Cc1nn(C)c(C)c1NS(=O)(=O)c1c(Cl)cc(-c2ccnc(N3CCNCC3)c2)cc1Cl CHEMBL1230468 IC50 3.0 nM
CCOC(=O)c1cnc2ccc(OCc3ccc(N4CCNCC4)nc3)cc2c1SCC CHEMBL4172452 Ki(app) 100.0 nM
CCOC(=O)c1cnc2ccc(OCc3ccc(NCCCN)nc3)cc2c1SCC CHEMBL4176755 Ki(app) 100.0 nM
CCOC(=O)c1cnc2ccc(OCc3ccc(N[C@@H]4CCNC4)nc3)cc2c1SCC CHEMBL4173973 Ki(app) 370.0 nM
CCOC(=O)c1cnc2ccc(OCc3ccc(NCCN)nc3)cc2c1SCC CHEMBL4168895 Ki(app) 410.0 nM
CCSc1c(C(=O)N2CCOCC2)cnc2ccc(OCc3ccccc3)cc12 CHEMBL4161807 Ki(app) 590.0 nM
CCOC(=O)c1cnc2ccc(OCc3ccc(NC4CCNCC4)nc3)cc2c1SCC CHEMBL4163264 Ki(app) 690.0 nM
