O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c(Nc2ccccc2)c1)N1CCC(N2CCCC2)CC1 CHEMBL2426364 IC50 24.0 nM
Clc1cc(N2CCC(N3CCCC3)CC2)ccc1CCN1CCCC1 CHEMBL3134130 IC50 37.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c(NCc2ccccc2)c1)N1CCC(N2CCCC2)CC1 CHEMBL2426365 IC50 39.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c2ccccc12)N1CCC(N2CCCC2)CC1 CHEMBL2426360 IC50 43.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c(Cc2ccccc2)c1)N1CCC(N2CCCC2)CC1 CHEMBL2426366 IC50 48.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)cc1)N1CCC(N2CCCC2)CC1 CHEMBL2426498 IC50 48.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CCN1CCC1 CHEMBL3134144 IC50 48.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c(Oc2ccccc2)c1)N1CCC(N2CCCC2)CC1 CHEMBL2426367 IC50 53.0 nM
OCC1(CO)CN(CCc2ccc(N3CCC(N4CCCC4)CC3)cc2)C1 CHEMBL3134146 IC50 59.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c(-c2ccccc2)c1)N1CCC(N2CCCC2)CC1 CHEMBL2426368 IC50 61.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)nc1)N1CCC(N2CCCC2)CC1 CHEMBL2424678 IC50 61.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CCN1CCCC1 CHEMBL3134131 IC50 62.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)s1)N1CCC(N2CCCC2)CC1 CHEMBL2426363 IC50 68.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CCCN1CCCC1 CHEMBL3134134 IC50 70.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c(Br)c1)N1CCC(N2CCCC2)CC1 CHEMBL2426476 IC50 74.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)cc1)N1CCCC(N2CCCC2)CC1 CHEMBL2426496 IC50 74.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CCN1CCCCC1 CHEMBL3134126 IC50 80.0 nM
C[N+]1(C2CCN(C(=O)c3ccc(C(=O)N4CCC(N5CCCC5)CC4)cc3)CC2)CCCC1 CHEMBL2426489 IC50 81.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c([N+](=O)[O-])c1)N1CCC(N2CCCC2)CC1 CHEMBL2426477 IC50 88.0 nM
O=C(c1ccc(C(=O)N2CC3CCC(C2)C3N2CCCC2)cc1)N1CCC(N2CCCC2)CC1 CHEMBL2426495 IC50 92.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)cc1)N1CCC(C2CCCN2)CC1 CHEMBL2426490 IC50 92.0 nM
O=C(c1ccc(S(=O)(=O)N2CCC(N3CCCC3)CC2)cc1)N1CCC(N2CCCC2)CC1 CHEMBL2426481 IC50 97.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CCN1CCCCCC1 CHEMBL3134125 IC50 100.0 nM
O=C(c1ccc(C(=O)N2CCCC(N3CCCC3)CC2)cc1)N1CCCC(N2CCCC2)CC1 CHEMBL2426469 IC50 110.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)c(C(=O)N2CCC(N3CCCC3)CC2)c1)N1CCC(N2CCCC2)CC1 CHEMBL2426480 IC50 110.0 nM
c1cc(CN2CCCC2)cc(N2CCC(N3CCCC3)CC2)c1 CHEMBL3134136 IC50 120.0 nM
c1cc(CCN2CCCC2)cc(N2CCC(N3CCCC3)CC2)c1 CHEMBL3134135 IC50 120.0 nM
CCN1Cc2ccc(NC(=O)c3ccc(C(=O)N4CCC(C5CCCN5)CC4)c(Nc4ccccc4)c3)cc2C1 CHEMBL2424677 IC50 130.0 nM
O=C(c1c(F)c(F)c(C(=O)N2CCC(N3CCCC3)CC2)c(F)c1F)N1CCC(N2CCCC2)CC1 CHEMBL2426358 IC50 130.0 nM
O=C(c1ccc(CN2CCC(N3CCCC3)CC2)cc1)N1CCC(N2CCCC2)CC1 CHEMBL2426483 IC50 130.0 nM
CCN1Cc2ccc(NC(=O)c3ccc(C(=O)N4CC5CCC(C4)C5N4CCCC4)cc3)cc2C1 CHEMBL2426374 IC50 150.0 nM
O=C(c1ccc(N2CCC(N3CCCC3)CC2)cc1)N1CCC(N2CCCC2)CC1 CHEMBL2426482 IC50 150.0 nM
CCN1Cc2ccc(NC(=O)c3ccc(C(=O)N4CCC(C5CCCN5)CC4)cc3Nc3ccccc3)cc2C1 CHEMBL2426376 IC50 160.0 nM
CCN1Cc2ccc(NC(=O)c3ccc(C(=O)N4CCC(C5CCCN5)CC4)cc3)cc2C1 CHEMBL2426375 IC50 160.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)cc1)N1CCC(N2CCCCC2)CC1 CHEMBL2426484 IC50 160.0 nM
CN(C)C1CCN(C(=O)c2ccc(C(=O)N3CCC(N4CCCC4)CC3)cc2)CC1 CHEMBL2426488 IC50 180.0 nM
Cc1cc(C(=O)N2CCC(N3CCCC3)CC2)c(C)cc1C(=O)N1CCC(N2CCCC2)CC1 CHEMBL2426359 IC50 210.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)cc1)N1CCC(N2CCCCCC2)CC1 CHEMBL2426485 IC50 210.0 nM
Nc1cc(C(=O)N2CCC(N3CCCC3)CC2)ccc1C(=O)N1CCC(N2CCCC2)CC1 CHEMBL2426478 IC50 220.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)C2)cc1)N1CCC(N2CCCC2)CC1 CHEMBL2426462 IC50 220.0 nM
CC(C1CCN(C(=O)c2ccc(C(=O)N3CCC(N4CCCC4)CC3)cc2)CC1)N1CCN(C)CC1 CHEMBL2426494 IC50 250.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CCN1CC2(COC2)C1 CHEMBL3134129 IC50 270.0 nM
O=C(c1ccc(C(=O)N2CC3CCC(C2)C3N2CCCC2)cc1)N1CC2CCC(C1)C2N1CCCC1 CHEMBL2426470 IC50 280.0 nM
O=C(c1cccc(C(=O)N2CCC(N3CCCC3)CC2)c1)N1CCC(N2CCCC2)CC1 CHEMBL2426497 IC50 290.0 nM
O=C(c1ccc(C(=O)N2CC(N3CCCC3)C2)cc1)N1CCC(N2CCCC2)CC1 CHEMBL2426461 IC50 300.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)o1)N1CCC(N2CCCC2)CC1 CHEMBL2426362 IC50 310.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1N1CCC(N2CCCC2)CC1 CHEMBL3134140 IC50 320.0 nM
O=C(NCCCN1CCCC1)c1ccc(C(=O)N2CCC(N3CCCC3)CC2)cc1 CHEMBL2426463 IC50 340.0 nM
CCN1Cc2ccc(NC(=O)c3ccc(C(=O)N4CCC(N5CCCC5)CC4)cc3)cc2C1 CHEMBL2426373 IC50 350.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCC3)CC2)cc1)N1CCC(N2CCC2)CC1 CHEMBL2426471 IC50 350.0 nM
O=C(c1ccccc1C(=O)N1CCC(N2CCCC2)CC1)N1CCC(N2CCCC2)CC1 CHEMBL2426479 IC50 350.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CN1CCCC1 CHEMBL3134133 IC50 350.0 nM
N#CC1CCN(CCc2ccc(N3CCC(N4CCCC4)CC3)cc2)C1 CHEMBL3134142 IC50 360.0 nM
O=C1CCN(CCc2ccc(N3CCC(N4CCCC4)CC3)cc2)C1 CHEMBL3134143 IC50 390.0 nM
O=C(c1ccc2cc(C(=O)N3CCC(N4CCCC4)CC3)ccc2c1)N1CCC(N2CCCC2)CC1 CHEMBL2426361 IC50 450.0 nM
O=C(c1ccc(C(=O)N2CCC3(CCNC3)CC2)cc1)N1CCC(N2CCCC2)CC1 CHEMBL2426466 IC50 560.0 nM
c1cc(N2CCC(N3CCCCC3)CC2)ccc1CCN1CCCC1 CHEMBL3134132 IC50 580.0 nM
O=C(c1ccc(C(=O)N2CCC(C3CCCN3)CC2)cc1)N1CCC(C2CCCN2)CC1 CHEMBL2426472 IC50 640.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CCN1CCC2(C1)OCCO2 CHEMBL3134128 IC50 650.0 nM
O=C(c1ccc(C(=O)N2CCC(N3CCCC3)CC2)cc1)N1CCC(C2CCNCC2)CC1 CHEMBL2426491 IC50 740.0 nM
CN1CCC(N2CCN(C(=O)c3ccc(C(=O)N4CCC(N5CCCC5)CC4)cc3)CC2)CC1 CHEMBL2426493 IC50 770.0 nM
c1cc(N2CCC(N3CCCC3)CC2)ccc1CCN1CCOCC1 CHEMBL3134127 IC50 850.0 nM
FC1(F)CN(CCc2ccc(N3CCC(N4CCCC4)CC3)cc2)C1 CHEMBL3134145 IC50 1000.0 nM