N#CC1=C(N)Oc2c(ccc3ccccc23)C1c1cccc([N+](=O)[O-])c1 CHEMBL321336 IC50 8.7 nM
COc1cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc(OC)c1OC CHEMBL228363 IC50 9.1 nM
C#CCOc1c(OC)cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL5188413 IC50 11.0 nM
CCOc1c(OC)cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL5184353 IC50 14.0 nM
C=CCOc1c(OC)cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL5198083 IC50 14.0 nM
N#CC1=C(N)Oc2c(ccc3ccccc23)C1c1ccc(Cl)c(F)c1 CHEMBL4442805 IC50 16.0 nM
CCCOc1c(OC)cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL5176963 IC50 30.0 nM
CCCCOc1c(OC)cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL5176572 IC50 30.0 nM
CCOc1c(Br)cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL5198730 IC50 36.8 nM
COc1ccc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL591374 IC50 40.0 nM
CCOc1c(I)cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL5192004 IC50 50.0 nM
COc1cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc(OC)c1OC(C)C CHEMBL5203253 IC50 60.0 nM
N#CC1=C(N)Oc2c(ccc3ccccc23)C1c1cc(F)c(F)c(F)c1 CHEMBL5192001 IC50 70.0 nM
COc1ccc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1[N+](=O)[O-] CHEMBL5173047 IC50 110.0 nM
N#CC1=C(N)Oc2c(ccc3ccccc23)C1c1cccc(S(F)(F)(F)(F)F)c1 CHEMBL4436683 IC50 130.0 nM
COc1cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)c(Br)c(OC)c1OC CHEMBL5194887 IC50 130.0 nM
CSc1ccc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1 CHEMBL4441682 IC50 210.0 nM
CSc1ccc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1F CHEMBL5187002 IC50 240.0 nM
N#CC1=C(N)Oc2c(ccc3ccccc23)C1c1ccc(C#N)cc1 CHEMBL4567907 IC50 390.0 nM
COc1ccc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1C CHEMBL5188662 IC50 400.0 nM
CCCCCOc1c(OC)cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1OC CHEMBL5179347 IC50 400.0 nM
COc1ccc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1Br CHEMBL5203497 IC50 420.0 nM
Cc1ccc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)cc1 CHEMBL4513667 IC50 430.0 nM
COc1cc(C2C(C#N)=C(N)Oc3c2ccc2ccccc32)ccc1OCc1ccccc1 CHEMBL4585739 IC50 1000.0 nM