEMBL4289695 IC50 1000.0 nM
O=C(O)c1ccnc(-n2nccc2OCc2ccc(F)cc2OCc2ccc(F)cc2)c1 CHEMBL4290069 IC50 1000.0 nM
Cc1ccc(COc2ccnn2-c2cc(C(=O)O)ccn2)c(Cl)c1 CHEMBL4283926 IC50 1000.0 nM
Cc1ccc(COc2ccnn2-c2cc(C(=O)O)ccn2)c(C)c1 CHEMBL4289921 IC50 1000.0 nM
COc1cc(C)ccc1COc1ccnn1-c1cc(C(=O)O)ccn1 CHEMBL4288884 IC50 1000.0 nM
O=C(O)c1ccnc(-n2nccc2OCc2ccc(Cl)c(OCC3CC3)c2)c1 CHEMBL4287561 IC50 1000.0 nM
Cc1ccc2c(c1)CCCC2Cn1cnc(-c2cc(-c3nn[nH]c3C(F)(F)F)ccn2)c1 CHEMBL4290800 IC50 1000.0 nM
Cn1cnc(-c2cc(-c3nn[nH]c3F)ccn2)c1-c1ccc(F)cc1OCC1CC1 CHEMBL4277370 IC50 1000.0 nM
O=C(O)c1ccnc(-c2cn(CCN3CCCC3)cn2)c1 CHEMBL4294777 IC50 1000.0 nM
CN1CCC(Cn2cnc(-c3cc(C(=O)O)ccn3)c2)CC1 CHEMBL4287989 IC50 1000.0 nM
CC(=O)OCn1nnc(-c2ccnc(-c3ncn(Cc4ccccc4Cl)c3-c3ccc(F)cc3)c2)n1 CHEMBL4289480 IC50 1000.0 nM
CC(C)(C)C(=O)OCn1nnc(-c2ccnc(-c3ncn(Cc4ccccc4Cl)c3-c3ccc(F)cc3)c2)n1 CHEMBL4285770 IC50 1000.0 nM
Cn1nnc(-c2ccnc(-c3cn(Cc4ccccc4Cl)cn3)c2)n1 CHEMBL4285921 IC50 1000.0 nM
CC(C)(C)C(=O)OCn1nnc(-c2ccnc(-c3cn(Cc4ccccc4Cl)cn3)c2)n1 CHEMBL4286299 IC50 1000.0 nM