COc1nc(N(CC(C)(C)F)c2cc(C(F)(F)F)ccc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL3903201 IC50 0.248 nM
COc1nc(N(CC(C)C)c2cc(Cl)c(F)cc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4549822 IC50 0.28 nM
COc1nc(N(CC(C)(C)F)c2cc(Cl)c(F)cc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL3961833 IC50 0.28 nM
COc1nc(N(CC(C)C)c2cc(C(F)(F)F)ccc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4567083 IC50 0.36 nM
COc1cc(N(CC(C)C)c2ccc(F)c3ccccc23)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4464773 IC50 0.381 nM
CCCN(c1cnc(C(=O)[C@H]2C[C@@H]2C(=O)O)c(OC)n1)c1cc(Cl)c(F)cc1F CHEMBL3914270 IC50 0.483 nM
COc1cc(N(CC(C)(C)F)c2cc(Cl)c(F)cc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4562583 IC50 0.6 nM
CCCN(c1cnc(C(=O)[C@H]2C[C@@H]2C(=O)O)c(OC)c1)c1ccc(F)c2ccccc12 CHEMBL4563433 IC50 0.626 nM
COc1cc(N(CC(C)(C)F)c2cc(C(F)(F)F)ccc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4584584 IC50 0.63 nM
COc1cc(N(CC(C)C)c2cc(C(F)(F)F)ccc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL3971210 IC50 0.658 nM
COc1cc(N(CC(C)C)c2cc(Cl)c(F)cc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4574439 IC50 0.7 nM
COc1cc(N(CC2CC2)c2ccc(F)c3ccccc23)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4441362 IC50 0.758 nM
CCN(c1cnc(C(=O)[C@H]2C[C@@H]2C(=O)O)c(OC)c1)c1ccc(F)c2ccccc12 CHEMBL4476024 IC50 1.05 nM
COc1cc(N(CC2CC2)c2ccc(Cl)c3ccccc23)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4454609 fIC50 1.1 nM
COc1cc(N(CC2CC2)c2cc(Cl)c(F)cc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4545014 IC50 1.97 nM
CCOC(=O)Cc1csc(NC(=S)NC(C)c2cccc3ccccc23)n1 CHEMBL5417047 IC50 2.0 nM
COc1cc(N(CC2CC2)c2cc(C(F)(F)F)ccc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4545950 IC50 2.08 nM
COc1nc(C(=O)[C@H]2C[C@@H]2C(=O)O)ncc1N(CC1CC1)c1cccc2ccccc12 CHEMBL4525972 IC50 2.4 nM
COc1cc(N(CC2CC2)c2cc(Cl)ccc2F)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4467942 IC50 3.71 nM
COc1cc(N(CC(C)C)c2cccc(C(F)(F)F)c2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4574370 IC50 4.74 nM
COc1cc(N(CC2CC2)c2ccc(Cl)c(Cl)c2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4442047 IC50 4.94 nM
Cc1ccc(NC(=S)NC(C)c2cccc3ccccc23)nc1 CHEMBL5432381 IC50 5.0 nM
COc1cc(N(CC2CC2)c2ccc(F)c(Cl)c2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4576647 IC50 5.26 nM
COc1cc(N(CC2CC2)c2cccc(C(F)(F)F)c2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4567339 IC50 6.42 nM
CCCN(c1cccc(C(F)(F)F)c1)c1cnc(C(=O)[C@H]2C[C@@H]2C(=O)O)c(OC)c1 CHEMBL4439499 IC50 7.9 nM
COc1cc(N(CC(C)(C)F)c2cccc(C(F)(F)F)c2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4439148 IC50 8.65 nM
COc1cc(N(CC2CC2)c2ccc3c4c(cccc24)CC3)cnc1C(=O)C1CC1C(=O)O CHEMBL3910305 IC50 9.0 nM
COc1cc(N(CC(F)(F)F)c2cccc(C(F)(F)F)c2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4445815 IC50 11.5 nM
CCN(c1cccc(C(F)(F)F)c1)c1cnc(C(=O)[C@H]2C[C@@H]2C(=O)O)c(OC)c1 CHEMBL4531985 IC50 13.0 nM
COc1cc(N(Cc2ccc(F)cc2)c2cccc(C(F)(F)F)c2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4565208 IC50 13.5 nM
COc1nc(C(=O)[C@@H]2C[C@H]2C(=O)O)ncc1N(CC1CC1)c1ccc(Cl)c2ccccc12 CHEMBL4456770 IC50 15.5 nM
COc1nc(C(=O)C2CC2C(=O)O)ncc1N(CC1CC1)c1ccc(Cl)c2ccccc12 CHEMBL3938992 IC50 17.0 nM
COc1cccc(C(=O)c2ccc(C(=O)c3ccc(N(CC4CC4)c4ccc(Cl)cc4)cn3)cc2C(=O)O)c1 CHEMBL3942442 IC50 18.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)c3ccccc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3904248 IC50 18.0 nM
COc1cc(N(CC2CC2)c2ccc(F)c3ccccc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3968407 IC50 18.0 nM
COc1nc(C(=O)C2CC2C(=O)O)ncc1N(CC1CC1)c1ccc(C)c2ccccc12 CHEMBL3925432 IC50 18.0 nM
COc1cc(N(CC2CC2)c2ccc(C(F)(F)F)c3ccccc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3939700 IC50 19.0 nM
COc1nc(C(=O)C2CC2C(=O)O)ncc1N(CC1CC1)c1ccc(F)c2ccccc12 CHEMBL3947774 IC50 19.0 nM
COc1ccc(C2(C(=O)c3ccc(C(=O)c4ccc(N(C)c5ccc(Cl)cc5)cn4)cc3C(=O)O)CC2)cc1 CHEMBL3953858 IC50 22.0 nM
COc1cc(N(Cc2ccc(C)cc2)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3962857 IC50 22.0 nM
COc1cc(N(CC2CC2)c2cccc3ccccc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3943416 IC50 24.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)cc2)cnc1C(=O)[C@@H]1C[C@H]1C(=O)O CHEMBL4465323 IC50 24.3 nM
COc1cc(N(CC2CC2)c2cccc3c(C(F)(F)F)cccc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3972363 IC50 25.0 nM
COc1cc(N(CC2CC2)c2ccc(F)c3ccccc23)ccc1C(=O)C1CC1C(=O)O CHEMBL3978910 IC50 26.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3ccc4c(c3)OCCO4)c(C(=O)O)c2)nc1 CHEMBL3897151 IC50 27.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)cc2)cnc1C(=O)c1cccc(C(=O)O)c1 CHEMBL4440468 IC50 27.4 nM
COc1cc(N(CC2CC2)c2ccc3ccccc3c2)cnc1C(=O)C1CC1C(=O)O CHEMBL3920940 IC50 28.0 nM
COc1ccc(C(=O)c2ccc(C(=O)c3ccc(N(CC4CC4)c4ccc(Cl)cc4)cn3)cc2C(=O)O)cc1 CHEMBL3958548 IC50 29.0 nM
O=C(c1ccc(C(=O)c2cccc(O)c2)c(C(=O)O)c1)c1ccc(N(CC2CC2)c2ccc(Cl)cc2)cn1 CHEMBL3898467 IC50 30.0 nM
CC(C)Cc1ccc(C(C)c2nc3cc(CCC(=O)O)ccc3n2Cc2ccccc2Cl)cc1 CHEMBL4251024 IC50 30.0 nM
COc1cc(N(CC2CC2)c2ccc3cccc4c3c2CC4)cnc1C(=O)C1CC1C(=O)O CHEMBL3901235 IC50 31.0 nM
COc1cc(N(CC(C)(C)O)c2cccc(C(F)(F)F)c2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4466708 IC50 31.8 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C3(c4ccccc4)CCCCC3)c(C(=O)O)c2)nc1 CHEMBL3956435 IC50 32.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C3(c4ccccc4)CC3)c(C(=O)O)c2)nc1 CHEMBL3929575 IC50 32.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)cc2)cnc1C(=O)C1CC1C(=O)O CHEMBL3975898 IC50 34.0 nM
COc1cc(N(Cc2ccc3ccccc3c2)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3980648 IC50 34.0 nM
COc1cc(N(CC2CC2)c2ccc(C)c3ccccc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3952129 IC50 35.0 nM
COc1ccccc1C(=O)Nc1ccc(C(=O)c2ccc(N(C)c3ccc(Cl)cc3)cn2)cc1C(=O)O CHEMBL4460916 IC50 35.0 nM
COc1cc(N(CC2(C)CC2)c2ccc(Cl)cc2)cnc1C(=O)C1CC1C(=O)O CHEMBL3909825 IC50 38.0 nM
COc1cc(N(Cc2cccc(Cl)c2)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3906988 IC50 39.0 nM
COc1cc(N(CC2CC2)c2ccc(F)c3ccccc23)cnc1C(=O)C1CC1c1nnn[nH]1 CHEMBL3937915 IC50 39.0 nM
O=C(c1ccc(C(=O)C2(c3ccccc3)CC2)c(C(=O)O)c1)c1ccc(N(CC2CC2)c2ccc(Cl)cc2)cn1 CHEMBL3919389 IC50 41.0 nM
COc1ccc(C(=O)c2ccc(C(=O)c3ccc(N(CC4CC4)c4ccc(Cl)cc4F)cn3)cc2C(=O)O)cc1 CHEMBL3961231 IC50 46.0 nM
COc1cc(N(CC2CC2)c2cccc3ccccc23)ccc1C(=O)C1CC1C(=O)O CHEMBL3983776 IC50 46.0 nM
COc1cc(N(CC2(C)CC2)c2ccc3c(c2)CCC3)cnc1C(=O)C1CC1C(=O)O CHEMBL3936884 IC50 47.0 nM
COc1ccc(C(=O)c2ccc(C(=O)c3ccc(N(C)c4ccc(Cl)cc4)cn3)cc2C(=O)O)cc1 CHEMBL3909369 IC50 50.0 nM
COc1nc(C(=O)C2CC2C(=O)O)ncc1N(CC1CC1)c1cccc2ccccc12 CHEMBL3916445 IC50 50.0 nM
COc1cc(N(Cc2ccc(C(F)(F)F)cc2F)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3930479 IC50 53.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3cccc(C(F)(F)F)c3)c(C(=O)O)c2)nc1 CHEMBL3932466 IC50 54.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C(C)(C)c3ccccc3)c(C(=O)O)c2)nc1 CHEMBL3920701 IC50 55.0 nM
COc1cc(N(CC2CC2)c2ccc(C)c3ccccc23)ncc1C(=O)C1CC1C(=O)O CHEMBL3975465 IC50 56.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)CCC3CCCCC3)c(C(=O)O)c2)nc1 CHEMBL3961385 IC50 59.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3cccc(OC(F)(F)F)c3)c(C(=O)O)c2)nc1 CHEMBL3953130 IC50 60.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)c3ccccc23)ccc1C(=O)C1CC1C(=O)O CHEMBL3917485 IC50 61.0 nM
COc1cc(N(CC2CC2)c2ccc(C)c3ccccc23)ccc1C(=O)C1CC1C(=O)O CHEMBL3908538 IC50 62.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C34CC5CC(CC(C5)C3)C4)c(C(=O)O)c2)nc1 CHEMBL3951613 IC50 65.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)cc2)ccc1C(=O)C1CC1C(=O)O CHEMBL3922937 IC50 65.0 nM
COc1cc(N(Cc2cccc3ccccc23)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3935671 IC50 66.0 nM
COc1cc(N(Cc2cccc(C)c2C)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3898699 IC50 67.0 nM
COc1ccc(C(=O)c2ccc(C(=O)c3ccc(N(C)c4ccc(Cl)cc4)cn3)cc2C(=O)O)c(OC)c1 CHEMBL3983499 IC50 68.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)cc2)cnc1C(=O)C1CC1C(=O)NS(=O)(=O)c1ccccc1 CHEMBL3928255 IC50 68.0 nM
COc1cc(N(Cc2ccc(Cl)cc2)CC2CC2)ccc1C(=O)C1CC1C(=O)O CHEMBL3959510 IC50 68.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)cc2)cnc1C(=O)C1CC1C(=O)NS(=O)(=O)c1ccccc1F CHEMBL3942668 IC50 74.0 nM
COc1cc(N(CC2CC2)c2ccc(C)c(C)c2)ccc1C(=O)C1CC1C(=O)O CHEMBL3894959 IC50 75.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C3(c4ccccc4)CCCC3)c(C(=O)O)c2)nc1 CHEMBL3918897 IC50 76.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3ccc4c(c3)OCO4)c(C(=O)O)c2)nc1 CHEMBL3949468 IC50 77.0 nM
CCOc1ccc(C(=O)c2ccc(C(=O)c3ccc(N(C)c4ccc(Cl)cc4)cn3)cc2C(=O)O)cc1OCC CHEMBL3964233 IC50 77.0 nM
CN(c1ccc(C(F)(F)F)cc1)c1ccc(C(=O)c2ccc(C(=O)c3ccccc3)c(C(=O)O)c2)nc1 CHEMBL3899516 IC50 78.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)CC3CCCC3)c(C(=O)O)c2)nc1 CHEMBL3969203 IC50 81.0 nM
COc1ccc(S(=O)(=O)NC(=O)C2CC2C(=O)c2ncc(N(CC3CC3)c3ccc(Cl)cc3)cc2OC)cc1 CHEMBL3977284 IC50 81.0 nM
COc1cc(N(Cc2cccc(C(F)(F)F)c2C)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3952747 IC50 88.0 nM
CCCCCCC(=O)c1ccc(C(=O)c2ccc(N(C)c3ccc(Cl)cc3)cn2)cc1C(=O)O CHEMBL3891539 IC50 90.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C3CC4CCC3C4)c(C(=O)O)c2)nc1 CHEMBL3904404 IC50 94.0 nM
COc1cc(N(CC2CC2)c2cccc3ccccc23)cnc1C(=O)C1CC1c1nnn[nH]1 CHEMBL3953106 IC50 96.0 nM
CCOc1ccc(C(=O)c2ccc(C(=O)c3ccc(N(C)c4ccc(Cl)cc4)cn3)cc2C(=O)O)cc1 CHEMBL3981047 IC50 101.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3cccs3)c(C(=O)O)c2)nc1 CHEMBL3926899 IC50 104.0 nM
COc1cc(N(Cc2ccc(F)cc2)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3925042 IC50 105.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)c3ccccc23)cnc1C(=O)CCCC(=O)O CHEMBL4565235 IC50 109.0 nM
COc1cc(N(Cc2cccc(C(F)(F)F)c2Cl)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3961421 IC50 112.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3ccc(F)cc3)c(C(=O)O)c2)nc1 CHEMBL3950817 IC50 126.0 nM
CCC(=O)c1ccc(C(=O)c2ccc(N(CC3CC3)c3ccc(Cl)cc3)cn2)cc1C(=O)O CHEMBL3963802 IC50 129.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C3CC3c3ccccc3)c(C(=O)O)c2)nc1 CHEMBL3951511 IC50 141.0 nM
COc1cc(N(c2ccc(Cl)cc2)C(C2CC2)C(F)(F)F)cnc1C(=O)C1CC1C(=O)O CHEMBL3899164 IC50 149.0 nM
COc1cc(N(Cc2ccc(F)c(Cl)c2F)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3925717 IC50 152.0 nM
COc1cc(N(CC2CC2)c2ccc(C(F)(F)F)c3cccnc23)ccc1C(=O)C1CC1C(=O)O CHEMBL3973922 IC50 152.0 nM
COc1ccccc1C(=O)c1ccc(C(=O)c2ccc(N(C)c3ccc(Cl)cc3)cn2)cc1C(=O)O CHEMBL3923753 IC50 154.0 nM
COc1cc(N(CC2CC2)c2ccccc2)cnc1C(=O)[C@H]1C[C@@H]1C(=O)O CHEMBL4440339 IC50 158.0 nM
COc1cc(N(Cc2cccc(C)c2)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3939467 IC50 171.0 nM
CCc1ccc(N(C)c2ccc(C(=O)c3ccc(C(=O)c4ccccc4)c(C(=O)O)c3)nc2)cc1 CHEMBL3946767 IC50 184.0 nM
COc1cc(N(Cc2ccc(C)c(F)c2F)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3970803 IC50 185.0 nM
COc1cccc(CC(=O)c2ccc(C(=O)c3ccc(N(C)c4ccc(Cl)cc4)cn3)cc2C(=O)O)c1 CHEMBL3954606 IC50 192.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3ccc([N+](=O)[O-])cc3)c(C(=O)O)c2)nc1 CHEMBL3962261 IC50 202.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3ccc(C(F)(F)F)cc3)c(C(=O)O)c2)nc1 CHEMBL3955107 IC50 216.0 nM
COc1cc(N(CC2CC2)c2ccc(C(F)(F)F)c3cccnc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3977331 IC50 229.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)CC(C)(C)C)c(C(=O)O)c2)nc1 CHEMBL3966445 IC50 235.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)c3ccccc3C(F)(F)F)c(C(=O)O)c2)nc1 CHEMBL3954515 IC50 245.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C3CCCCC3)c(C(=O)O)c2)nc1 CHEMBL3986600 IC50 246.0 nM
Cc1ccc(N(C)c2ccc(C(=O)c3ccc(C(=O)c4ccccc4)c(C(=O)O)c3)nc2)cc1 CHEMBL3908334 IC50 250.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)Cc3ccccc3)c(C(=O)O)c2)nc1 CHEMBL3941304 IC50 257.0 nM
COCC(C1CC1)N(c1ccc(Cl)cc1)c1cnc(C(=O)C2CC2C(=O)O)c(OC)c1 CHEMBL3923713 IC50 263.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)cc2)cnc1C(=O)C1CC1C(=O)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 CHEMBL3915672 IC50 277.0 nM
COc1cc(N(CC2CC2)c2ccc(C)c3ncccc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3942345 IC50 279.0 nM
CC(=O)c1ccc(C(=O)c2ccc(N(CC3CC3)c3ccc(Cl)cc3)cn2)cc1C(=O)O CHEMBL3957224 IC50 307.0 nM
COc1cc(N(Cc2cccc(C(F)(F)F)c2F)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3941165 IC50 331.0 nM
COc1cc(N(CC2CC2)c2ccc(Cl)cc2)cnc1C(=O)C1CC1C(=O)NS(=O)(=O)C1CC1 CHEMBL3952482 IC50 356.0 nM
COc1cc(N(CC2CC2)c2ccc(C)c3ncccc23)ccc1C(=O)C1CC1C(=O)O CHEMBL3935516 IC50 359.0 nM
COc1cc(N(Cc2ccc(F)c(F)c2F)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3949929 IC50 370.0 nM
CC(c1ccc(Oc2ccccc2)cc1)c1nc2cc(-c3n[nH]c(=S)o3)ccc2[nH]1 CHEMBL5190547 IC50 400.0 nM
COc1ccc(C(=O)c2ccc(C(=O)c3ccc(N(CC(F)(F)F)c4ccc(Cl)cc4F)cn3)cc2C(=O)O)cc1 CHEMBL3921041 IC50 401.0 nM
O=C(c1ccc(C(=O)C2CC2)c(C(=O)O)c1)c1ccc(N(CC2CC2)c2ccc(Cl)cc2)cn1 CHEMBL3952925 IC50 424.0 nM
O=C(O)C1CC1C(=O)c1ccc(N(CC2CC2)c2ccc(Cl)cc2)cn1 CHEMBL3944475 IC50 424.0 nM
Cc1cc(Cl)ccc1N(C)c1ccc(C(=O)c2ccc(C(=O)c3ccccc3)c(C(=O)O)c2)nc1 CHEMBL3911656 IC50 442.0 nM
COc1cc(N(CC2CC2)c2cccc3c(C)ccnc23)cnc1C(=O)C1CC1C(=O)O CHEMBL3947697 IC50 445.0 nM
COc1cc(N(Cc2cc(F)cc3c2OCOC3)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3964542 IC50 478.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C(C)(C)C)c(C(=O)O)c2)nc1 CHEMBL3905951 IC50 491.0 nM
COc1cc(N(Cc2cc(Cl)cc3c2OCO3)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3926733 IC50 588.0 nM
O=C(O)C1CC1C(=O)c1ccc(N(Cc2ccc(Cl)cc2)CC2CC2)cn1 CHEMBL3911029 IC50 636.0 nM
S=c1[nH]nc(-c2ccc3[nH]c(-c4ccc(OCc5ccccc5)cc4)nc3c2)o1 CHEMBL5187474 IC50 700.0 nM
COc1cc(N(Cc2c(Cl)cccc2Cl)CC2CC2)cnc1C(=O)C1CC1C(=O)O CHEMBL3969030 IC50 800.0 nM
CN(c1ccc(Cl)cc1)c1ccc(C(=O)c2ccc(C(=O)C3CCCO3)c(C(=O)O)c2)nc1 CHEMBL3985155 IC50 860.0 nM