CCCS(=O)(=O)Nc1cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)cc(OC)c1OC CHEMBL4781373 IC50 1.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(CC(C)C)c3n2)cc1 CHEMBL4847211 IC50 3.0 nM
CC(C)(C)S(=O)(=O)c1cc2c(Nc3ccc4scnc4c3)ncnc2cc1OCCO CHEMBL4514780 IC50 4.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4ccccc4Cl)c(=O)n(C)c3n2)cc1 CHEMBL4853179 IC50 4.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(OC(=O)CC23CC4CC(CC(C4)C2)C3)c(OC)c1)C(C)C)C(=O)OCC CHEMBL5180843 EC50 4.5 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4ccc(O)cc4)c(=O)n(C)c3n2)cc1 CHEMBL4870434 IC50 5.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(Cc4cccc(S(C)(=O)=O)c4)c3n2)cc1 CHEMBL4864576 IC50 5.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(Cc4ccccc4)c3n2)cc1 CHEMBL4858463 IC50 9.0 nM
Cc1ccc2oc(N=C(N)NC(=O)C(C)(C)C)nc2c1 CHEMBL1595790 EC50 10.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(CCOC)c3n2)cc1 CHEMBL4859716 IC50 13.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4ccccc4)c(=O)n(C)c3n2)cc1 CHEMBL136244 IC50 14.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4ccccc4)c(=O)n(CC)c3n2)cc1 CHEMBL136106 IC50 15.0 nM
CCCS(=O)(=O)Nc1cc(-c2cc(-c3cccc(N4CCNCC4)c3)cnc2N)cc(F)c1OC CHEMBL4799077 IC50 16.0 nM
CC(C)c1ccc(-c2nc3ccccc3s2)cc1 CHEMBL1351908 EC50 20.0 nM
Cn1c(=O)c(-c2ccccc2Cl)cc2cnc(Nc3cccc(S(C)(=O)=O)c3)nc21 CHEMBL4861488 IC50 20.0 nM
Cn1c(=O)c(-c2c(Cl)cccc2Cl)cc2cnc(Nc3cccc(S(C)(=O)=O)c3)nc21 CHEMBL4864600 IC50 22.0 nM
CCCS(=O)(=O)Nc1cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)cc(F)c1OC CHEMBL4789724 IC50 26.0 nM
O=C(Nc1ccc(OC(F)(F)F)cc1)c1ccc(CN2CCc3ccccc3C2)cc1 CHEMBL1713298 IC50 30.0 nM
CCCCCCCCCCCC(=O)Oc1ccc(/C=C/C(=O)NCC(=O)N[C@H](C(=O)N[C@H](CCC(=O)OCC)C(=O)OCC)C(C)C)cc1OC CHEMBL5070781 EC50 30.0 nM
CC(C)[C@H](NC(=O)CNC(=O)/C=C/c1cccc(-c2ccccc2)c1)C(=O)N[C@H](CCC(=O)OC1CCCC1)C(=O)OC1CCCC1 CHEMBL5187281 EC50 35.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)cc1 CHEMBL49120 IC50 37.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@@H]1C[C@H]1c1ccc(F)c(F)c1)C(C)C)C(=O)OCC CHEMBL5077049 EC50 39.0 nM
CC(C)(C)c1ccc(C(=O)O/N=C(\N)c2ccccn2)cc1 CHEMBL1468181 EC50 40.0 nM
COc1cc(/C=C/C(=O)NCC(=O)N[C@H](C(=O)N[C@H](CCC(=O)OC2CCCC2)C(=O)OC2CCCC2)C(C)C)ccc1O CHEMBL5079672 EC50 40.0 nM
COc1cc(/C=C/C(=O)NCC(=O)N[C@H](C(=O)N[C@H](CCC(=O)OC2CCCC2)C(=O)OC2CCCC2)C(C)C)ccc1OC(=O)CC12CC3CC(CC(C3)C1)C2 CHEMBL5203244 EC50 44.0 nM
CC(=O)N[C@@H]1[C@@H](O[C@H](C)C(=O)N[C@@H](C)C(=O)N[C@H](CCC(=O)O)C(N)=O)[C@H](O)[C@@H](CO)O[C@H]1O CHEMBL369794 EC50 46.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(O)c(OC)c1)C(C)C)C(=O)OCC CHEMBL4090558 EC50 46.0 nM
CCOc1cc(NS(=O)(=O)C(C)C)cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)c1 CHEMBL4795976 IC50 46.0 nM
CCCS(=O)(=O)Nc1cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)cc(Cl)c1OC CHEMBL4793153 IC50 46.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1cccc(-c2ccccc2)c1)C(C)C)C(=O)OCC CHEMBL5207301 EC50 47.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc([N+](=O)[O-])cc1)C(C)C)C(=O)OCC CHEMBL5086803 EC50 49.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)C1CC1c1ccc(F)c(F)c1)C(C)C)C(=O)OCC CHEMBL4069541 EC50 49.0 nM
COc1cc(NS(=O)(=O)c2ccccc2)cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)c1 CHEMBL4776631 IC50 53.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1cccc(Oc2ccccc2)c1)C(C)C)C(=O)OCC CHEMBL5193116 EC50 61.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(OC(C)=O)c(OC)c1)C(C)C)C(=O)OCC CHEMBL5085864 EC50 62.0 nM
COc1cc(/C=C/C(=O)NCC(=O)N[C@H](C(=O)N[C@H](CCC(=O)OC2CCCC2)C(=O)OC2CCCC2)C(C)C)ccc1OC(C)=O CHEMBL5077437 EC50 63.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H]1C[C@@H]1c1ccc(F)c(F)c1)C(C)C)C(=O)OCC CHEMBL5075343 EC50 66.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(C(C)C)cc1)C(C)C)C(=O)OCC CHEMBL5090188 EC50 71.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1cccc([N+](=O)[O-])c1)C(C)C)C(=O)OCC CHEMBL5192766 EC50 82.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(Cc4ccc(S(C)(=O)=O)cc4)c3n2)cc1 CHEMBL4874031 IC50 94.0 nM
COC(=O)Cc1nn(-c2nc3ccccc3s2)c(O)c1/C(C)=N/c1ccc(OC)cc1 CHEMBL3194944 EC50 100.0 nM
CCCCOc1nc(N)c2nc(O)n(Cc3ccc(C(=O)NCCCCCC(=O)Oc4ccc(/C=C/C(=O)NCC(=O)N[C@H](C(=O)N[C@H](CCC(=O)OCC)C(=O)OCC)C(C)C)cc4OC)cc3)c2n1 CHEMBL5178827 EC50 114.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)/C=C/c1ccc(O)c(OC)c1)C(=O)OCC CHEMBL4060406 EC50 121.0 nM
COc1cc(NS(=O)(=O)C(C)C)cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)c1 CHEMBL4781705 IC50 121.0 nM
CCCS(=O)(=O)Nc1cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)cc(C)c1OC CHEMBL4788375 IC50 129.0 nM
CC(C)[C@H](NC(=O)CNC(=O)/C=C/c1cccc(Oc2ccccc2)c1)C(=O)N[C@H](CCC(=O)OC1CCCC1)C(=O)OC1CCCC1 CHEMBL5184036 EC50 130.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1cccc(Br)c1)C(C)C)C(=O)OCC CHEMBL5182728 EC50 135.0 nM
Cn1c(=O)c(-c2c(Cl)cccc2Cl)cc2cnc(Nc3ccc(S(C)(=O)=O)cc3)nc21 CHEMBL4868894 IC50 136.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4ccc(Cl)cc4Cl)c(=O)n(C)c3n2)cc1 CHEMBL4849134 IC50 160.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(F)c(F)c1)C(C)C)C(=O)OCC CHEMBL4068530 EC50 172.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)/C=C/c1ccc(F)c(F)c1)C(=O)OCC CHEMBL4094910 EC50 172.0 nM
CC1Cc2cc(S(=O)(=O)N3CCN(c4ccc([N+](=O)[O-])cc4)CC3)ccc2N1C(=O)C1CC1 CHEMBL1732337 IC50 200.0 nM
CC(=O)N[C@H]1C(O)O[C@H](CO)[C@@H](O)[C@@H]1O[C@H](C)C(=O)N[C@@H](C)C(=O)N[C@H](CCC(=O)O)C(N)=O CHEMBL1779325 Kd 200.0 nM
Cn1c(=O)c(-c2ccc(F)cc2Cl)cc2cnc(Nc3cccc(S(C)(=O)=O)c3)nc21 CHEMBL4867716 IC50 218.0 nM
CC(C)COc1ccc(C(=O)Nc2sc3c(c2C(=O)O)CC(C)(C)OC3)cc1 CHEMBL1380661 EC50 220.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccccc1)C(C)C)C(=O)OCC CHEMBL4059862 EC50 223.0 nM
CCCS(=O)(=O)Nc1cc(OC)cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)c1 CHEMBL4800115 IC50 243.0 nM
CCCCCCCCCCCC(=O)Oc1ccc(/C=C/C(=O)NCC(=O)N[C@H](C(=O)N[C@H](CCC(=O)OC2CCCC2)C(=O)OC2CCCC2)C(C)C)cc1OC CHEMBL5073412 EC50 243.0 nM
CSc1ccc(NC(=O)c2ccc(CN3CCc4ccccc4C3)cc2)cc1 CHEMBL1704728 IC50 260.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4ccccc4)c(=O)n(CCO)c3n2)cc1 CHEMBL4871544 IC50 270.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)C1CC1c1ccc(F)c(F)c1)C(=O)OCC CHEMBL4088641 EC50 276.0 nM
COC(=O)c1ccc2nc(Nc3nc4c(F)cc(F)cc4s3)sc2c1 CHEMBL1480238 EC50 300.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1cc2cc(Br)ccc2o1)C(C)C)C(=O)OCC CHEMBL5176249 EC50 316.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)C1CC1c1ccc(OC)c(OC)c1)C(C)C)C(=O)OCC CHEMBL5079466 EC50 322.0 nM
CC(C)Oc1cc(NS(=O)(=O)C(C)C)cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)c1 CHEMBL4792496 IC50 323.0 nM
CCCS(=O)(=O)Nc1cc(-c2cncc(-c3ccc(N4CCNCC4)cc3)c2)cc(F)c1OC CHEMBL4782505 IC50 352.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)C1CC1c1ccc(O)c(OC)c1)C(C)C)C(=O)OCC CHEMBL5079980 EC50 369.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)/C=C/c1ccccc1)C(=O)OCC CHEMBL4098290 EC50 388.0 nM
COc1ccc(N2CCN(S(=O)(=O)c3ccc4c(c3)CC(C)N4C(=O)C3CC3)CC2)cc1 CHEMBL1450407 IC50 390.0 nM
COc1cc(NS(C)(=O)=O)cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)c1 CHEMBL4784430 IC50 390.0 nM
CCOC(=O)c1ccc(NC(=O)c2ccc(CN3CCc4ccccc4C3)cc2)cc1 CHEMBL1569174 IC50 400.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(C)cc1)C(C)C)C(=O)OCC CHEMBL5204917 EC50 402.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(Cl)cc1)C(C)C)C(=O)OCC CHEMBL5186060 EC50 412.0 nM
CN(C)c1cccc(Oc2cc3c(cc2NC(=O)COCc2ccc(C(F)(F)F)cc2)NC(=O)[C@@H](CCC(=O)N2CCC(F)CC2)NC3=O)c1 CHEMBL4097753 IC50 420.0 nM
CCCS(=O)(=O)Nc1cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)ccc1OC CHEMBL4786742 IC50 420.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@H](CCc1ccccc1)NC(=O)CNC(=O)/C=C/c1ccc(O)c(OC)c1)C(=O)OCC CHEMBL5180997 EC50 420.0 nM
Cc1cc(C(=O)COC(=O)c2ccccc2Br)c(C)n1CC1CCCO1 CHEMBL1597561 EC50 460.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)OCC CHEMBL4074427 EC50 472.0 nM
CCCCOC(=O)CC1c2cccc(C)c2S(=O)(=O)N1C(=O)c1ccccc1C(F)(F)F CHEMBL4792557 IC50 480.0 nM
Cc1ccc(-c2cc3cnc(Nc4cccc(S(C)(=O)=O)c4)nc3n(C)c2=O)c(Cl)c1 CHEMBL4875011 IC50 480.0 nM
Cc1ccc(-n2c(C)cc(/C=c3/sc4nc5ccccc5n4c3=O)c2C)cc1 CHEMBL3210725 EC50 490.0 nM
O=C(COCc1ccc(C(F)(F)F)cc1)Nc1cc2ncn(CC(=O)N3CCCC(F)(F)C3)c(=O)c2cc1Oc1cccc(N2CCOCC2)c1 CHEMBL4740438 IC50 500.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4ccc(OC)cc4)c(=O)n(C)c3n2)cc1 CHEMBL4852513 IC50 510.0 nM
COc1cc(NS(=O)(=O)C(C)C)cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2C)c1 CHEMBL4792227 IC50 523.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(Br)cc1)C(C)C)C(=O)OCC CHEMBL5176732 EC50 534.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(N)cc1)C(C)C)C(=O)OCC CHEMBL5082818 EC50 542.0 nM
COC(=O)Cn1cnc2cc(NC(=O)COCc3ccc(C(F)(F)F)cc3)c(Oc3cccc(N4CCOCC4)c3)cc2c1=O CHEMBL4753767 IC50 550.0 nM
Cc1cc(/C=C2\SC(=S)N(C)C2=O)c(C)n1-c1ccc(O)cc1 CHEMBL1507251 EC50 570.0 nM
CCOc1ccc(NC(=O)c2ccc(CN3CCc4ccccc4C3)cc2)cc1 CHEMBL1569954 IC50 570.0 nM
COC(=O)CC[C@@H]1NC(=O)c2cc(Oc3cccc(N(C)C)c3)c(NC(=O)COCc3ccc(C(F)(F)F)cc3)cc2NC1=O CHEMBL4065255 IC50 590.0 nM
COc1cc(-c2cc(-c3ccc(N4CCNCC4)cc3)cnc2N)cc(F)c1OC CHEMBL4781201 IC50 595.0 nM
CCC(=O)N1c2ccc(S(=O)(=O)N3CCN(c4ccc(Cl)cc4)CC3)cc2CC1C CHEMBL1709705 IC50 600.0 nM
Cn1nccc1C(=O)NC1CCCc2c1cnn2-c1ccccc1F CHEMBL1531328 EC50 610.0 nM
CN(CCc1nc2ccccc2n1CC(=O)Nc1ccc2c(c1)CCC2)S(=O)(=O)c1ccccc1 CHEMBL4778195 IC50 630.0 nM
CN(C)c1cccc(Oc2cc3c(=O)n(CC(=O)N4CCCC(F)(F)C4)cnc3cc2NC(=O)COCc2ccc(C(F)(F)F)cc2)c1 CHEMBL4749022 IC50 660.0 nM
Cc1oc(-c2ccccc2Cl)nc1CSc1nc(O)c2c(n1)CCCC2 CHEMBL1380813 EC50 730.0 nM
Cn1c(=O)c(-c2cc(Cl)ccc2Cl)cc2cnc(Nc3cccc(S(C)(=O)=O)c3)nc21 CHEMBL4853711 IC50 730.0 nM
Cn1c(=O)[nH]c(=O)c2c1nc([N+](=O)[O-])n2Cc1ccccc1 CHEMBL1419822 IC50 748.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1cc2cc([N+](=O)[O-])ccc2o1)C(C)C)C(=O)OCC CHEMBL5184105 EC50 760.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(OC)c(OC)c1)C(C)C)C(=O)OCC CHEMBL5084692 EC50 763.0 nM
O=C(NCCCOc1ccc(C(F)(F)F)cc1)c1cc2ncn(CC(=O)N3CCCC(F)(F)C3)c(=O)c2cc1-c1cccc(Cl)c1 CHEMBL4785218 IC50 770.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)c1cc2ccc(-c3ccccc3)cc2[nH]1)C(=O)OCC CHEMBL4080248 EC50 777.0 nM
CCCOc1ccc(/C=N/NC(=S)Nc2ccccc2[N+](=O)[O-])c(O)c1 CHEMBL3195322 EC50 780.0 nM
COc1ccc(NC(=O)c2ccc(CN3CCc4ccccc4C3)cc2)cc1 CHEMBL1700405 IC50 780.0 nM
CCOC(=O)CC[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)/C=C/c1ccc(OC(C)C)cc1)C(C)C)C(=O)OCC CHEMBL5208149 EC50 795.0 nM
CN(C)c1cccc(Oc2cc3c(=O)[nH]cnc3cc2NC(=O)COCc2ccc(C(F)(F)F)cc2)c1 CHEMBL4781741 IC50 800.0 nM
O=C(NCCCOc1ccc(C(F)(F)F)cc1)c1cc2ncn(CC(=O)N3CCCCC3)c(=O)c2cc1-c1cccc(Cl)c1 CHEMBL4747890 IC50 800.0 nM
CN(C)c1cccc(Oc2cc3c(cc2NC(=O)COCc2ccc(C(F)(F)F)cc2)NC(=O)[C@@H](CCC(=O)N2CCC(F)(F)CC2)NC3=O)c1 CHEMBL4076733 IC50 810.0 nM
O=C(NCCCOc1ccc(C(F)(F)F)cc1)c1cc2nc[nH]c(=O)c2cc1-c1cccc(Cl)c1 CHEMBL4750880 IC50 840.0 nM
COC(=O)CC[C@H]1NC(=O)c2cc(Oc3cccc(N(C)C)c3)c(NC(=O)COCc3ccc(C(F)(F)F)cc3)cc2NC1=O CHEMBL4087264 IC50 870.0 nM
Cn1c(=O)c(-c2ccc(Cl)cc2Cl)cc2cnc(Nc3cccc(S(C)(=O)=O)c3)nc21 CHEMBL4859351 IC50 878.0 nM
CN(C)c1cccc(Oc2cc3c(cc2NC(=O)COCc2ccc(Cl)cc2)NC(=O)[C@@H](CCC(=O)N2CCCCC2)NC3=O)c1 CHEMBL4089565 IC50 900.0 nM
CCCCOC(=O)CC1c2cccc(C)c2S(=O)(=O)N1C(=O)c1cccc(C(F)(F)F)c1 CHEMBL4784208 IC50 930.0 nM
C[C@@H]1NC(=O)c2cc(Oc3cccc(N(C)C)c3)c(NC(=O)COCc3ccc(C(F)(F)F)cc3)cc2NC1=O CHEMBL4080835 IC50 940.0 nM
O=C(CSc1nc(O)c2c(-c3ccccc3)csc2n1)Nc1ccccc1 CHEMBL1333821 EC50 950.0 nM
CCN(CC)CCOc1ccc(Nc2ncc3cc(-c4ccc(Cl)cc4)c(=O)n(C)c3n2)cc1 CHEMBL4852860 IC50 950.0 nM
COC(=O)Cn1cnc2cc(NC(=O)COCc3ccc(C(F)(F)F)cc3)c(Oc3cccc(N(C)C)c3)cc2c1=O CHEMBL4794272 IC50 990.0 nM
COC(=O)Cn1cnc2cc(C(=O)NCCCOc3ccc(C(F)(F)F)cc3)c(-c3cccc(Cl)c3)cc2c1=O CHEMBL4742329 IC50 1000.0 nM