COc1ccccc1-c1ccc([C@H](C)Nc2cncc(N3C(=O)OC[C@@H]3C(C)C)n2)cc1 CHEMBL4210711 pIC50 2.512 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)C(OC(=O)Cc1c(C)[nH]c2ccccc12)C(F)(F)F CHEMBL4217078 IC50 18.0 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cc1c(C)[nH]c2cc(C(=N)N)ccc12 CHEMBL4206734 IC50 23.0 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cc1c(C)[nH]c2cnccc12 CHEMBL4216138 IC50 100.0 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cc1c(C)[nH]c2ccc(C(=N)N)cc12 CHEMBL4212718 IC50 100.0 nM
C#Cc1ccc2c(CC(=O)OCC(=O)Nc3c(C)nn(-c4ccccc4)c3C)c(C)[nH]c2c1 CHEMBL4210314 IC50 130.0 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cc1c(C)[nH]c2ccccc12 CHEMBL4218203 IC50 130.0 nM
C#Cc1[nH]c2ccccc2c1CC(=O)OCC(=O)Nc1c(C)nn(-c2ccccc2)c1C CHEMBL4203947 IC50 150.0 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cc1c(C)[nH]c2ncccc12 CHEMBL4211164 IC50 190.0 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cc1c(C)[nH]c2ccc(Cl)cc12 CHEMBL4207925 IC50 250.0 nM
C#Cc1ccc2[nH]c(C)c(CC(=O)OCC(=O)Nc3c(C)nn(-c4ccccc4)c3C)c2c1 CHEMBL4214705 IC50 250.0 nM
Cc1[nH]c2ccccc2c1CC(=O)NCC(=O)Nc1cnn(-c2ccccc2)c1C CHEMBL4218314 IC50 290.0 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cc1c(C)[nH]c2ccncc12 CHEMBL4211677 IC50 490.0 nM
Cc1nn(-c2ccccc2)c(C)c1NC(=O)COC(=O)Cn1c(C)cc2ccccc21 CHEMBL4212332 IC50 640.0 nM
NCc1ccc(NC(=O)c2cc3ccccc3cc2O)cc1 CHEMBL4861066 Ki 800.0 nM
NCc1ccc(NC(=O)c2c([O-])ccc[n+]2Cc2nccn2Cc2ccccc2)cc1 CHEMBL4208878 IC50 890.0 nM
COc1ccc2c(O)c(C(=O)Nc3ccc(CN)cc3)ccc2c1 CHEMBL4862261 Ki 1000.0 nM