O=C(NCC1CC1)c1cc(N2CC[C@H](O)C2)nc(N2CCC[C@@H](c3ccccc3)C2)n1 CHEMBL4794048 pIC50 72.44 nM
O=C(NCC1CC1)c1cc(N2CC[C@@H](O)C2)nc(N2CCC[C@@H](c3ccccc3)C2)n1 CHEMBL4761882 pIC50 109.65 nM
CN(C)c1cc(C(=O)NCC2CC2)nc(N2CCC[C@@H](c3ccccc3)C2)n1 CHEMBL4782800 pIC50 112.2 nM
CN(CCc1ccccc1)c1cc(C(=O)NCC2CC2)nc(N(C)CCc2ccccc2)n1 CHEMBL4752937 pIC50 154.88 nM
O=C(NCC1CC1)c1cc(N2CCOCC2)nc(N2CCC[C@@H](c3ccccc3)C2)n1 CHEMBL4754918 pIC50 208.93 nM
CN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCCC2)n1 CHEMBL4751223 pIC50 223.87 nM
CN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCC(O)C2)n1 CHEMBL4783103 pIC50 223.87 nM
CN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CC[C@H](O)C2)n1 CHEMBL4759968 pIC50 234.42 nM
O=C(NCC1CC1)c1cc(N2CC[C@H](O)C2)nc(N2CCC[C@H](c3ccccc3)C2)n1 CHEMBL4760293 pIC50 251.19 nM
CC(C)N(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCOCC2)n1 CHEMBL4752023 pIC50 281.84 nM
CN(C)c1cc(C(=O)NCC2CC2)nc(N(C)CCc2ccccc2)n1 CHEMBL4747615 pIC50 288.4 nM
CN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CC[C@@H](O)C2)n1 CHEMBL4764910 pIC50 302.0 nM
O=C(NCC1CC1)c1cc(N2CC[C@@H](O)C2)nc(N2CCC[C@H](c3ccccc3)C2)n1 CHEMBL4750592 pIC50 323.59 nM
O=C(NCC1CC1)c1cc(N2CCOCC2)nc(N2CCCC(c3ccccc3)C2)n1 CHEMBL4760794 pIC50 380.19 nM
O=C(NCC1CC1)c1cc(N2CCOCC2)nc(N2CCCC2Cc2ccccc2)n1 CHEMBL4752088 pIC50 380.19 nM
CN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCCC(F)(F)C2)n1 CHEMBL4746912 pIC50 389.05 nM
CN(C)c1cc(C(=O)NCC2CC2)nc(N2CCC[C@H](c3ccccc3)C2)n1 CHEMBL4750134 pIC50 407.38 nM
CN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCC2)n1 CHEMBL4795010 pIC50 426.58 nM
CN(CCc1ccccc1-c1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCOCC2)n1 CHEMBL4764783 pIC50 489.78 nM
CCN(CC)c1cc(C(=O)NCC2CC2)nc(N(C)CCc2ccccc2)n1 CHEMBL4787774 pIC50 501.19 nM
O=C(NCC1CC1)c1cc(N2CCOCC2)nc(N(CCc2ccccc2)CCc2ccccc2)n1 CHEMBL4743071 pIC50 524.81 nM
CN(CCc1ccccc1Oc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCOCC2)n1 CHEMBL4750396 pIC50 602.56 nM
CCN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCOCC2)n1 CHEMBL4756143 pIC50 645.65 nM
CN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCCCC2)n1 CHEMBL4741598 pIC50 645.65 nM
COC1CCN(c2cc(C(=O)NCC3CC3)nc(N(C)CCc3ccccc3)n2)C1 CHEMBL4792394 pIC50 707.95 nM
O=C(NCC1CC1)c1cc(N2CCOCC2)nc(N(CCc2ccccc2)Cc2ccccc2)n1 CHEMBL4764562 pIC50 741.31 nM
O=C(NCC1CC1)c1cc(N2CCOCC2)nc(N2CCCCC2Cc2ccccc2)n1 CHEMBL4787757 pIC50 741.31 nM
COc1ccccc1CCN(C)c1nc(C(=O)NCC2CC2)cc(N2CCOCC2)n1 CHEMBL4795013 pIC50 776.25 nM
CN(CCc1ccccc1)c1nc(C(=O)NCC2CC2)cc(N2CCOCC2)n1 CHEMBL4790197 pIC50 812.83 nM
COC(=O)CNC(=O)c1cc(N2CCOCC2)nc(N(C)CCc2ccccc2)n1 CHEMBL4747267 pIC50 831.76 nM
CNc1cc(C(=O)NCC2CC2)nc(N(C)CCc2ccccc2)n1 CHEMBL4762577 pIC50 851.14 nM
Cc1ccccc1CCN(C)c1nc(C(=O)NCC2CC2)cc(N2CCOCC2)n1 CHEMBL4789858 pIC50 891.25 nM
C#CCNC(=O)c1cc(N2CCOCC2)nc(N(C)CCc2ccccc2)n1 CHEMBL4795197 pIC50 912.01 nM
CN(CCc1ccccc1Cl)c1nc(C(=O)NCC2CC2)cc(N2CCOCC2)n1 CHEMBL4745098 pIC50 977.24 nM
O=C(NCC1CC1)c1cc(N2CCOCC2)nc(N2CCN(Cc3ccccc3)C(c3ccccc3)C2)n1 CHEMBL4764089 pIC50 1000.0 nM
CN(CCO)c1cc(C(=O)NCC2CC2)nc(N(C)CCc2ccccc2)n1 CHEMBL4777828 pIC50 1000.0 nM