COc1cccc(Nc2[nH]nc(-c3ccc(NS(=O)(=O)C(F)F)cc3)c2C(N)=O)c1 CHEMBL5421128 Kd 0.7 nM
CC(C)S(=O)(=O)Nc1ccc(-c2n[nH]c(Nc3ccccc3)c2C(N)=O)cc1 CHEMBL5396374 Kd 150.0 nM
C[C@@H](Oc1cc(-c2cnn(C3CCNCC3)c2)cnc1N)c1c(Cl)ccc(F)c1Cl CHEMBL601719 Kd 217.0 nM
Nc1nccnc1C(=O)O[C@@H](C(=O)Nc1ccc(F)cc1)c1ccccc1 CHEMBL4440337 Kd 230.0 nM
CN(c1ccc(NC(=O)Nc2ccc(OC(F)(F)F)cc2)cc1)c1ccnc(Nc2cccc(S(N)(=O)=O)c2)n1 CHEMBL188381 Kd 530.0 nM
CN1C(=O)[C@@H](N2CCc3cn(Cc4ccccc4)nc3C2=O)COc2ccccc21 CHEMBL4088216 pIC50 1000.0 nM
CN1C(=O)[C@@H](N2CCc3c(nn(Cc4ccccc4)c3Br)C2=O)COc2ccccc21 CHEMBL4549667 pIC50 1000.0 nM
CN1C(=O)[C@@H](N2CCc3cn(CC4CCS(=O)(=O)CC4)nc3C2=O)COc2ccccc21 CHEMBL4097778 pIC50 1000.0 nM
